KR100758620B1 - 4-알콕시 사이클로헥산-1 아미노 카복실산 에스테르 및그의 제조방법 - Google Patents

4-알콕시 사이클로헥산-1 아미노 카복실산 에스테르 및그의 제조방법 Download PDF

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KR100758620B1
KR100758620B1 KR1020027017196A KR20027017196A KR100758620B1 KR 100758620 B1 KR100758620 B1 KR 100758620B1 KR 1020027017196 A KR1020027017196 A KR 1020027017196A KR 20027017196 A KR20027017196 A KR 20027017196A KR 100758620 B1 KR100758620 B1 KR 100758620B1
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South Korea
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formula
iii
compound
cis
general formula
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Korean (ko)
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KR20030058944A (ko
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힘믈러토마스
피셔라이너
갈렌캄프베른트
크놉스한스-요아힘
물더루베르투스
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바이엘 크롭사이언스 아게
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Assigned to 바이엘 인텔렉쳐 프로퍼티 게엠베하 reassignment 바이엘 인텔렉쳐 프로퍼티 게엠베하 권리의 전부이전등록 Assignors: 바이엘 크롭사이언스 악티엔게젤샤프트
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/09—Geometrical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1020027017196A 2000-07-05 2001-06-22 4-알콕시 사이클로헥산-1 아미노 카복실산 에스테르 및그의 제조방법 Expired - Lifetime KR100758620B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10032587.4 2000-07-05
DE10032587A DE10032587A1 (de) 2000-07-05 2000-07-05 4-Alkoxy-cyclohexan-1-amino-carbonsäureester und Verfahren zu ihrer Herstellung
PCT/EP2001/007115 WO2002002532A1 (de) 2000-07-05 2001-06-22 4-alkoxy-cyclohexan-1-amino-carbonsäureester und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
KR20030058944A KR20030058944A (ko) 2003-07-07
KR100758620B1 true KR100758620B1 (ko) 2007-09-13

Family

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Family Applications (1)

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KR1020027017196A Expired - Lifetime KR100758620B1 (ko) 2000-07-05 2001-06-22 4-알콕시 사이클로헥산-1 아미노 카복실산 에스테르 및그의 제조방법

Country Status (15)

Country Link
US (3) US7148377B2 (https=)
EP (1) EP1309562B1 (https=)
JP (5) JP5127106B2 (https=)
KR (1) KR100758620B1 (https=)
CN (2) CN1286820C (https=)
AT (1) ATE394379T1 (https=)
AU (1) AU2001272504A1 (https=)
BR (1) BR0112245B1 (https=)
DE (2) DE10032587A1 (https=)
DK (1) DK1309562T3 (https=)
ES (1) ES2305090T3 (https=)
IL (3) IL153561A0 (https=)
MX (1) MXPA02012889A (https=)
WO (1) WO2002002532A1 (https=)
ZA (1) ZA200300005B (https=)

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DE10032587A1 (de) * 2000-07-05 2002-01-17 Bayer Ag 4-Alkoxy-cyclohexan-1-amino-carbonsäureester und Verfahren zu ihrer Herstellung
DE10213051B4 (de) * 2002-03-23 2013-03-07 Grünenthal GmbH Substituierte 4-Aminocyclohexanole
DE10231333A1 (de) * 2002-07-11 2004-01-22 Bayer Cropscience Ag Cis-Alkoxysubstituierte spirocyclische 1-H-Pyrrolidin-2,4-dion-Derivate
DE10239479A1 (de) * 2002-08-28 2004-03-04 Bayer Cropscience Ag Substituierte spirocyclische Ketoenole
DE10241062A1 (de) * 2002-09-05 2003-11-27 Bosch Gmbh Robert Strukturkörper mit einem elektrochemisch erzeugten porösen Bereich
DE102006057037A1 (de) * 2006-12-04 2008-06-05 Bayer Cropscience Ag cis-Alkoxyspirocyclische biphenylsubstituierte Tetramsäure-Derivate
BR112013018973A2 (pt) 2011-01-25 2017-09-19 Bayer Ip Gmbh processo para a preparação de derivados de 1-h-pirrolidina-2,4-diona
BR112013021021A2 (pt) 2011-02-17 2016-08-02 Bayer Ip Gmbh 3- (bifenil - 3 - il) - 8, 8 - difluoro - 4 - hidroxi - 1 - azaspiro [4, 5] dec - 3 - eno - 2 - onas substituídas para terapia e cetoenóis espirocíclicos substituídos com halogéneo
DE102011080405A1 (de) 2011-08-04 2013-02-07 Bayer Pharma AG Substituierte 3-(Biphenyl-3-yl)-8,8-difluor-4-hydroxy-1-azaspiro[4.5]dec-3-en-2-one zur Therapie
CN103429573B (zh) * 2011-03-11 2016-01-20 拜耳知识产权有限责任公司 顺式-烷氧基取代的螺环1h-吡咯烷-2,4-二酮衍生物
DE102011080406A1 (de) 2011-08-04 2013-02-07 Bayer Pharma AG Substituierte 3-(Biphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro8[4.5]dec-3-en-2-one
TWI579260B (zh) * 2012-03-28 2017-04-21 拜耳智慧財產有限公司 用於製備順式－烷氧基－取代之螺環狀苯基乙醯基胺基酸酯及順式－烷氧基－取代之螺環狀１ｈ－吡咯啶－２，４－二酮衍生物之方法
US9751865B2 (en) 2013-12-23 2017-09-05 Syngenta Limited Dihydro-hydantoin derivatives with herbicidal activity
CN107857722A (zh) * 2017-11-21 2018-03-30 河南紫微星化学有限公司 一种螺虫乙酯的新型制备方法
CN110128288B (zh) * 2018-02-02 2023-07-28 浙江九洲药业股份有限公司 一种氨基取代的环戊烷甲酸烷基酯衍生物的制备方法
CN111574389B (zh) * 2020-05-14 2023-08-18 河北威远生物化工有限公司 1-氨基-4-取代环己基羧酸及其盐的顺式异构体的制备方法
CN120957968A (zh) 2023-04-07 2025-11-14 安道麦马克西姆有限公司 由环状氨基酸合成环酮
WO2025150038A1 (en) * 2024-01-09 2025-07-17 Adama Makhteshim Ltd. A method for separation of cis and trans isomers of hydantoin-containing spiro-compound from an isomeric mixture

Citations (2)

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WO1997017092A1 (en) * 1995-11-09 1997-05-15 Emory University Amino acid analogs for tumor imaging
WO1998056387A1 (en) * 1997-06-10 1998-12-17 Unisearch Limited Method of treatment of liver tumours and pharmaceutical compositions for use therein

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JPS5523822B2 (https=) 1971-12-14 1980-06-25
AU666040B2 (en) * 1992-10-28 1996-01-25 Bayer Aktiengesellschaft Substituted 1-H-3-aryl-pyrrolidine-2,4-dione derivatives
DE4425617A1 (de) * 1994-01-28 1995-08-03 Bayer Ag 1-H-3-Aryl-pyrrolidin-2,4-dion-Derivate
DE4431730A1 (de) * 1994-02-09 1995-08-10 Bayer Ag Substituierte 1H-3-Aryl-pyrrolidin-2,4-dion-Derivate
ES2190786T3 (es) * 1994-04-05 2003-08-16 Bayer Cropscience Ag 1-h-3-aril-pirrolidin-2,4-dionas alcoxi-alquil-substituidas como herbicidas y pesticidas.
US6358887B1 (en) * 1995-02-13 2002-03-19 Bayer Aktiengesellschaft 2-Phenyl-substituted heterocyclic 1,3-ketonols as herbicides and pesticides
CN1131209C (zh) * 1995-05-09 2003-12-17 拜尔公司 可用作杀虫剂和除草剂的烷基－二卤代苯基取代的酮烯醇
MX9710373A (es) * 1995-06-28 1998-07-31 Bayer Ag Fenilcetoenoles 2,4,5-trisubstituidos para el empleo como pesticidas y herbicidas.
CN1152860C (zh) * 1995-06-30 2004-06-09 拜尔公司 二烷基-卤代苯基取代的酮-烯醇
CN1215390A (zh) * 1996-04-02 1999-04-28 拜尔公司 取代的苯基酮烯醇杀虫剂及除草剂
ES2275796T3 (es) * 1996-08-05 2007-06-16 Bayer Cropscience Ag Fenilcetoenoles 2- y 2,5-substituidos.
DE10032587A1 (de) * 2000-07-05 2002-01-17 Bayer Ag 4-Alkoxy-cyclohexan-1-amino-carbonsäureester und Verfahren zu ihrer Herstellung
US6380426B1 (en) * 2001-09-26 2002-04-30 Council Of Scientific And Industrial Research Process for the preparation of a carboxylic acid

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997017092A1 (en) * 1995-11-09 1997-05-15 Emory University Amino acid analogs for tumor imaging
WO1998056387A1 (en) * 1997-06-10 1998-12-17 Unisearch Limited Method of treatment of liver tumours and pharmaceutical compositions for use therein

Also Published As

Publication number Publication date
CN1286820C (zh) 2006-11-29
EP1309562A1 (de) 2003-05-14
JP2012255027A (ja) 2012-12-27
MXPA02012889A (es) 2004-07-30
BR0112245A (pt) 2003-06-24
IL153561A0 (en) 2003-07-06
ZA200300005B (en) 2004-01-02
CN1616436A (zh) 2005-05-18
AU2001272504A1 (en) 2002-01-14
WO2002002532A1 (de) 2002-01-10
US20090156402A1 (en) 2009-06-18
US7511153B2 (en) 2009-03-31
DK1309562T3 (da) 2008-08-11
JP5127106B2 (ja) 2013-01-23
BR0112245B1 (pt) 2013-09-10
US7803967B2 (en) 2010-09-28
US20070043219A1 (en) 2007-02-22
JP5899091B2 (ja) 2016-04-06
DE10032587A1 (de) 2002-01-17
EP1309562B1 (de) 2008-05-07
JP2004502678A (ja) 2004-01-29
IL153561A (en) 2008-08-07
US7148377B2 (en) 2006-12-12
ES2305090T3 (es) 2008-11-01
JP5899092B2 (ja) 2016-04-06
DE50113943D1 (de) 2008-06-19
IL190905A (en) 2010-05-31
CN1183118C (zh) 2005-01-05
JP5805561B2 (ja) 2015-11-04
HK1057897A1 (en) 2004-04-23
JP2012107076A (ja) 2012-06-07
US20040039223A1 (en) 2004-02-26
JP2014167018A (ja) 2014-09-11
ATE394379T1 (de) 2008-05-15
CN1436176A (zh) 2003-08-13
JP2012255028A (ja) 2012-12-27
KR20030058944A (ko) 2003-07-07
IL190905A0 (en) 2008-11-03

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