KR102013567B1 - ６-(피페리딘-４-일옥시)-２ｈ-이소퀴놀린-１-온 하이드로클로라이드의 다형체 - Google Patents
６-(피페리딘-４-일옥시)-２ｈ-이소퀴놀린-１-온 하이드로클로라이드의 다형체 Download PDFInfo
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- KR102013567B1 KR102013567B1 KR1020147003355A KR20147003355A KR102013567B1 KR 102013567 B1 KR102013567 B1 KR 102013567B1 KR 1020147003355 A KR1020147003355 A KR 1020147003355A KR 20147003355 A KR20147003355 A KR 20147003355A KR 102013567 B1 KR102013567 B1 KR 102013567B1
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- South Korea
- Prior art keywords
- polymorph
- yloxy
- isoquinolin
- hydrochloride
- piperidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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| EP11305891.1 | 2011-07-08 | ||
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| EP11306034.7 | 2011-12-29 | ||
| EP11306034 | 2011-12-29 | ||
| PCT/EP2012/062444 WO2013007519A1 (en) | 2011-07-08 | 2012-06-27 | Polymorphs of 6-(piperidin-4-yloxy)-2h-isoquinolin-1-one hydrochloride |
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| KR20140046460A KR20140046460A (ko) | 2014-04-18 |
| KR102013567B1 true KR102013567B1 (ko) | 2019-08-23 |
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| CN109810173B (zh) * | 2017-11-21 | 2020-11-27 | 首都医科大学 | 二氢异喹啉-3-甲酰-TARGD(aa)aa,其制备,抗静脉血栓活性和应用 |
| CN119630643A (zh) * | 2022-08-01 | 2025-03-14 | 瓦洛健康公司 | 用于制备6-取代的-1-(2h)-异喹啉酮的方法和中间化合物 |
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| WO2008077550A1 (en) * | 2006-12-27 | 2008-07-03 | Sanofi-Aventis | Substituted isoquinoline and isoquinolinone derivatives as inhibitors of rho-kinase |
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| SK9742002A3 (en) * | 2000-01-07 | 2003-02-04 | Transform Pharmaceuticals Inc | High-throughput formation, identification, and analysis of diverse solid-forms |
| NZ565668A (en) * | 2005-07-26 | 2010-09-30 | Sanofi Aventis | Piperidinyl-substituted isoquinolone derivatives as RHO-kinase inhibitors |
| TW200738682A (en) | 2005-12-08 | 2007-10-16 | Organon Nv | Isoquinoline derivatives |
| BRPI0821837A2 (pt) * | 2007-12-26 | 2015-06-16 | Sanofi Aventis | Processo para a preparação de 6-substituídas-1-(2h)-isoquinolinonas |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| AU2012283277A1 (en) | 2014-02-27 |
| CY1117545T1 (el) | 2017-04-26 |
| HK1192234A1 (zh) | 2014-08-15 |
| KR20140046460A (ko) | 2014-04-18 |
| RU2014104357A (ru) | 2015-08-20 |
| SI2729461T1 (sl) | 2016-06-30 |
| JP2014518236A (ja) | 2014-07-28 |
| HRP20160358T1 (hr) | 2016-05-06 |
| ES2567317T3 (es) | 2016-04-21 |
| PL2729461T3 (pl) | 2016-06-30 |
| CA2843777C (en) | 2018-11-06 |
| EP2729461B1 (en) | 2016-01-20 |
| CN103781777A (zh) | 2014-05-07 |
| DK2729461T3 (en) | 2016-04-11 |
| CA2843777A1 (en) | 2013-01-17 |
| EP2729461A1 (en) | 2014-05-14 |
| HUE028550T2 (en) | 2016-12-28 |
| WO2013007519A1 (en) | 2013-01-17 |
| IN2014CN00834A (enExample) | 2015-04-03 |
| AU2012283277B2 (en) | 2016-07-21 |
| US20130012479A1 (en) | 2013-01-10 |
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