KR20140072177A - 헤테로사이클릴피리(미)디닐피라졸 - Google Patents

헤테로사이클릴피리(미)디닐피라졸 Download PDF

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Publication number
KR20140072177A
KR20140072177A KR1020147011919A KR20147011919A KR20140072177A KR 20140072177 A KR20140072177 A KR 20140072177A KR 1020147011919 A KR1020147011919 A KR 1020147011919A KR 20147011919 A KR20147011919 A KR 20147011919A KR 20140072177 A KR20140072177 A KR 20140072177A
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KR
South Korea
Prior art keywords
alkyl
group
butyl
cycloalkyl
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
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KR1020147011919A
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English (en)
Korean (ko)
Inventor
알렉산더 수다우
헨드릭 헬름케
스테판 힐레브란트
아모스 마테스
라르스 로드펠트
피에르 바스나이레
위르겐 벤팅
페터 다멘
울리케 바헨도르프-노이만
필리프 데스보르데스
앤-소피 레브스톡
Original Assignee
바이엘 인텔렉쳐 프로퍼티 게엠베하
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 바이엘 인텔렉쳐 프로퍼티 게엠베하 filed Critical 바이엘 인텔렉쳐 프로퍼티 게엠베하
Publication of KR20140072177A publication Critical patent/KR20140072177A/ko
Ceased legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/052Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020147011919A 2011-10-06 2012-10-04 헤테로사이클릴피리(미)디닐피라졸 Ceased KR20140072177A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11184138.3 2011-10-06
EP11184138 2011-10-06
PCT/EP2012/069557 WO2013050434A1 (en) 2011-10-06 2012-10-04 Heterocyclylpyri(mi)dinylpyrazole

Publications (1)

Publication Number Publication Date
KR20140072177A true KR20140072177A (ko) 2014-06-12

Family

ID=46968225

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020147011919A Ceased KR20140072177A (ko) 2011-10-06 2012-10-04 헤테로사이클릴피리(미)디닐피라졸

Country Status (18)

Country Link
US (1) US9314026B2 (enExample)
EP (1) EP2763993B1 (enExample)
JP (1) JP6211522B2 (enExample)
KR (1) KR20140072177A (enExample)
CN (1) CN103958518B (enExample)
AU (1) AU2012320578B2 (enExample)
BR (1) BR112014008222A2 (enExample)
CL (1) CL2014000807A1 (enExample)
CO (1) CO6920305A2 (enExample)
DK (1) DK2763993T3 (enExample)
ES (1) ES2632584T3 (enExample)
IN (1) IN2014CN02475A (enExample)
MX (1) MX351460B (enExample)
PL (1) PL2763993T3 (enExample)
RU (1) RU2627272C2 (enExample)
UA (1) UA114410C2 (enExample)
WO (1) WO2013050434A1 (enExample)
ZA (1) ZA201403228B (enExample)

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CN111107902A (zh) * 2017-03-14 2020-05-05 丹娜法伯癌症研究所 Bax活化的用于诱导细胞死亡的小分子致敏
WO2021227906A1 (zh) * 2020-05-12 2021-11-18 苏州阿尔脉生物科技有限公司 一种作为cdk抑制剂的吡啶乙酰胺类衍生物、其制备方法及用途

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Also Published As

Publication number Publication date
CO6920305A2 (es) 2014-04-10
DK2763993T3 (en) 2017-07-24
IN2014CN02475A (enExample) 2015-06-19
PL2763993T3 (pl) 2017-09-29
RU2627272C2 (ru) 2017-08-04
NZ622704A (en) 2016-05-27
AU2012320578B2 (en) 2017-03-02
ZA201403228B (en) 2017-08-30
JP2014528961A (ja) 2014-10-30
AU2012320578A1 (en) 2014-04-10
JP6211522B2 (ja) 2017-10-11
ES2632584T3 (es) 2017-09-14
WO2013050434A1 (en) 2013-04-11
US20140364456A1 (en) 2014-12-11
CN103958518B (zh) 2017-07-04
CN103958518A (zh) 2014-07-30
BR112014008222A2 (pt) 2017-04-25
UA114410C2 (uk) 2017-06-12
MX2014003918A (es) 2014-04-25
US9314026B2 (en) 2016-04-19
CL2014000807A1 (es) 2014-09-05
RU2014117822A (ru) 2015-11-20
MX351460B (es) 2017-10-16
EP2763993A1 (en) 2014-08-13
EP2763993B1 (en) 2017-04-19

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