KR20070052693A - 폴리헤테로시클릭 화합물 및 대사성 글루타메이트 수용체길항제로서 이들의 용도 - Google Patents

폴리헤테로시클릭 화합물 및 대사성 글루타메이트 수용체길항제로서 이들의 용도 Download PDF

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Publication number
KR20070052693A
KR20070052693A KR1020067015825A KR20067015825A KR20070052693A KR 20070052693 A KR20070052693 A KR 20070052693A KR 1020067015825 A KR1020067015825 A KR 1020067015825A KR 20067015825 A KR20067015825 A KR 20067015825A KR 20070052693 A KR20070052693 A KR 20070052693A
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South Korea
Prior art keywords
alkyl
methyl
phenyl
triazol
chloro
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Ceased
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KR1020067015825A
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English (en)
Korean (ko)
Inventor
잘라지 알로라
루이스 에드워드
메트빈 아이작
아니카 컬스
카린 스타프
압델말릭 슬래씨
토미스라브 스테파낙
데이비드 웬스보
타오 진
비욘 홈
Original Assignee
아스트라제네카 아베
엔피에스 파마슈티칼즈, 인코포레이티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34886130&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20070052693(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 아스트라제네카 아베, 엔피에스 파마슈티칼즈, 인코포레이티드 filed Critical 아스트라제네카 아베
Publication of KR20070052693A publication Critical patent/KR20070052693A/ko
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07—ORGANIC CHEMISTRY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020067015825A 2004-02-18 2005-02-17 폴리헤테로시클릭 화합물 및 대사성 글루타메이트 수용체길항제로서 이들의 용도 Ceased KR20070052693A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54529204P 2004-02-18 2004-02-18
USUS60/545,292 2004-02-18

Publications (1)

Publication Number Publication Date
KR20070052693A true KR20070052693A (ko) 2007-05-22

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ID=34886130

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KR1020067015825A Ceased KR20070052693A (ko) 2004-02-18 2005-02-17 폴리헤테로시클릭 화합물 및 대사성 글루타메이트 수용체길항제로서 이들의 용도

Country Status (20)

Country Link
US (2) US20070185100A1 (https=)
EP (1) EP1716143A1 (https=)
JP (1) JP2007523181A (https=)
KR (1) KR20070052693A (https=)
CN (1) CN1918154A (https=)
AR (1) AR047966A1 (https=)
AU (1) AU2005214378A1 (https=)
BR (1) BRPI0507481A (https=)
CA (1) CA2555272A1 (https=)
IL (1) IL177058A0 (https=)
MX (1) MXPA06009023A (https=)
NO (1) NO20063469L (https=)
NZ (1) NZ548693A (https=)
RU (1) RU2381226C2 (https=)
SG (1) SG149900A1 (https=)
TW (1) TW200538179A (https=)
UA (1) UA82434C2 (https=)
UY (1) UY28764A1 (https=)
WO (1) WO2005080386A1 (https=)
ZA (1) ZA200606314B (https=)

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WO2009054792A1 (en) * 2007-10-26 2009-04-30 Astrazeneca Ab Aminopyridine derivatives as modulators of mglur5
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JP2013518085A (ja) 2010-02-01 2013-05-20 ノバルティス アーゲー ＣＲＦ−１受容体アンタゴニストとしてのピラゾロ［５，１ｂ］オキサゾール誘導体
JP5748777B2 (ja) 2010-02-02 2015-07-15 ノバルティス アーゲー Ｃｒｆ受容体アンタゴニストとしてのシクロヘキシルアミド誘導体
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NZ548693A (en) 2010-05-28
UA82434C2 (uk) 2008-04-10
UY28764A1 (es) 2005-06-30
EP1716143A1 (en) 2006-11-02
JP2007523181A (ja) 2007-08-16
NO20063469L (no) 2006-11-15
TW200538179A (en) 2005-12-01
BRPI0507481A (pt) 2007-07-17
SG149900A1 (en) 2009-02-27
CA2555272A1 (en) 2005-09-01
IL177058A0 (en) 2006-12-10
US20060025414A1 (en) 2006-02-02
RU2381226C2 (ru) 2010-02-10
MXPA06009023A (es) 2007-03-08
ZA200606314B (en) 2007-12-27
WO2005080386A1 (en) 2005-09-01
US20070185100A1 (en) 2007-08-09
AU2005214378A1 (en) 2005-09-01
AR047966A1 (es) 2006-03-15
RU2006127572A (ru) 2008-03-27

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