KR20010085553A - 도파민 재수용 저해물질로 구성된 조성물 및 이를이용하는 방법 - Google Patents
도파민 재수용 저해물질로 구성된 조성물 및 이를이용하는 방법 Download PDFInfo
- Publication number
- KR20010085553A KR20010085553A KR1020017002288A KR20017002288A KR20010085553A KR 20010085553 A KR20010085553 A KR 20010085553A KR 1020017002288 A KR1020017002288 A KR 1020017002288A KR 20017002288 A KR20017002288 A KR 20017002288A KR 20010085553 A KR20010085553 A KR 20010085553A
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- KR
- South Korea
- Prior art keywords
- sibutramine
- didesmethyl
- desmethyl
- metabolite
- racemic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Child & Adolescent Psychology (AREA)
- Addiction (AREA)
- Otolaryngology (AREA)
- Gynecology & Obstetrics (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Psychology (AREA)
- Toxicology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Information Transfer Systems (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9766598P | 1998-08-24 | 1998-08-24 | |
| US9930698P | 1998-09-02 | 1998-09-02 | |
| US09/372,158 US6331571B1 (en) | 1998-08-24 | 1999-08-11 | Methods of treating and preventing attention deficit disorders |
| US60/099,306 | 1999-08-11 | ||
| US60/097,665 | 1999-08-11 | ||
| PCT/US1999/019167 WO2000010551A2 (en) | 1998-08-24 | 1999-08-23 | Methods of using and compositions comprising dopamine reuptake inhibitors |
| US???? | 2000-01-12 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020067012844A Division KR100887008B1 (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를 이용하는방법 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20010085553A true KR20010085553A (ko) | 2001-09-07 |
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Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020017002288A Ceased KR20010085553A (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를이용하는 방법 |
| KR1020087001197A Ceased KR20080011354A (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를 이용하는방법 |
| KR1020067012844A Expired - Fee Related KR100887008B1 (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를 이용하는방법 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087001197A Ceased KR20080011354A (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를 이용하는방법 |
| KR1020067012844A Expired - Fee Related KR100887008B1 (ko) | 1998-08-24 | 1999-08-23 | 도파민 재수용 저해물질로 구성된 조성물 및 이를 이용하는방법 |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US6331571B1 (https=) |
| EP (2) | EP1107746B1 (https=) |
| JP (1) | JP2002523366A (https=) |
| KR (3) | KR20010085553A (https=) |
| CN (1) | CN100415222C (https=) |
| AT (1) | ATE279184T1 (https=) |
| AU (2) | AU772303B2 (https=) |
| CA (1) | CA2341441C (https=) |
| CZ (1) | CZ2001677A3 (https=) |
| DE (1) | DE69921157T2 (https=) |
| DK (1) | DK1107746T3 (https=) |
| ES (1) | ES2226435T3 (https=) |
| HU (1) | HUP0103408A3 (https=) |
| ID (1) | ID28638A (https=) |
| IL (2) | IL141531A0 (https=) |
| NO (1) | NO20010943L (https=) |
| NZ (1) | NZ510193A (https=) |
| PL (1) | PL200264B1 (https=) |
| PT (1) | PT1107746E (https=) |
| WO (1) | WO2000010551A2 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100618176B1 (ko) * | 2004-12-02 | 2006-09-01 | 휴먼팜 주식회사 | 시부트라민 주석산염, 이의 제조 방법 및 이를 포함하는약학적 조성물 |
| KR100632470B1 (ko) * | 2005-02-25 | 2006-10-12 | 민연식 | 결정성 시부트라민 캄실레이트염과 이의 제조방법 |
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| US6339106B1 (en) * | 1999-08-11 | 2002-01-15 | Sepracor, Inc. | Methods and compositions for the treatment and prevention of sexual dysfunction |
| US6974838B2 (en) | 1998-08-24 | 2005-12-13 | Sepracor Inc. | Methods of treating or preventing pain using sibutramine metabolites |
| US6323242B1 (en) | 1998-12-02 | 2001-11-27 | Peter Sterling Mueller | Treatment of disorders secondary to organic impairments |
| US6696495B2 (en) * | 1998-12-02 | 2004-02-24 | Snowden Pharmaceuticals, Llc | Treatment of disorders secondary to organic impairments |
| MXPA01009404A (es) * | 1999-03-19 | 2004-03-19 | Abbott Gmbh & Co Kg | Metodo para tratar trastornos de alimentacion. |
| DE60022692T2 (de) * | 1999-07-01 | 2006-06-22 | Pharmacia & Upjohn Co. Llc, Kalamazoo | (S,S)-Reboxetin zur Behandlung von Migränekopfschmerzen |
| US6399826B1 (en) | 1999-08-11 | 2002-06-04 | Sepracor Inc. | Salts of sibutramine metabolites, methods of making sibutramine metabolites and intermediates useful in the same, and methods of treating pain |
| WO2002036540A2 (en) * | 2000-11-02 | 2002-05-10 | Torrent Pharmaceuticals Ltd | PROCESS FOR PREPARATION OF β-PHENETHYLAMINE DERIVATIVE |
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| KR20060080817A (ko) * | 2005-01-06 | 2006-07-11 | 씨제이 주식회사 | 시부트라민의 디카복실산염 |
| JP2008526836A (ja) * | 2005-01-06 | 2008-07-24 | シージェー チェイルジェダン コーポレーション | シブトラミンの無機酸塩 |
| KR20060093564A (ko) * | 2005-02-22 | 2006-08-25 | 종근당바이오 주식회사 | 무수 시부트라민 말산염 및 이의 제조 방법 |
| PL385455A1 (pl) * | 2005-04-22 | 2008-11-24 | Teva Pharmaceuticals Usa,Inc. | Doustna rozpadająca się farmaceutyczna tabletka preparatów olanzapiny |
| WO2006136945A1 (en) * | 2005-06-17 | 2006-12-28 | Pfizer Products Inc. | METABOLITES OF 1_ [_6- (1-ETHYL-l-HYDROXY-PROPYL) -PYRIDIN-3-YL] -3- [2- (4-METHYL-PIPERAZIN-I-YL) -BE NZYL] -PYRR0LIDIN-2-0NE AS SERATONIN RECEPTOR ANTAGONISTS |
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-
1999
- 1999-08-11 US US09/372,158 patent/US6331571B1/en not_active Expired - Lifetime
- 1999-08-23 EP EP99945137A patent/EP1107746B1/en not_active Expired - Lifetime
- 1999-08-23 AU AU57817/99A patent/AU772303B2/en not_active Ceased
- 1999-08-23 EP EP04018454A patent/EP1475086A3/en not_active Withdrawn
- 1999-08-23 HU HU0103408A patent/HUP0103408A3/hu unknown
- 1999-08-23 KR KR1020017002288A patent/KR20010085553A/ko not_active Ceased
- 1999-08-23 KR KR1020087001197A patent/KR20080011354A/ko not_active Ceased
- 1999-08-23 PL PL346843A patent/PL200264B1/pl not_active IP Right Cessation
- 1999-08-23 ID IDW20010700A patent/ID28638A/id unknown
- 1999-08-23 PT PT99945137T patent/PT1107746E/pt unknown
- 1999-08-23 DK DK99945137T patent/DK1107746T3/da active
- 1999-08-23 DE DE69921157T patent/DE69921157T2/de not_active Expired - Lifetime
- 1999-08-23 WO PCT/US1999/019167 patent/WO2000010551A2/en not_active Ceased
- 1999-08-23 ES ES99945137T patent/ES2226435T3/es not_active Expired - Lifetime
- 1999-08-23 JP JP2000565873A patent/JP2002523366A/ja active Pending
- 1999-08-23 CZ CZ2001677A patent/CZ2001677A3/cs unknown
- 1999-08-23 CN CNB998124664A patent/CN100415222C/zh not_active Expired - Fee Related
- 1999-08-23 AT AT99945137T patent/ATE279184T1/de active
- 1999-08-23 IL IL14153199A patent/IL141531A0/xx unknown
- 1999-08-23 CA CA2341441A patent/CA2341441C/en not_active Expired - Fee Related
- 1999-08-23 NZ NZ510193A patent/NZ510193A/en not_active IP Right Cessation
- 1999-08-23 KR KR1020067012844A patent/KR100887008B1/ko not_active Expired - Fee Related
-
2001
- 2001-02-20 IL IL141531A patent/IL141531A/en not_active IP Right Cessation
- 2001-02-23 NO NO20010943A patent/NO20010943L/no not_active Application Discontinuation
- 2001-12-04 US US10/000,806 patent/US6538034B2/en not_active Expired - Lifetime
-
2003
- 2003-03-25 US US10/395,298 patent/US7071234B2/en not_active Expired - Fee Related
-
2004
- 2004-03-03 AU AU2004200875A patent/AU2004200875B2/en not_active Ceased
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100618176B1 (ko) * | 2004-12-02 | 2006-09-01 | 휴먼팜 주식회사 | 시부트라민 주석산염, 이의 제조 방법 및 이를 포함하는약학적 조성물 |
| KR100632470B1 (ko) * | 2005-02-25 | 2006-10-12 | 민연식 | 결정성 시부트라민 캄실레이트염과 이의 제조방법 |
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