KR20120088755A - Mglur4 알로스테릭 강화제, 조성물 및 신경 기능이상을 치료하는 방법 - Google Patents

Mglur4 알로스테릭 강화제, 조성물 및 신경 기능이상을 치료하는 방법 Download PDF

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KR20120088755A
KR20120088755A KR1020127013191A KR20127013191A KR20120088755A KR 20120088755 A KR20120088755 A KR 20120088755A KR 1020127013191 A KR1020127013191 A KR 1020127013191A KR 20127013191 A KR20127013191 A KR 20127013191A KR 20120088755 A KR20120088755 A KR 20120088755A
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optionally substituted
cycloalkyl
membered ring
alkyl
ring containing
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피. 제프리 콘
크레이그 더블유. 린즐리
코레이 알. 홉킨스
콜린 엠. 니스웬더
로코 디. 고글리오티
제임스 엠. 살로비치
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벤더르빌트 유니버시티
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KR1020127013191A 2009-10-22 2010-10-22 Mglur4 알로스테릭 강화제, 조성물 및 신경 기능이상을 치료하는 방법 Withdrawn KR20120088755A (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US25406209P 2009-10-22 2009-10-22
US61/254,062 2009-10-22
US29272510P 2010-01-06 2010-01-06
US61/292,725 2010-01-06
PCT/US2010/053837 WO2011050316A1 (en) 2009-10-22 2010-10-22 Mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

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KR20120088755A true KR20120088755A (ko) 2012-08-08

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KR1020127013201A Withdrawn KR20120129869A (ko) 2009-10-22 2010-10-22 Mglur4 알로스테릭 강화제, 조성물 및 신경 기능이상을 치료하는 방법
KR1020127013191A Withdrawn KR20120088755A (ko) 2009-10-22 2010-10-22 Mglur4 알로스테릭 강화제, 조성물 및 신경 기능이상을 치료하는 방법

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US (2) US9180192B2 (enExample)
EP (2) EP2490537A4 (enExample)
JP (2) JP2013508413A (enExample)
KR (2) KR20120129869A (enExample)
CN (2) CN102665411A (enExample)
AU (2) AU2010310518A1 (enExample)
BR (2) BR112012009576A2 (enExample)
CA (2) CA2779298A1 (enExample)
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JP2012516355A (ja) 2009-01-28 2012-07-19 ヴァンダービルト ユニバーシティー mGLuR4アロステリック増強剤としての置換された1,1,3,3−テトラオキシドベンゾ[d][1,3,2]ジチアゾール、組成物、および神経機能不全を治療する方法
US8759377B2 (en) 2009-11-23 2014-06-24 Vanderbilt University Substituted dioxopiperidines and dioxopyrrolidines as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
CN102933572B (zh) 2010-04-07 2015-01-07 霍夫曼-拉罗奇有限公司 吡唑-4-基-杂环基-甲酰胺化合物及其使用方法
BR112014007203A2 (pt) 2011-09-27 2017-06-13 F.Hoffmann-La Roche Ag composto, composição farmacêutica, método de tratamento, utilização de um composto, conjunto e invenção
EP2853532B1 (en) 2013-09-28 2020-12-09 Instytut Farmakologii Polskiej Akademii Nauk 1,2,4-oxadiazole derivatives as allosteric modulators of metabotropic glutamate receptors belonging to group III
US10221172B2 (en) 2015-01-13 2019-03-05 Vanderbilt University Benzothiazole and benzisothiazole-substituted compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
WO2016123629A1 (en) 2015-01-30 2016-08-04 Vanderbilt University Indazole and azaindazole substituted compounds as mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
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