KR20050072445A - 비만 치료용의 멜라노코르틴 수용체 리간드로서의2-알킬-(2-아미노-3-아릴-프로피온일)-피페라진 유도체 및관련 화합물 - Google Patents

비만 치료용의 멜라노코르틴 수용체 리간드로서의2-알킬-(2-아미노-3-아릴-프로피온일)-피페라진 유도체 및관련 화합물 Download PDF

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KR20050072445A
KR20050072445A KR1020057006836A KR20057006836A KR20050072445A KR 20050072445 A KR20050072445 A KR 20050072445A KR 1020057006836 A KR1020057006836 A KR 1020057006836A KR 20057006836 A KR20057006836 A KR 20057006836A KR 20050072445 A KR20050072445 A KR 20050072445A
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South Korea
Prior art keywords
ethyl
oxo
methyl
piperazin
fluorophenyl
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KR1020057006836A
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Korean (ko)
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프랭크 홀락 에베티노
신롱 톈
위즐로 애덤 마주르
애니-오딜 콜슨
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더 프록터 앤드 갬블 캄파니
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Publication of KR20050072445A publication Critical patent/KR20050072445A/ko

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
KR1020057006836A 2002-10-23 2003-10-22 비만 치료용의 멜라노코르틴 수용체 리간드로서의2-알킬-(2-아미노-3-아릴-프로피온일)-피페라진 유도체 및관련 화합물 KR20050072445A (ko)

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US42057802P 2002-10-23 2002-10-23
US60/420,578 2002-10-23

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