KR102791105B1 - Rna 바이러스 감염을 치료하기 위한 페닐/피리딜-n-페닐/피리딜 유도체 - Google Patents

Rna 바이러스 감염을 치료하기 위한 페닐/피리딜-n-페닐/피리딜 유도체 Download PDF

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KR102791105B1
KR102791105B1 KR1020217001299A KR20217001299A KR102791105B1 KR 102791105 B1 KR102791105 B1 KR 102791105B1 KR 1020217001299 A KR1020217001299 A KR 1020217001299A KR 20217001299 A KR20217001299 A KR 20217001299A KR 102791105 B1 KR102791105 B1 KR 102791105B1
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acceptable salts
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KR20210039374A (ko
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디디어 셰레
자말 타지
플로렌스 마후토-베처
로메인 나즈만
줄리앙 산토
세실 아폴리
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아비박스
쌍트르 나셔날 드 라 르쉐르쉐 씨앙띠피끄
유니베르시테 드 몽펠리에
엥스띠뛰 퀴리
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
    • C07D239/12—Nitrogen atoms not forming part of a nitro radical
    • C07D239/14—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to said nitrogen atoms
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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