JPWO2024024760A1 - - Google Patents
Info
- Publication number
- JPWO2024024760A1 JPWO2024024760A1 JP2024537730A JP2024537730A JPWO2024024760A1 JP WO2024024760 A1 JPWO2024024760 A1 JP WO2024024760A1 JP 2024537730 A JP2024537730 A JP 2024537730A JP 2024537730 A JP2024537730 A JP 2024537730A JP WO2024024760 A1 JPWO2024024760 A1 JP WO2024024760A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
- C07D231/24—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms having sulfone or sulfonic acid radicals in the molecule
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
- C07H7/06—Heterocyclic radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022118259 | 2022-07-25 | ||
| JP2022118259 | 2022-07-25 | ||
| PCT/JP2023/027102 WO2024024760A1 (ja) | 2022-07-25 | 2023-07-25 | ピラゾロン化合物及びピラゾロン化剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2024024760A1 true JPWO2024024760A1 (https=) | 2024-02-01 |
| JPWO2024024760A5 JPWO2024024760A5 (https=) | 2024-11-12 |
| JP7782046B2 JP7782046B2 (ja) | 2025-12-08 |
Family
ID=89706371
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024537730A Active JP7782046B2 (ja) | 2022-07-25 | 2023-07-25 | ピラゾロン化合物及びピラゾロン化剤 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20250129030A1 (https=) |
| EP (1) | EP4563572A1 (https=) |
| JP (1) | JP7782046B2 (https=) |
| WO (1) | WO2024024760A1 (https=) |
Citations (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5980470A (ja) * | 1982-10-29 | 1984-05-09 | Konishiroku Photo Ind Co Ltd | オキソノ−ル染料の製造方法 |
| JPH03289653A (ja) * | 1990-04-06 | 1991-12-19 | Konica Corp | ハロゲン化銀カラー写真感光材料 |
| JPH0485538A (ja) * | 1990-07-28 | 1992-03-18 | Konica Corp | ハロゲン化銀カラー写真感光材料 |
| JPH08229302A (ja) * | 1995-02-24 | 1996-09-10 | Konica Corp | 固体微粒子の製造方法および製造装置 |
| JP2003059547A (ja) * | 2001-08-17 | 2003-02-28 | Nippon Kayaku Co Ltd | 色素増感光電変換素子 |
| JP2005015750A (ja) * | 2003-06-24 | 2005-01-20 | Yamada Chem Co Ltd | ペリミジン化合物 |
| WO2006129583A1 (ja) * | 2005-05-30 | 2006-12-07 | Genecare Research Institute Co., Ltd. | ピラゾロン誘導体 |
| WO2006129587A1 (ja) * | 2005-05-30 | 2006-12-07 | Genecare Research Institute Co., Ltd. | ピラゾロン誘導体を含有する医薬組成物 |
| JP2009093909A (ja) * | 2007-10-09 | 2009-04-30 | Konica Minolta Business Technologies Inc | 色素増感光電変換素子及びその製造方法 |
| CN110128345A (zh) * | 2019-05-13 | 2019-08-16 | 上海大学 | 一种吡唑酮衍生物的制备方法 |
-
2023
- 2023-07-25 WO PCT/JP2023/027102 patent/WO2024024760A1/ja not_active Ceased
- 2023-07-25 US US18/834,041 patent/US20250129030A1/en active Pending
- 2023-07-25 EP EP23846490.3A patent/EP4563572A1/en active Pending
- 2023-07-25 JP JP2024537730A patent/JP7782046B2/ja active Active
Patent Citations (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5980470A (ja) * | 1982-10-29 | 1984-05-09 | Konishiroku Photo Ind Co Ltd | オキソノ−ル染料の製造方法 |
| JPH03289653A (ja) * | 1990-04-06 | 1991-12-19 | Konica Corp | ハロゲン化銀カラー写真感光材料 |
| JPH0485538A (ja) * | 1990-07-28 | 1992-03-18 | Konica Corp | ハロゲン化銀カラー写真感光材料 |
| JPH08229302A (ja) * | 1995-02-24 | 1996-09-10 | Konica Corp | 固体微粒子の製造方法および製造装置 |
| JP2003059547A (ja) * | 2001-08-17 | 2003-02-28 | Nippon Kayaku Co Ltd | 色素増感光電変換素子 |
| JP2005015750A (ja) * | 2003-06-24 | 2005-01-20 | Yamada Chem Co Ltd | ペリミジン化合物 |
| WO2006129583A1 (ja) * | 2005-05-30 | 2006-12-07 | Genecare Research Institute Co., Ltd. | ピラゾロン誘導体 |
| WO2006129587A1 (ja) * | 2005-05-30 | 2006-12-07 | Genecare Research Institute Co., Ltd. | ピラゾロン誘導体を含有する医薬組成物 |
| JP2009093909A (ja) * | 2007-10-09 | 2009-04-30 | Konica Minolta Business Technologies Inc | 色素増感光電変換素子及びその製造方法 |
| CN110128345A (zh) * | 2019-05-13 | 2019-08-16 | 上海大学 | 一种吡唑酮衍生物的制备方法 |
Non-Patent Citations (3)
| Title |
|---|
| ANGELASTRO, ANTONIO ET AL.: "Galactose Oxidase Enables Modular Assembly of Conjugates from Native Antibodies with High Drug-to- A", CHEMSUSCHEM, vol. 15, e202102592, JPN6023042286, 20 January 2022 (2022-01-20), pages 1 - 4, ISSN: 0005738795 * |
| JANSON, NILS ET AL.: "Bifunctional Reagents for Formylglycine Conjugation: Pitfalls and Breakthroughs", CHEMBIOCHEM, vol. 21, JPN6023042285, 18 September 2020 (2020-09-18), pages 3580 - 3593, ISSN: 0005738794 * |
| KUDIRKA, ROMAS A. ET AL.: "Site-Specific Tandem Knoevenagel Condensation-Michael Addition To Generate Antibody-Drug Conjugates", ACS MED. CHEM. LETT., vol. 7, JPN6023042284, 30 August 2016 (2016-08-30), pages 994 - 998, ISSN: 0005738793 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4563572A1 (en) | 2025-06-04 |
| WO2024024760A1 (ja) | 2024-02-01 |
| US20250129030A1 (en) | 2025-04-24 |
| JP7782046B2 (ja) | 2025-12-08 |
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