KR20050085681A - 프로테아제 억제제와 같은 사이토크롬 ｐ450의 억제제와함께 비-뉴클레오시드 역전사효소 억제제(ｎｎｒｔｉ)를함유하는 배합물의 용도 - Google Patents
프로테아제 억제제와 같은 사이토크롬 ｐ450의 억제제와함께 비-뉴클레오시드 역전사효소 억제제(ｎｎｒｔｉ)를함유하는 배합물의 용도 Download PDFInfo
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- KR20050085681A KR20050085681A KR1020057011003A KR20057011003A KR20050085681A KR 20050085681 A KR20050085681 A KR 20050085681A KR 1020057011003 A KR1020057011003 A KR 1020057011003A KR 20057011003 A KR20057011003 A KR 20057011003A KR 20050085681 A KR20050085681 A KR 20050085681A
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- inhibitor
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A—HUMAN NECESSITIES
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- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
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- A—HUMAN NECESSITIES
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Life Sciences & Earth Sciences (AREA)
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- General Health & Medical Sciences (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US43369002P | 2002-12-16 | 2002-12-16 | |
| US60/433,690 | 2002-12-16 |
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| KR20050085681A true KR20050085681A (ko) | 2005-08-29 |
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| KR1020057011003A Withdrawn KR20050085681A (ko) | 2002-12-16 | 2003-12-15 | 프로테아제 억제제와 같은 사이토크롬 ｐ450의 억제제와함께 비-뉴클레오시드 역전사효소 억제제(ｎｎｒｔｉ)를함유하는 배합물의 용도 |
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| US (2) | US20040152625A1 (https=) |
| EP (1) | EP1575595A1 (https=) |
| JP (1) | JP2006511538A (https=) |
| KR (1) | KR20050085681A (https=) |
| CN (1) | CN1726041A (https=) |
| AU (1) | AU2003296647A1 (https=) |
| BR (1) | BR0317095A (https=) |
| CA (1) | CA2510143A1 (https=) |
| EA (1) | EA200500894A1 (https=) |
| EC (1) | ECSP055854A (https=) |
| HR (1) | HRP20050557A2 (https=) |
| IL (1) | IL169099A0 (https=) |
| MX (1) | MXPA05005773A (https=) |
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| PL (1) | PL376900A1 (https=) |
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| UA (1) | UA81003C2 (https=) |
| WO (1) | WO2004054586A1 (https=) |
| ZA (1) | ZA200502947B (https=) |
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| EP1944042A1 (en) | 2003-10-27 | 2008-07-16 | Vertex Pharmceuticals Incorporated | Combinations for HCV treatment |
| US7388008B2 (en) | 2004-08-02 | 2008-06-17 | Ambrilia Biopharma Inc. | Lysine based compounds |
| WO2006114001A1 (en) * | 2005-04-27 | 2006-11-02 | Ambrilia Biopharma Inc. | Method for improving pharmacokinetics of protease inhibitors and protease inhibitor precursors |
| ES2452718T3 (es) | 2005-11-30 | 2014-04-02 | Taimed Biologics, Inc. | Profármacos a base de lisina de inhibidores de la aspartil proteasa y procesos para su preparación |
| CN1907138B (zh) * | 2006-08-11 | 2011-01-12 | 华南师范大学 | 一种沙田柚子汁提取物及其提取方法和应用 |
| CA2664118A1 (en) | 2006-09-21 | 2008-07-03 | Ambrilia Biopharma Inc. | Protease inhibitors |
| RU2544010C2 (ru) | 2009-02-27 | 2015-03-10 | Энанта Фармасьютикалс, Инк. | Ингибиторы вируса гепатита с |
| PL2421527T3 (pl) * | 2009-04-25 | 2018-10-31 | F.Hoffmann-La Roche Ag | Sposoby poprawy właściwości farmakokinetycznych |
| EP2429568B1 (en) | 2009-05-13 | 2016-08-17 | Enanta Pharmaceuticals, Inc. | Macrocyclic compounds as hepatitis c virus inhibitors |
| US8653070B2 (en) | 2009-12-14 | 2014-02-18 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
| WO2014013014A1 (en) | 2012-07-18 | 2014-01-23 | Fundació Privada Centre De Regulació Genòmica (Crg) | Jak inhibitors for activation of epidermal stem cell populations |
| WO2018041989A1 (en) | 2016-09-02 | 2018-03-08 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods for diagnosing and treating refractory celiac disease type 2 |
| EP3947737A2 (en) | 2019-04-02 | 2022-02-09 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods of predicting and preventing cancer in patients having premalignant lesions |
| EP3955920A1 (en) | 2019-04-16 | 2022-02-23 | Institut National de la Santé et de la Recherche Médicale (INSERM) | Use of jak inhibitors for the treatment of painful conditions involving nav1.7 channels |
| WO2023222565A1 (en) | 2022-05-16 | 2023-11-23 | Institut National de la Santé et de la Recherche Médicale | Methods for assessing the exhaustion of hematopoietic stems cells induced by chronic inflammation |
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| US5539122A (en) * | 1989-05-23 | 1996-07-23 | Abbott Laboratories | Retroviral protease inhibiting compounds |
| IL111991A (en) * | 1994-01-28 | 2000-07-26 | Abbott Lab | Liquid pharmaceutical composition of HIV protease inhibitors in organic solvent |
| US6037157A (en) * | 1995-06-29 | 2000-03-14 | Abbott Laboratories | Method for improving pharmacokinetics |
| EP0986375A2 (en) * | 1997-04-07 | 2000-03-22 | Triangle Pharmaceuticals Inc. | Use of mkc-442 in combination with other antiviral agents |
| AU762349B2 (en) * | 1998-11-04 | 2003-06-26 | Pharmacia & Upjohn Company | Method for improving the pharmacokinetics of tipranavir |
| US6391919B1 (en) * | 2000-01-12 | 2002-05-21 | Bristol-Myers Squibb Pharma Company | Bis-amino acid sulfonamides containing substituted benzyl amines HIV protease inhibitors |
| TWI270547B (en) * | 2000-06-16 | 2007-01-11 | Boehringer Ingelheim Ca Ltd | Non-nucleoside reverse transcriptase inhibitors |
| ES2268499T3 (es) * | 2002-09-19 | 2007-03-16 | Boehringer Ingelheim (Canada) Ltd. | Inhibidores no nucleosidos de transcriptasa inveresa. |
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2003
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2007
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Also Published As
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| WO2004054586A1 (en) | 2004-07-01 |
| HRP20050557A2 (en) | 2006-05-31 |
| RS20050461A (sr) | 2007-08-03 |
| AU2003296647A1 (en) | 2004-07-09 |
| BR0317095A (pt) | 2005-10-25 |
| EP1575595A1 (en) | 2005-09-21 |
| MXPA05005773A (es) | 2005-08-16 |
| PL376900A1 (pl) | 2006-01-09 |
| NO20053455L (no) | 2005-08-10 |
| EA200500894A1 (ru) | 2006-02-24 |
| NZ541187A (en) | 2007-12-21 |
| US20080096832A1 (en) | 2008-04-24 |
| ECSP055854A (es) | 2006-01-16 |
| UA81003C2 (en) | 2007-11-26 |
| CA2510143A1 (en) | 2004-07-01 |
| US20040152625A1 (en) | 2004-08-05 |
| CN1726041A (zh) | 2006-01-25 |
| JP2006511538A (ja) | 2006-04-06 |
| IL169099A0 (en) | 2007-07-04 |
| ZA200502947B (en) | 2008-01-30 |
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