KR100568657B1 - 6,9-이치환 2-[트랜스-(4-아미노시클로헥실)아미노]퓨린 - Google Patents

6,9-이치환 2-[트랜스-(4-아미노시클로헥실)아미노]퓨린 Download PDF

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Publication number
KR100568657B1
KR100568657B1 KR1020007009424A KR20007009424A KR100568657B1 KR 100568657 B1 KR100568657 B1 KR 100568657B1 KR 1020007009424 A KR1020007009424 A KR 1020007009424A KR 20007009424 A KR20007009424 A KR 20007009424A KR 100568657 B1 KR100568657 B1 KR 100568657B1
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KR
South Korea
Prior art keywords
formula
group
integer
alkyl
amino
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KR1020007009424A
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English (en)
Korean (ko)
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KR20010041318A (ko
Inventor
제니퍼 에이. 듀몬트
알란 제이. 비톤티
데이비드 알. 보르셔딩
노톤 피. 피트
에이치. 란달 먼슨
패트릭 더블유. 케이. 셤
Original Assignee
아벤티스 파마슈티칼스 인크
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Publication of KR20010041318A publication Critical patent/KR20010041318A/ko
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Publication of KR100568657B1 publication Critical patent/KR100568657B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020007009424A 1998-02-26 1999-02-18 6,9-이치환 2-[트랜스-(4-아미노시클로헥실)아미노]퓨린 KR100568657B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3097598A 1998-02-26 1998-02-26
US09/030,975 1998-02-26

Publications (2)

Publication Number Publication Date
KR20010041318A KR20010041318A (ko) 2001-05-15
KR100568657B1 true KR100568657B1 (ko) 2006-04-07

Family

ID=21856977

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020007009424A KR100568657B1 (ko) 1998-02-26 1999-02-18 6,9-이치환 2-[트랜스-(4-아미노시클로헥실)아미노]퓨린

Country Status (14)

Country Link
KR (1) KR100568657B1 (es)
AR (1) AR018121A1 (es)
AT (1) ATE252583T1 (es)
DE (1) DE69912248T2 (es)
DK (1) DK1056744T3 (es)
ES (1) ES2207182T3 (es)
HK (1) HK1030949A1 (es)
ID (1) ID25444A (es)
NZ (1) NZ506235A (es)
OA (1) OA11455A (es)
PT (1) PT1056744E (es)
RU (1) RU2200162C2 (es)
TW (1) TWI225060B (es)
UA (1) UA66840C2 (es)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997016452A1 (en) * 1995-11-01 1997-05-09 Novartis Ag Purine derivatives and processes for their preparation
WO1997020842A1 (fr) * 1995-12-01 1997-06-12 Centre National De La Recherche Scientifique (C.N.R.S.) Nouveaux derives de purine possedant notamment des proprietes anti-proliferatives et leurs applications biologiques

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997016452A1 (en) * 1995-11-01 1997-05-09 Novartis Ag Purine derivatives and processes for their preparation
WO1997020842A1 (fr) * 1995-12-01 1997-06-12 Centre National De La Recherche Scientifique (C.N.R.S.) Nouveaux derives de purine possedant notamment des proprietes anti-proliferatives et leurs applications biologiques

Also Published As

Publication number Publication date
KR20010041318A (ko) 2001-05-15
ATE252583T1 (de) 2003-11-15
RU2200162C2 (ru) 2003-03-10
PT1056744E (pt) 2004-03-31
TWI225060B (en) 2004-12-11
UA66840C2 (uk) 2004-06-15
NZ506235A (en) 2003-02-28
DE69912248T2 (de) 2004-04-22
ID25444A (id) 2000-10-05
ES2207182T3 (es) 2004-05-16
OA11455A (en) 2003-12-05
DK1056744T3 (da) 2004-02-23
HK1030949A1 (en) 2001-05-25
DE69912248D1 (de) 2003-11-27
AR018121A1 (es) 2001-10-31

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