KR102186704B1 - 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 - Google Patents
서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 Download PDFInfo
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- KR102186704B1 KR102186704B1 KR1020190018619A KR20190018619A KR102186704B1 KR 102186704 B1 KR102186704 B1 KR 102186704B1 KR 1020190018619 A KR1020190018619 A KR 1020190018619A KR 20190018619 A KR20190018619 A KR 20190018619A KR 102186704 B1 KR102186704 B1 KR 102186704B1
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- sustained
- pharmaceutically acceptable
- acceptable salt
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- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/127—Liposomes
- A61K9/1274—Non-vesicle bilayer structures, e.g. liquid crystals, tubules, cubic phases, cochleates; Sponge phases
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Endocrinology (AREA)
- Zoology (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Dispersion Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020190018619A KR102186704B1 (ko) | 2019-02-18 | 2019-02-18 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
| US17/310,689 US20220125888A1 (en) | 2019-02-18 | 2020-02-17 | Sustained-release lipid preformulation and pharmaceutical composition for sustained-release injection in form of lipid solution containing same |
| MX2021009921A MX2021009921A (es) | 2019-02-18 | 2020-02-17 | Preformulacion de lipidos de liberacion sostenida y composicion farmacetica de liberacion sostenida inyectable en la forma de una solucion de lipidos que contiene a la misma. |
| EP20758601.7A EP3928762A4 (en) | 2019-02-18 | 2020-02-17 | DELAYED RELEASE LIPID PREFORMULATION AND PHARMACEUTICAL COMPOSITION FOR DELAYED RELEASE INJECTION IN THE FORM OF A LIPID SOLUTION THEREOF |
| CA3130252A CA3130252A1 (en) | 2019-02-18 | 2020-02-17 | Sustained-release lipid preformulation and pharmaceutical composition for sustained-release injection in form of lipid solution containing same |
| JP2021548193A JP7457727B2 (ja) | 2019-02-18 | 2020-02-17 | 徐放性脂質前製剤およびそれを含む脂質溶液の形態の徐放性注射用医薬組成物 |
| AU2020225991A AU2020225991A1 (en) | 2019-02-18 | 2020-02-17 | Sustained-release lipid preformulation and pharmaceutical composition for sustained-release injection in form of lipid solution containing same |
| PCT/KR2020/002182 WO2020171491A1 (ko) | 2019-02-18 | 2020-02-17 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
| CN202080015053.4A CN113490487B (zh) | 2019-02-18 | 2020-02-17 | 缓释型脂质预浓缩物及包含其的脂质溶液形式的缓释型注射用药物组合物 |
| KR1020200160620A KR102365844B1 (ko) | 2019-02-18 | 2020-11-26 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
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| KR1020190018619A KR102186704B1 (ko) | 2019-02-18 | 2019-02-18 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020200160620A Division KR102365844B1 (ko) | 2019-02-18 | 2020-11-26 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
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| KR20200100392A KR20200100392A (ko) | 2020-08-26 |
| KR102186704B1 true KR102186704B1 (ko) | 2020-12-04 |
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| KR1020190018619A KR102186704B1 (ko) | 2019-02-18 | 2019-02-18 | 서방성 지질 전구 제제 및 이를 포함하는 지질 용액 형태의 서방성 주사용 약학 조성물 |
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| Country | Link |
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| US (1) | US20220125888A1 (es) |
| EP (1) | EP3928762A4 (es) |
| JP (1) | JP7457727B2 (es) |
| KR (1) | KR102186704B1 (es) |
| CN (1) | CN113490487B (es) |
| AU (1) | AU2020225991A1 (es) |
| CA (1) | CA3130252A1 (es) |
| MX (1) | MX2021009921A (es) |
| WO (1) | WO2020171491A1 (es) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2023146187A1 (ko) * | 2022-01-27 | 2023-08-03 | 주식회사 티온랩테라퓨틱스 | 초기 방출 제어된 지질 융합 데포 조성물 및 이의 제조방법 |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115484935A (zh) * | 2020-02-14 | 2022-12-16 | G2G生物公司 | 包括含有glp-1类似物或其药学上可接受的盐的缓释微球的药物组合物 |
| WO2023080712A1 (ko) * | 2021-11-05 | 2023-05-11 | ㈜아이엠디팜 | 신규한 서방성 지질 전구 제제 및 이를 포함하는 서방성 주사용 약학 조성물 |
| CN117180281B (zh) * | 2023-11-08 | 2024-02-06 | 山东则正医药技术有限公司 | 棕榈酸帕利哌酮制剂及其制备方法和应用 |
Family Cites Families (11)
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|---|---|---|---|---|
| US5993850A (en) * | 1994-09-13 | 1999-11-30 | Skyepharma Inc. | Preparation of multivesicular liposomes for controlled release of encapsulated biologically active substances |
| ES2248908T7 (es) * | 1997-06-06 | 2014-11-24 | Depomed, Inc. | Formas de dosificación de fármacos por vía oral y retención gástrica para liberación continuada de fármacos altamente solubles |
| SE9703458D0 (sv) | 1997-09-25 | 1997-09-25 | Pharmacia & Upjohn Ab | Nicotine compositions and methods of formulation thereof |
| US20020102301A1 (en) * | 2000-01-13 | 2002-08-01 | Joseph Schwarz | Pharmaceutical solid self-emulsifying composition for sustained delivery of biologically active compounds and the process for preparation thereof |
| US8865021B2 (en) | 2003-11-07 | 2014-10-21 | Camurus Ab | Compositions of lipids and cationic peptides |
| DE602005008247D1 (de) | 2004-06-04 | 2008-08-28 | Camurus Ab | Flüssige depotformulierungen |
| KR101494594B1 (ko) * | 2011-08-30 | 2015-02-23 | 주식회사 종근당 | 약리학적 활성물질의 서방성 지질 초기제제 및 이를 포함하는 약제학적 조성물 |
| KR101586789B1 (ko) | 2012-12-28 | 2016-01-19 | 주식회사 종근당 | 양이온성 약리학적 활성물질의 서방성 지질 초기제제 및 이를 포함하는 약제학적 조성물 |
| KR101586790B1 (ko) * | 2012-12-28 | 2016-01-19 | 주식회사 종근당 | 음이온성 약리학적 활성물질의 서방성 지질 초기제제 및 이를 포함하는 약제학적 조성물 |
| CN106491519B (zh) * | 2016-12-09 | 2020-01-21 | 广州中大南沙科技创新产业园有限公司 | 局部麻醉药的立方液晶原位凝胶注射剂及其制备方法 |
| KR102096391B1 (ko) * | 2019-10-11 | 2020-04-06 | (주)아이엠디팜 | 액상결정 구조체를 형성하는 오메가-3-지방산 조성물 |
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2019
- 2019-02-18 KR KR1020190018619A patent/KR102186704B1/ko active IP Right Grant
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2020
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- 2020-02-17 JP JP2021548193A patent/JP7457727B2/ja active Active
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023146187A1 (ko) * | 2022-01-27 | 2023-08-03 | 주식회사 티온랩테라퓨틱스 | 초기 방출 제어된 지질 융합 데포 조성물 및 이의 제조방법 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2020171491A1 (ko) | 2020-08-27 |
| EP3928762A4 (en) | 2022-11-16 |
| EP3928762A1 (en) | 2021-12-29 |
| MX2021009921A (es) | 2021-10-13 |
| CN113490487B (zh) | 2023-04-18 |
| US20220125888A1 (en) | 2022-04-28 |
| CA3130252A1 (en) | 2020-08-27 |
| AU2020225991A1 (en) | 2021-09-02 |
| JP2022520858A (ja) | 2022-04-01 |
| JP7457727B2 (ja) | 2024-03-28 |
| KR20200100392A (ko) | 2020-08-26 |
| CN113490487A (zh) | 2021-10-08 |
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