AU2012320578B2 - Heterocyclylpyri(mi)dinylpyrazole - Google Patents

Heterocyclylpyri(mi)dinylpyrazole Download PDF

Info

Publication number
AU2012320578B2
AU2012320578B2 AU2012320578A AU2012320578A AU2012320578B2 AU 2012320578 B2 AU2012320578 B2 AU 2012320578B2 AU 2012320578 A AU2012320578 A AU 2012320578A AU 2012320578 A AU2012320578 A AU 2012320578A AU 2012320578 B2 AU2012320578 B2 AU 2012320578B2
Authority
AU
Australia
Prior art keywords
plants
compounds
formula
methyl
species
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2012320578A
Other languages
English (en)
Other versions
AU2012320578A1 (en
Inventor
Jurgen Benting
Peter Dahmen
Philippe Desbordes
Hendrik Helmke
Stefan Hillebrand
Amos Mattes
Anne-Sophie Rebstock
Lars Rodefeld
Alexander Sudau
Ulrike Wachendorff-Neumann
Pierre Wasnaire
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Intellectual Property GmbH
Original Assignee
Bayer Intellectual Property GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Intellectual Property GmbH filed Critical Bayer Intellectual Property GmbH
Publication of AU2012320578A1 publication Critical patent/AU2012320578A1/en
Application granted granted Critical
Publication of AU2012320578B2 publication Critical patent/AU2012320578B2/en
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/052Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2012320578A 2011-10-06 2012-10-04 Heterocyclylpyri(mi)dinylpyrazole Ceased AU2012320578B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11184138 2011-10-06
EP11184138.3 2011-10-06
PCT/EP2012/069557 WO2013050434A1 (en) 2011-10-06 2012-10-04 Heterocyclylpyri(mi)dinylpyrazole

Publications (2)

Publication Number Publication Date
AU2012320578A1 AU2012320578A1 (en) 2014-04-10
AU2012320578B2 true AU2012320578B2 (en) 2017-03-02

Family

ID=46968225

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2012320578A Ceased AU2012320578B2 (en) 2011-10-06 2012-10-04 Heterocyclylpyri(mi)dinylpyrazole

Country Status (18)

Country Link
US (1) US9314026B2 (enExample)
EP (1) EP2763993B1 (enExample)
JP (1) JP6211522B2 (enExample)
KR (1) KR20140072177A (enExample)
CN (1) CN103958518B (enExample)
AU (1) AU2012320578B2 (enExample)
BR (1) BR112014008222A2 (enExample)
CL (1) CL2014000807A1 (enExample)
CO (1) CO6920305A2 (enExample)
DK (1) DK2763993T3 (enExample)
ES (1) ES2632584T3 (enExample)
IN (1) IN2014CN02475A (enExample)
MX (1) MX351460B (enExample)
PL (1) PL2763993T3 (enExample)
RU (1) RU2627272C2 (enExample)
UA (1) UA114410C2 (enExample)
WO (1) WO2013050434A1 (enExample)
ZA (1) ZA201403228B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112015012656B1 (pt) 2012-11-30 2021-12-21 Injekta Environmental Pty Ltd Composição de remediação do solo e estabilização de poros do solo e método de aprimoramento de uma estrutura do solo
PH12017502334B1 (en) * 2015-06-29 2023-05-26 Astrazeneca Ab Polycyclic amide derivative as cdk9 inhibitors
CA3054452A1 (en) * 2017-03-14 2018-09-20 Dana-Farber Cancer Institute, Inc. Small molecule sensitization of bax activation for induction of cell death
EP4140997A4 (en) * 2020-05-12 2023-09-06 Suzhou Alphama Biotechnology Co., Ltd. PYRIDINE ACETAMIDE DERIVATIVE AS CDK INHIBITOR, PREPARATION METHOD AND USE THEREOF

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009076440A2 (en) * 2007-12-12 2009-06-18 E.I. Du Pont De Nemours And Company Fungicidal bicyclic pyrazoles

Family Cites Families (59)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US18156A (en) 1857-09-08 Edward pate and saml
US4272417A (en) 1979-05-22 1981-06-09 Cargill, Incorporated Stable protective seed coating
US4245432A (en) 1979-07-25 1981-01-20 Eastman Kodak Company Seed coatings
US4808430A (en) 1987-02-27 1989-02-28 Yazaki Corporation Method of applying gel coating to plant seeds
GB8727737D0 (en) 1987-11-26 1987-12-31 Ici Plc Antitumour agents
GB8810120D0 (en) 1988-04-28 1988-06-02 Plant Genetic Systems Nv Transgenic nuclear male sterile plants
US5344992A (en) 1990-04-26 1994-09-06 Ciba-Geigy Corporation Process for the preparation of linear 1,3-diketones
US5559137A (en) 1994-05-16 1996-09-24 Smithkline Beecham Corp. Compounds
JP4469422B2 (ja) 1995-04-20 2010-05-26 アメリカン シアナミド コンパニー 構造に基づきデザインされた除草剤耐性生産物
US5876739A (en) 1996-06-13 1999-03-02 Novartis Ag Insecticidal seed coating
TR200000235T2 (tr) 1997-05-22 2000-05-22 G.D. Searle &Co. p38 kinaz inhibitörleri olarak ikame edilmiş pirazoller.
RU2249591C2 (ru) 1997-05-22 2005-04-10 Дж.Д. Серл Энд Ко. 3(5)-гетероарилзамещенные пиразолы в качестве ингибиторов киназы p38
US6514977B1 (en) 1997-05-22 2003-02-04 G.D. Searle & Company Substituted pyrazoles as p38 kinase inhibitors
US6503904B2 (en) 1998-11-16 2003-01-07 Syngenta Crop Protection, Inc. Pesticidal composition for seed treatment
CA2356263C (en) 1998-12-25 2009-04-21 Teikoku Hormone Mfg. Co., Ltd. Aminopyrazole derivatives
AU7922100A (en) 1999-10-25 2001-05-08 Basf Aktiengesellschaft Agrochemical compositions containing pyrazoles as the active agents and use of said compositions as plant protection agents with a fungicidal action
PE20020506A1 (es) * 2000-08-22 2002-07-09 Glaxo Group Ltd Derivados de pirazol fusionados como inhibidores de la proteina cinasa
US6660690B2 (en) 2000-10-06 2003-12-09 Monsanto Technology, L.L.C. Seed treatment with combinations of insecticides
AU2002239348A1 (en) * 2000-12-15 2002-06-24 Glaxo Group Limited Pyrazolopyridine derivatives
ATE301653T1 (de) * 2000-12-15 2005-08-15 Glaxo Group Ltd Pyrazolopyridine
ES2296910T3 (es) 2001-01-22 2008-05-01 Sankyo Company, Limited Compuestos sustituidos con grupo amino biciclicos.
DE60201074T2 (de) * 2001-03-08 2005-09-15 Smithkline Beecham Corp. Pyrazolopyridinderivate
US20020134012A1 (en) 2001-03-21 2002-09-26 Monsanto Technology, L.L.C. Method of controlling the release of agricultural active ingredients from treated plant seeds
JP2004525150A (ja) * 2001-03-30 2004-08-19 スミスクライン ビーチャム コーポレーション 治療用化合物としてのピラゾロピリジン類の使用
EP1382603B1 (en) 2001-04-26 2008-07-23 Eisai R&D Management Co., Ltd. Nitrogenous fused-ring compound having pyrazolyl group as substituent and medicinal composition thereof
US20050080113A1 (en) 2001-06-11 2005-04-14 Shigenori Ohkawa Medicinal compositions
GB0129476D0 (en) 2001-12-10 2002-01-30 Syngenta Participations Ag Organic compounds
ES2292839T3 (es) * 2001-12-11 2008-03-16 Smithkline Beecham Corporation Derivados de pirazolo-piridina como agentes contra el herpes.
ATE365740T1 (de) 2002-05-10 2007-07-15 Smithkline Beecham Corp Substituierte pyrazolopyrimidine
EP1553096B1 (en) 2002-09-25 2012-10-31 Ube Industries, Ltd. Pyrazole compounds
SE0203654D0 (sv) 2002-12-09 2002-12-09 Astrazeneca Ab New compounds
EA009517B1 (ru) * 2003-06-27 2008-02-28 Байер Кропсайенс Аг Пиразолопиримидины
WO2005012258A1 (ja) 2003-07-30 2005-02-10 Kyowa Hakko Kogyo Co., Ltd. タンパク質キナーゼ阻害剤
US20080207685A1 (en) 2003-11-20 2008-08-28 Eli Lilly And Company Heterocyclic Compounds As Modulators Of Peroxisome Proliferator Activated Receptors, Useful For The Treatment And/Or Prevention Of Disorders Modulated By A Ppar
US7459562B2 (en) 2004-04-23 2008-12-02 Bristol-Myers Squibb Company Monocyclic heterocycles as kinase inhibitors
TWI326282B (en) * 2004-04-28 2010-06-21 Mitsubishi Tanabe Pharma Corp Heterocyclic compound
TW200614993A (en) 2004-06-11 2006-05-16 Akzo Nobel Nv 4-phenyl-pyrimidine-2-carbonitrile derivatives
ATE527258T1 (de) 2004-07-28 2011-10-15 Takeda Pharmaceutical Pyrroloä2,3-cüpyridinverbindung, verfahren zu deren herstellung und anwendung
WO2006055245A2 (en) * 2004-11-17 2006-05-26 Smithkline Beecham Corporation Process for preparing pyrazolopyridine compounds
US7473784B2 (en) 2005-08-01 2009-01-06 Bristol-Myers Squibb Company Benzothiazole and azabenzothiazole compounds useful as kinase inhibitors
AU2006283504B2 (en) 2005-08-24 2011-08-25 E. I. Du Pont De Nemours And Company Compositions providing tolerance to multiple herbicides and methods of use thereof
WO2007024843A2 (en) 2005-08-26 2007-03-01 Smithkline Beecham Corporation Pyrimidinyl-pyrazole inhibitors of aurora kinases
WO2007027777A2 (en) 2005-08-31 2007-03-08 Monsanto Technology Llc Nucleotide sequences encoding insecticidal proteins
GB0605120D0 (en) 2006-03-14 2006-04-26 Novartis Ag Organic Compounds
TW200811134A (en) 2006-07-12 2008-03-01 Irm Llc Compounds and compositions as protein kinase inhibitors
DK2324008T3 (da) 2008-07-24 2012-07-23 Nerviano Medical Sciences Srl Diarylpyrazol som protein kinase inhibitorer
EP2367797A1 (en) 2008-11-26 2011-09-28 Arena Pharmaceuticals, Inc. Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (pgi2) receptor useful for the treatment of disorders related thereto
EP2198710A1 (de) 2008-12-19 2010-06-23 Bayer CropScience AG Verwendung von 5-Pyridin-4yl-(1,3)Thiazole zur Bekämpfung phytopathogener Pilze
EP2308866A1 (de) * 2009-10-09 2011-04-13 Bayer CropScience AG Phenylpyri(mi)dinylpyrazole und ihre Verwendung als Fungizide
AR079545A1 (es) * 2009-12-21 2012-02-01 Bayer Cropscience Ag Tienilpiri(mi)dinilazol
AR081810A1 (es) 2010-04-07 2012-10-24 Bayer Cropscience Ag Piridinilpirazoles biciclicos
EP2402345A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazole fused bicyclic compounds
EP2402338A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402337A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402340A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402343A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazole-fused bicyclic compounds
EP2402339A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402344A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazole fused bicyclic compounds
PL2763987T3 (pl) * 2011-10-06 2019-01-31 Bayer Cropscience Ag Heterocyklilopiry(mi)dynylopirazole jako środki grzybobójcze

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009076440A2 (en) * 2007-12-12 2009-06-18 E.I. Du Pont De Nemours And Company Fungicidal bicyclic pyrazoles

Also Published As

Publication number Publication date
BR112014008222A2 (pt) 2017-04-25
RU2627272C2 (ru) 2017-08-04
EP2763993B1 (en) 2017-04-19
CN103958518A (zh) 2014-07-30
JP2014528961A (ja) 2014-10-30
AU2012320578A1 (en) 2014-04-10
KR20140072177A (ko) 2014-06-12
NZ622704A (en) 2016-05-27
ZA201403228B (en) 2017-08-30
JP6211522B2 (ja) 2017-10-11
UA114410C2 (uk) 2017-06-12
IN2014CN02475A (enExample) 2015-06-19
PL2763993T3 (pl) 2017-09-29
CO6920305A2 (es) 2014-04-10
US20140364456A1 (en) 2014-12-11
MX2014003918A (es) 2014-04-25
MX351460B (es) 2017-10-16
ES2632584T3 (es) 2017-09-14
DK2763993T3 (en) 2017-07-24
EP2763993A1 (en) 2014-08-13
CN103958518B (zh) 2017-07-04
CL2014000807A1 (es) 2014-09-05
US9314026B2 (en) 2016-04-19
WO2013050434A1 (en) 2013-04-11
RU2014117822A (ru) 2015-11-20

Similar Documents

Publication Publication Date Title
US9247748B2 (en) Bis(difluoromethyl)pyrazoles as fungicides
WO2012175513A1 (en) Thienylpyri(mi)dinylpyrazole
US9220266B2 (en) Ketoheteroarylpiperidine and -piperazine derivatives as fungicides
US20110301197A1 (en) Bis(difluoromethyl)pyrazoles as Fungicides
AU2012320578B2 (en) Heterocyclylpyri(mi)dinylpyrazole
AU2012320581B2 (en) Heterocyclylpyri (mi) dinylpyrazole as fungicidals
US8507472B2 (en) Bicyclic pyridinylpyrazoles
TW201331204A (zh) 雜環吡(嘧)啶基吡唑
NZ623290B2 (en) Heterocyclylpyri (mi) dinylpyrazole as fungicidals
NZ622704B2 (en) Heterocyclylpyri(mi)dinylpyrazole

Legal Events

Date Code Title Description
FGA Letters patent sealed or granted (standard patent)
MK14 Patent ceased section 143(a) (annual fees not paid) or expired