KR20170033321A - 아졸벤젠 유도체의 결정 - Google Patents
아졸벤젠 유도체의 결정 Download PDFInfo
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- KR20170033321A KR20170033321A KR1020177002444A KR20177002444A KR20170033321A KR 20170033321 A KR20170033321 A KR 20170033321A KR 1020177002444 A KR1020177002444 A KR 1020177002444A KR 20177002444 A KR20177002444 A KR 20177002444A KR 20170033321 A KR20170033321 A KR 20170033321A
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- South Korea
- Prior art keywords
- crystal
- activity
- thiazole
- acid
- compound
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Images
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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- A—HUMAN NECESSITIES
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| JP2014155031 | 2014-07-30 | ||
| JPJP-P-2014-155031 | 2014-07-30 | ||
| PCT/JP2015/071512 WO2016017696A1 (fr) | 2014-07-30 | 2015-07-29 | Cristal de dérivé de benzène et d'azole |
Publications (1)
| Publication Number | Publication Date |
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| KR20170033321A true KR20170033321A (ko) | 2017-03-24 |
Family
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| KR1020177002444A KR20170033321A (ko) | 2014-07-30 | 2015-07-29 | 아졸벤젠 유도체의 결정 |
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| Country | Link |
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| EP (1) | EP3176165B1 (fr) |
| JP (1) | JP6230713B2 (fr) |
| KR (1) | KR20170033321A (fr) |
| CN (1) | CN106536519B (fr) |
| AR (1) | AR101363A1 (fr) |
| AU (1) | AU2015297489B2 (fr) |
| BR (1) | BR112017001659A2 (fr) |
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| CY (1) | CY1120933T1 (fr) |
| DK (1) | DK3176165T3 (fr) |
| ES (1) | ES2693382T3 (fr) |
| HR (1) | HRP20181789T1 (fr) |
| IL (1) | IL250144B (fr) |
| LT (1) | LT3176165T (fr) |
| MX (1) | MX370375B (fr) |
| MY (1) | MY179339A (fr) |
| NZ (1) | NZ729045A (fr) |
| PH (1) | PH12017500123A1 (fr) |
| PL (1) | PL3176165T3 (fr) |
| PT (1) | PT3176165T (fr) |
| RS (1) | RS57797B1 (fr) |
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| SA (1) | SA517380786B1 (fr) |
| SG (1) | SG11201700742UA (fr) |
| SI (1) | SI3176165T1 (fr) |
| TR (1) | TR201818775T4 (fr) |
| TW (1) | TWI687418B (fr) |
| WO (1) | WO2016017696A1 (fr) |
| ZA (1) | ZA201700491B (fr) |
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| GB201300552D0 (en) * | 2013-01-14 | 2013-02-27 | Moog Bv | Motion simulator |
| JP6134072B2 (ja) * | 2014-07-30 | 2017-05-24 | 帝人ファーマ株式会社 | キサンチンオキシダーゼ阻害薬 |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1992009279A1 (fr) | 1990-11-30 | 1992-06-11 | Teijin Limited | Derive de 2-arylthiazole et composition pharmaceutique contenant ce derive |
| WO1996031211A1 (fr) | 1995-04-07 | 1996-10-10 | Teijin Limited | Agent protecteur pour organe ou tissu |
| JP2002105067A (ja) | 2000-09-28 | 2002-04-10 | Teijin Ltd | ２−フェニルチアゾール誘導体、およびそれを有効成分とする医薬組成物 |
| WO2010018458A2 (fr) | 2008-08-12 | 2010-02-18 | Crystalgenomics, Inc. | Dérivés de phénol et leurs procédés d'utilisation |
| WO2010128163A2 (fr) | 2009-05-08 | 2010-11-11 | Pike Pharma Gmbh | Inhibiteurs à petite molécule du virus de la grippe a et b et de la réplication du virus respiratoire syncytial |
| WO2011101867A2 (fr) | 2010-02-19 | 2011-08-25 | Cadila Healthcare Limited | Sels essentiellement purs de fébuxostat et leurs procédés de préparation |
| WO2011139886A2 (fr) | 2010-04-29 | 2011-11-10 | Dr. Reddy's Laboratories Ltd. | Préparation of fébuxostat |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006514009A (ja) * | 2002-11-14 | 2006-04-27 | セルメド オンコロジー （ユーエスエイ）， インコーポレイテッド | ペプチドデホルミラーゼ活性化プロドラッグ |
| JPWO2007043401A1 (ja) * | 2005-10-07 | 2009-04-16 | キッセイ薬品工業株式会社 | 含窒素複素環化合物およびそれを含有する医薬組成物 |
| WO2008126770A1 (fr) * | 2007-04-05 | 2008-10-23 | Astellas Pharma Inc. | Procédé de production d'un dérivé d'acide triarylcarboxylique |
| JP5378988B2 (ja) | 2007-04-11 | 2013-12-25 | キッセイ薬品工業株式会社 | ５員環へテロ環誘導体及びその医薬用途 |
| TWI606048B (zh) * | 2013-01-31 | 2017-11-21 | 帝人製藥股份有限公司 | 唑苯衍生物 |
-
2015
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- 2015-07-29 AU AU2015297489A patent/AU2015297489B2/en not_active Ceased
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- 2015-07-29 SI SI201530420T patent/SI3176165T1/sl unknown
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- 2015-07-29 CA CA2955485A patent/CA2955485A1/fr not_active Abandoned
- 2015-07-29 TW TW104124555A patent/TWI687418B/zh not_active IP Right Cessation
- 2015-07-29 EP EP15827012.4A patent/EP3176165B1/fr active Active
- 2015-07-29 PT PT15827012T patent/PT3176165T/pt unknown
- 2015-07-29 WO PCT/JP2015/071512 patent/WO2016017696A1/fr active Application Filing
- 2015-07-29 LT LTEP15827012.4T patent/LT3176165T/lt unknown
- 2015-07-29 JP JP2016538400A patent/JP6230713B2/ja not_active Expired - Fee Related
- 2015-07-29 TR TR2018/18775T patent/TR201818775T4/tr unknown
- 2015-07-29 PL PL15827012T patent/PL3176165T3/pl unknown
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- 2015-07-29 RU RU2017106058A patent/RU2675854C2/ru active
- 2015-07-29 BR BR112017001659-1A patent/BR112017001659A2/pt active Search and Examination
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- 2015-07-29 CN CN201580040558.5A patent/CN106536519B/zh not_active Expired - Fee Related
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2017
- 2017-01-16 IL IL25014417A patent/IL250144B/en active IP Right Grant
- 2017-01-20 ZA ZA2017/00491A patent/ZA201700491B/en unknown
- 2017-01-20 PH PH12017500123A patent/PH12017500123A1/en unknown
- 2017-01-24 SA SA517380786A patent/SA517380786B1/ar unknown
-
2018
- 2018-10-30 HR HRP20181789TT patent/HRP20181789T1/hr unknown
- 2018-11-29 CY CY181101270T patent/CY1120933T1/el unknown
Patent Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1992009279A1 (fr) | 1990-11-30 | 1992-06-11 | Teijin Limited | Derive de 2-arylthiazole et composition pharmaceutique contenant ce derive |
| WO1996031211A1 (fr) | 1995-04-07 | 1996-10-10 | Teijin Limited | Agent protecteur pour organe ou tissu |
| JP2002105067A (ja) | 2000-09-28 | 2002-04-10 | Teijin Ltd | ２−フェニルチアゾール誘導体、およびそれを有効成分とする医薬組成物 |
| WO2010018458A2 (fr) | 2008-08-12 | 2010-02-18 | Crystalgenomics, Inc. | Dérivés de phénol et leurs procédés d'utilisation |
| WO2010128163A2 (fr) | 2009-05-08 | 2010-11-11 | Pike Pharma Gmbh | Inhibiteurs à petite molécule du virus de la grippe a et b et de la réplication du virus respiratoire syncytial |
| WO2011101867A2 (fr) | 2010-02-19 | 2011-08-25 | Cadila Healthcare Limited | Sels essentiellement purs de fébuxostat et leurs procédés de préparation |
| WO2011139886A2 (fr) | 2010-04-29 | 2011-11-10 | Dr. Reddy's Laboratories Ltd. | Préparation of fébuxostat |
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