KR101054237B1 - 플리반세린 다형체 α를 함유하는 신규한 약제학적 조성물 - Google Patents
플리반세린 다형체 α를 함유하는 신규한 약제학적 조성물 Download PDFInfo
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- KR101054237B1 KR101054237B1 KR1020047018741A KR20047018741A KR101054237B1 KR 101054237 B1 KR101054237 B1 KR 101054237B1 KR 1020047018741 A KR1020047018741 A KR 1020047018741A KR 20047018741 A KR20047018741 A KR 20047018741A KR 101054237 B1 KR101054237 B1 KR 101054237B1
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Classifications
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02011224 | 2002-05-22 | ||
| EP02011224.9 | 2002-05-22 | ||
| PCT/EP2003/005226 WO2003097058A1 (en) | 2002-05-22 | 2003-05-19 | New pharmaceutical compositions containing flibanserin polymorph a |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20040111668A KR20040111668A (ko) | 2004-12-31 |
| KR101054237B1 true KR101054237B1 (ko) | 2011-08-08 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020047018741A KR101054237B1 (ko) | 2002-05-22 | 2003-05-19 | 플리반세린 다형체 α를 함유하는 신규한 약제학적 조성물 |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP1511489B1 (pt) |
| JP (1) | JP3919788B2 (pt) |
| KR (1) | KR101054237B1 (pt) |
| CN (3) | CN101002780A (pt) |
| AT (1) | ATE499939T1 (pt) |
| BR (1) | BRPI0311189B8 (pt) |
| CA (1) | CA2483597C (pt) |
| CY (1) | CY1111470T1 (pt) |
| DE (1) | DE60336225D1 (pt) |
| DK (1) | DK1511489T3 (pt) |
| EA (1) | EA007185B1 (pt) |
| EC (1) | ECSP045493A (pt) |
| ES (1) | ES2361994T3 (pt) |
| HR (1) | HRP20041092B1 (pt) |
| IL (1) | IL164440A0 (pt) |
| ME (1) | MEP55308A (pt) |
| MX (1) | MXPA04011487A (pt) |
| NO (1) | NO329414B1 (pt) |
| NZ (1) | NZ537253A (pt) |
| PL (1) | PL211062B1 (pt) |
| RS (1) | RS51718B (pt) |
| SI (1) | SI1511489T1 (pt) |
| UA (1) | UA80135C2 (pt) |
| WO (1) | WO2003097058A1 (pt) |
| ZA (1) | ZA200408151B (pt) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10675280B2 (en) | 2001-10-20 | 2020-06-09 | Sprout Pharmaceuticals, Inc. | Treating sexual desire disorders with flibanserin |
| UA78974C2 (en) | 2001-10-20 | 2007-05-10 | Boehringer Ingelheim Pharma | Use of flibanserin for treating disorders of sexual desire |
| US20050239798A1 (en) * | 2004-04-22 | 2005-10-27 | Boehringer Ingelheim Pharmaceuticals, Inc. | Method for the treatment of premenstrual and other female sexual disorders |
| WO2006096439A2 (en) * | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of schizophrenia and related diseases |
| EP1888071A1 (en) * | 2005-05-19 | 2008-02-20 | Boehringer Ingelheim International GmbH | Method for the treatment of drug-induced sexual dysfunction |
| JP2008540672A (ja) * | 2005-05-19 | 2008-11-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 病状に起因する性的機能不全の治療方法 |
| US8227476B2 (en) | 2005-08-03 | 2012-07-24 | Sprout Pharmaceuticals, Inc. | Use of flibanserin in the treatment of obesity |
| CA2626134C (en) | 2005-10-29 | 2013-12-24 | Boehringer Ingelheim International Gmbh | Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders |
| US20070105869A1 (en) * | 2005-11-08 | 2007-05-10 | Stephane Pollentier | Use of flibanserin for the treatment of pre-menopausal sexual desire disorders |
| WO2008000760A1 (en) | 2006-06-30 | 2008-01-03 | Boehringer Ingelheim International Gmbh | Flibanserin for the treatment of urinary incontinence and related diseases |
| EP2054041A2 (en) | 2006-08-14 | 2009-05-06 | Boehringer Ingelheim International GmbH | Formulations of flibanserin and method for manufacturing the same |
| CL2007002214A1 (es) | 2006-08-14 | 2008-03-07 | Boehringer Ingelheim Int | Composicion farmaceutica en la forma de comprimido, donde al menos la longitud del comprimido en el estado anterior de la aplicacion es al menos 7/12 del diametro pilorico del paciente y despues de ingerirlo en estado alimentado, la longitud del comp |
| AR062321A1 (es) | 2006-08-25 | 2008-10-29 | Boehringer Ingelheim Int | Sistema de liberacion controlada y metodo para fabricarlo |
| EP2097389B1 (en) | 2006-12-20 | 2011-09-14 | Boehringer Ingelheim International GmbH | Sulfated benzimidazolone derivatives having mixed serotonine receptor affinity |
| EP1955699A1 (en) * | 2007-02-08 | 2008-08-13 | Boehringer Ingelheim Pharma GmbH & Co. KG | Use of flibanserin for the treatment of insomnia |
| CL2008002693A1 (es) | 2007-09-12 | 2009-10-16 | Boehringer Ingelheim Int | Uso de flibanserina para el tratamiento de sintomas vasomotores seleccionados de sofocos, sudores nocturnos, cambios de estado de animo e irritabilidad |
| EP2090297A1 (en) * | 2008-02-13 | 2009-08-19 | Boehringer Ingelheim International GmbH | Formulations of flibanserin |
| DE102008047910A1 (de) | 2008-09-19 | 2010-03-25 | Molkerei Meggle Wasserburg Gmbh & Co. Kg | Tablettierhilfsstoff auf Laktose- und Cellulosebasis |
| US20120010216A1 (en) * | 2010-07-06 | 2012-01-12 | Brown Arthur M | Pharmaceutical compositions containing vanoxerine |
| CN104926734B (zh) * | 2015-07-07 | 2017-04-05 | 苏州立新制药有限公司 | 氟班色林的制备方法 |
| CN108699007A (zh) * | 2016-01-31 | 2018-10-23 | 孟晓明 | 氟班色林的新晶型及其制备方法及其用途 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0526434A1 (en) * | 1991-07-30 | 1993-02-03 | BOEHRINGER INGELHEIM ITALIA S.p.A. | Benzimidazolone derivatives as 5-HT1A and 5-HT2 antagonists |
| KR20040023704A (ko) * | 2001-08-02 | 2004-03-18 | 비다켐 에스. 피. 에이. | 플리반세린의 안정한 다형체, 이의 기술적 제조 방법 및약제 제조시 이의 용도 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10138273A1 (de) * | 2001-08-10 | 2003-02-27 | Boehringer Ingelheim Pharma | Arzneimittel mit neuroprotektiver Wirkung |
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2003
- 2003-05-19 WO PCT/EP2003/005226 patent/WO2003097058A1/en active Application Filing
- 2003-05-19 AT AT03730069T patent/ATE499939T1/de active
- 2003-05-19 CN CNA2007100014771A patent/CN101002780A/zh active Pending
- 2003-05-19 JP JP2004505057A patent/JP3919788B2/ja not_active Expired - Fee Related
- 2003-05-19 PL PL372457A patent/PL211062B1/pl unknown
- 2003-05-19 CN CNA038117029A patent/CN1655789A/zh active Pending
- 2003-05-19 CN CN201110122058XA patent/CN102240289A/zh active Pending
- 2003-05-19 RS YU98704A patent/RS51718B/en unknown
- 2003-05-19 SI SI200331994T patent/SI1511489T1/sl unknown
- 2003-05-19 BR BRPI0311189A patent/BRPI0311189B8/pt not_active IP Right Cessation
- 2003-05-19 ES ES03730069T patent/ES2361994T3/es not_active Expired - Lifetime
- 2003-05-19 ME MEP-553/08A patent/MEP55308A/xx unknown
- 2003-05-19 DE DE60336225T patent/DE60336225D1/de not_active Expired - Lifetime
- 2003-05-19 EP EP03730069A patent/EP1511489B1/en not_active Expired - Lifetime
- 2003-05-19 NZ NZ537253A patent/NZ537253A/en not_active IP Right Cessation
- 2003-05-19 DK DK03730069.6T patent/DK1511489T3/da active
- 2003-05-19 MX MXPA04011487A patent/MXPA04011487A/es active IP Right Grant
- 2003-05-19 UA UA20041210555A patent/UA80135C2/uk unknown
- 2003-05-19 EA EA200401515A patent/EA007185B1/ru not_active IP Right Cessation
- 2003-05-19 CA CA2483597A patent/CA2483597C/en not_active Expired - Fee Related
- 2003-05-19 KR KR1020047018741A patent/KR101054237B1/ko active IP Right Grant
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2004
- 2004-10-05 IL IL16444004A patent/IL164440A0/xx unknown
- 2004-10-08 ZA ZA200408151A patent/ZA200408151B/en unknown
- 2004-10-22 NO NO20044547A patent/NO329414B1/no not_active IP Right Cessation
- 2004-11-19 HR HRP20041092AA patent/HRP20041092B1/hr not_active IP Right Cessation
- 2004-12-13 EC EC2004005493A patent/ECSP045493A/es unknown
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- 2011-05-17 CY CY20111100475T patent/CY1111470T1/el unknown
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0526434A1 (en) * | 1991-07-30 | 1993-02-03 | BOEHRINGER INGELHEIM ITALIA S.p.A. | Benzimidazolone derivatives as 5-HT1A and 5-HT2 antagonists |
| KR20040023704A (ko) * | 2001-08-02 | 2004-03-18 | 비다켐 에스. 피. 에이. | 플리반세린의 안정한 다형체, 이의 기술적 제조 방법 및약제 제조시 이의 용도 |
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