KR20040097332A - 아실-3-카복시페닐우레아 유도체, 이의 제조방법 및 용도 - Google Patents

아실-3-카복시페닐우레아 유도체, 이의 제조방법 및 용도 Download PDF

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Publication number
KR20040097332A
KR20040097332A KR10-2004-7016149A KR20047016149A KR20040097332A KR 20040097332 A KR20040097332 A KR 20040097332A KR 20047016149 A KR20047016149 A KR 20047016149A KR 20040097332 A KR20040097332 A KR 20040097332A
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KR
South Korea
Prior art keywords
alkyl
cycloalkyl
alkynyl
alkenyl
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
KR10-2004-7016149A
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English (en)
Korean (ko)
Inventor
데포사엘리자베쓰
카데라이트디터
쇼에나핑거칼
클라분데토마스
부르거한스외르크
헤를링안드레아스
벤트칼울리히
폰뢰데른에리히
엔센알폰스
Original Assignee
아벤티스 파마 도이칠란트 게엠베하
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 아벤티스 파마 도이칠란트 게엠베하 filed Critical 아벤티스 파마 도이칠란트 게엠베하
Publication of KR20040097332A publication Critical patent/KR20040097332A/ko
Withdrawn legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/46—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
    • C07C275/48—Y being a hydrogen or a carbon atom
    • C07C275/54—Y being a carbon atom of a six-membered aromatic ring, e.g. benzoylureas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR10-2004-7016149A 2002-04-11 2003-03-28 아실-3-카복시페닐우레아 유도체, 이의 제조방법 및 용도 Withdrawn KR20040097332A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10215908A DE10215908B4 (de) 2002-04-11 2002-04-11 Acyl-3-carboxyphenyl-harnstoffderivate und deren Verwendung als Arzneimittel
DE10215908.4 2002-04-11
PCT/EP2003/003254 WO2003084923A1 (de) 2002-04-11 2003-03-28 Acyl-3-carboxyphenyl-harnstoffderivate, verfahren zu deren herstellung und deren verwendung

Publications (1)

Publication Number Publication Date
KR20040097332A true KR20040097332A (ko) 2004-11-17

Family

ID=28684936

Family Applications (1)

Application Number Title Priority Date Filing Date
KR10-2004-7016149A Withdrawn KR20040097332A (ko) 2002-04-11 2003-03-28 아실-3-카복시페닐우레아 유도체, 이의 제조방법 및 용도

Country Status (23)

Country Link
EP (1) EP1497263B1 (https=)
JP (1) JP4328212B2 (https=)
KR (1) KR20040097332A (https=)
CN (1) CN1263734C (https=)
AR (1) AR039402A1 (https=)
AT (1) ATE404532T1 (https=)
AU (1) AU2003232192A1 (https=)
BR (1) BR0309130A (https=)
CA (1) CA2481819A1 (https=)
DE (2) DE10215908B4 (https=)
HR (1) HRP20040931A2 (https=)
HU (1) HUP0500203A2 (https=)
IL (1) IL164248A0 (https=)
MA (1) MA27195A1 (https=)
MX (1) MXPA04009239A (https=)
NO (1) NO20044881L (https=)
NZ (1) NZ535833A (https=)
PL (1) PL371317A1 (https=)
RS (1) RS88704A (https=)
RU (1) RU2004133046A (https=)
TW (1) TW200401765A (https=)
WO (1) WO2003084923A1 (https=)
ZA (1) ZA200407361B (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10215907A1 (de) * 2002-04-11 2003-11-06 Aventis Pharma Gmbh Acyl-4-carboxyphenyl-harnstoffderivate, Verfahren zu deren Herstellung und deren Verwendung
DE10306502B4 (de) * 2003-02-17 2005-03-17 Aventis Pharma Deutschland Gmbh Substituierte 3-(Benzoylureido)-thiophenderivate und sie enthaltende Arzneimittel
DE10308352A1 (de) 2003-02-27 2004-09-09 Aventis Pharma Deutschland Gmbh Arylcycloalkylderivate mit verzweigten Seitenketten, Verfahren zu ihrer Herstellung und ihre Anwendung als Arzneimittel
US7148246B2 (en) 2003-02-27 2006-12-12 Sanofi-Aventis Deutschland Gmbh Cycloalkyl derivatives having bioisosteric carboxylic acid groups, processes for their preparation and their use as pharmaceuticals
DE10308355A1 (de) 2003-02-27 2004-12-23 Aventis Pharma Deutschland Gmbh Aryl-cycloalkyl substituierte Alkansäurederivate, Verfahren zu ihrer Herstellung und ihre Anwendung als Arzneimittel
DE10308353A1 (de) 2003-02-27 2004-12-02 Aventis Pharma Deutschland Gmbh Diarylcycloalkylderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE10308351A1 (de) 2003-02-27 2004-11-25 Aventis Pharma Deutschland Gmbh 1,3-substituierte Cycloalkylderivate mit sauren, meist heterocyclischen Gruppen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
US7241787B2 (en) 2004-01-25 2007-07-10 Sanofi-Aventis Deutschland Gmbh Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments
EP1586573B1 (en) 2004-04-01 2007-02-07 Sanofi-Aventis Deutschland GmbH Oxadiazolones, processes for their preparation and their use as pharmaceuticals
DE102005026762A1 (de) 2005-06-09 2006-12-21 Sanofi-Aventis Deutschland Gmbh Azolopyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen
PE20110235A1 (es) 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA867420B (en) * 1985-09-30 1987-05-27 Union Carbide Corp Pesticidal 1-(4-aryloxyphenyl)-3-benzoyl urea compounds and process for preparation
GB9313268D0 (en) * 1993-06-28 1993-08-11 Zeneca Ltd Chemical compounds
FI974437A7 (fi) * 1995-06-06 1997-12-05 Pfizer Substituoituja N-(indoli-2-karbonyyli)amideja ja johdannaisia glykogee nifosforylaasi-inhibiittoreina
WO2000056707A1 (en) * 1999-03-24 2000-09-28 Sepracor, Inc. Diaryl thioethers, compositions and uses thereof
US20010053791A1 (en) * 2000-03-16 2001-12-20 Babcock Walter C. Glycogen phosphorylase inhibitor
TR200401029T4 (tr) * 2000-06-09 2004-06-21 Aventis Pharma Deutschland Gmbh Asilfenil-üre türevleri, imalat yöntemleri ve ilaç maddesi olarak kullanımları
GB0021831D0 (en) * 2000-09-06 2000-10-18 Astrazeneca Ab Chemical compounds
PE20021091A1 (es) * 2001-05-25 2003-02-04 Aventis Pharma Gmbh Derivados de fenilurea sustituidos con carbonamida y procedimiento para su preparacion

Also Published As

Publication number Publication date
HK1075650A1 (en) 2005-12-23
CN1263734C (zh) 2006-07-12
PL371317A1 (en) 2005-06-13
IL164248A0 (en) 2005-12-18
EP1497263B1 (de) 2008-08-13
TW200401765A (en) 2004-02-01
NZ535833A (en) 2006-03-31
DE10215908B4 (de) 2005-08-18
WO2003084923A1 (de) 2003-10-16
AR039402A1 (es) 2005-02-16
HRP20040931A2 (en) 2005-02-28
ATE404532T1 (de) 2008-08-15
BR0309130A (pt) 2005-02-01
JP2005522481A (ja) 2005-07-28
CN1646486A (zh) 2005-07-27
MXPA04009239A (es) 2005-01-25
AU2003232192A1 (en) 2003-10-20
ZA200407361B (en) 2006-02-22
MA27195A1 (fr) 2005-01-03
DE50310320D1 (de) 2008-09-25
RS88704A (sr) 2007-02-05
DE10215908A1 (de) 2003-11-06
CA2481819A1 (en) 2003-10-16
NO20044881L (no) 2005-01-07
RU2004133046A (ru) 2005-04-20
EP1497263A1 (de) 2005-01-19
JP4328212B2 (ja) 2009-09-09
HUP0500203A2 (hu) 2005-06-28

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Legal Events

Date Code Title Description
PA0105 International application

Patent event date: 20041008

Patent event code: PA01051R01D

Comment text: International Patent Application

PG1501 Laying open of application
PC1203 Withdrawal of no request for examination
WITN Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid