KR20060130697A - 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 - Google Patents

신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 Download PDF

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KR20060130697A
KR20060130697A KR1020067020318A KR20067020318A KR20060130697A KR 20060130697 A KR20060130697 A KR 20060130697A KR 1020067020318 A KR1020067020318 A KR 1020067020318A KR 20067020318 A KR20067020318 A KR 20067020318A KR 20060130697 A KR20060130697 A KR 20060130697A
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South Korea
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alkyl
hydrogen
methoxy
hydroxy
hexahydro
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Korean (ko)
Inventor
베아테 슈미트
디터 플로커치
아르민 하첼만
크리스토프 치트
요하네스 바르지히
데겐하르트 막스
한스-페터 클라이
울리히 카우츠
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알타나 파마 아게
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/10—Aza-phenanthrenes
    • C07D221/12—Phenanthridines
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Cardiology (AREA)
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  • Diabetes (AREA)
  • Hematology (AREA)
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  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
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  • Communicable Diseases (AREA)
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  • Transplantation (AREA)
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KR1020067020318A 2004-03-10 2005-03-09 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 Ceased KR20060130697A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP04100990.3 2004-03-10
EP04100990 2004-03-10
EP04106677.0 2004-12-17
EP04106677 2004-12-17

Publications (1)

Publication Number Publication Date
KR20060130697A true KR20060130697A (ko) 2006-12-19

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KR1020067020318A Ceased KR20060130697A (ko) 2004-03-10 2005-03-09 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도

Country Status (15)

Country Link
US (1) US20070185149A1 (enExample)
EP (1) EP1725534A1 (enExample)
JP (1) JP2007527901A (enExample)
KR (1) KR20060130697A (enExample)
CN (1) CN1926113B (enExample)
AR (1) AR049324A1 (enExample)
AU (1) AU2005221832A1 (enExample)
BR (1) BRPI0508481A (enExample)
CA (1) CA2558391A1 (enExample)
IL (1) IL177496A0 (enExample)
MX (1) MXPA06009892A (enExample)
NO (1) NO20064415L (enExample)
NZ (1) NZ549254A (enExample)
TW (1) TW200600499A (enExample)
WO (1) WO2005087745A1 (enExample)

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AR049419A1 (es) * 2004-03-03 2006-08-02 Altana Pharma Ag Hidroxi-6-fenilfenantridinas sustituidas con heterociclilo
EP1791847A2 (en) 2004-09-08 2007-06-06 Altana Pharma AG Novel 3-thia-10-aza-phenanthrene derivatives
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NZ560268A (en) 2005-03-02 2010-12-24 Nycomed Gmbh Novel salts of 6-heterocyclyl substituted hexahydrophenanthridine derivatives
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
US20100041662A1 (en) 2006-10-30 2010-02-18 Sandrine Ferrand Heterocyclic compounds as antiinflammatory agents
JP5362729B2 (ja) 2007-10-04 2013-12-11 エフ．ホフマン−ラ ロシュ アーゲー シクロプロピルアリールアミド誘導体及びその使用
WO2009087224A1 (en) 2008-01-11 2009-07-16 Novartis Ag Pyrimidines as kinase inhibitors
WO2010102980A1 (en) * 2009-03-09 2010-09-16 Basf Se Process for preparing substituted 2-nitrobiphenyls
UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
JP5959541B2 (ja) 2011-02-25 2016-08-02 ノバルティス アーゲー Ｔｒｋ阻害剤としてのピラゾロ［１，５−ａ］ピリジン

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WO2005087745A8 (en) 2006-10-26
AR049324A1 (es) 2006-07-19
JP2007527901A (ja) 2007-10-04
NO20064415L (no) 2006-10-10
AU2005221832A1 (en) 2005-09-22
BRPI0508481A (pt) 2007-07-31
US20070185149A1 (en) 2007-08-09
EP1725534A1 (en) 2006-11-29
TW200600499A (en) 2006-01-01
WO2005087745A1 (en) 2005-09-22
CN1926113B (zh) 2010-06-23
MXPA06009892A (es) 2007-03-01
CN1926113A (zh) 2007-03-07
CA2558391A1 (en) 2005-09-22
IL177496A0 (en) 2006-12-10

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