JPWO2023214577A5 - - Google Patents
Info
- Publication number
- JPWO2023214577A5 JPWO2023214577A5 JP2024519230A JP2024519230A JPWO2023214577A5 JP WO2023214577 A5 JPWO2023214577 A5 JP WO2023214577A5 JP 2024519230 A JP2024519230 A JP 2024519230A JP 2024519230 A JP2024519230 A JP 2024519230A JP WO2023214577 A5 JPWO2023214577 A5 JP WO2023214577A5
- Authority
- JP
- Japan
- Prior art keywords
- peptide
- protecting group
- solvent
- amino acid
- sulfoxide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022075743 | 2022-05-02 | ||
| PCT/JP2023/017114 WO2023214577A1 (ja) | 2022-05-02 | 2023-05-02 | ジケトピペラジン形成による欠損を抑制するペプチド合成方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2023214577A1 JPWO2023214577A1 (https=) | 2023-11-09 |
| JPWO2023214577A5 true JPWO2023214577A5 (https=) | 2026-03-06 |
Family
ID=88646535
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024519230A Pending JPWO2023214577A1 (https=) | 2022-05-02 | 2023-05-02 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20250353875A1 (https=) |
| EP (1) | EP4509517A1 (https=) |
| JP (1) | JPWO2023214577A1 (https=) |
| KR (1) | KR20250006193A (https=) |
| CN (1) | CN119213009A (https=) |
| TW (1) | TW202409059A (https=) |
| WO (1) | WO2023214577A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202446781A (zh) | 2011-12-28 | 2024-12-01 | 日商中外製藥股份有限公司 | 胜肽化合物之製造方法 |
| KR20250007021A (ko) | 2017-06-09 | 2025-01-13 | 추가이 세이야쿠 가부시키가이샤 | N-치환 아미노산을 포함하는 펩타이드의 합성 방법 |
| BR112022007535A2 (pt) | 2019-11-07 | 2022-07-12 | Chugai Pharmaceutical Co Ltd | Composto peptídico cíclico tendo ação inibitória de kras |
| EP4056580A4 (en) | 2019-11-07 | 2023-12-06 | Chugai Seiyaku Kabushiki Kaisha | METHOD FOR PRODUCING A PEPTIDE COMPOUND COMPRISING A STERICALLY HINDERED AMINO ACID |
| US12312379B2 (en) | 2021-05-07 | 2025-05-27 | Chugai Seiyaku Kabushiki Kaisha | Methods for producing cyclic compounds comprising N-substituted amino acid residues |
| JP7823181B2 (ja) | 2022-05-06 | 2026-03-03 | 中外製薬株式会社 | Ｈｒａｓおよびｎｒａｓに対して選択的なｋｒａｓ阻害作用を有する環状化合物 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6112011B2 (ja) * | 2011-05-31 | 2017-04-12 | 味の素株式会社 | ペプチドの製造方法 |
| TW202446781A (zh) | 2011-12-28 | 2024-12-01 | 日商中外製藥股份有限公司 | 胜肽化合物之製造方法 |
| WO2018021233A1 (ja) * | 2016-07-25 | 2018-02-01 | 積水メディカル株式会社 | 新規キサンテン保護剤 |
| CN110869544B (zh) | 2017-06-09 | 2024-03-08 | 中外制药株式会社 | 膜透过性高的环状肽化合物及包含其的文库 |
| KR20250007021A (ko) | 2017-06-09 | 2025-01-13 | 추가이 세이야쿠 가부시키가이샤 | N-치환 아미노산을 포함하는 펩타이드의 합성 방법 |
| EP3730497B1 (en) * | 2017-12-19 | 2022-11-16 | Sekisui Medical Co., Ltd. | Novel alkyl diphenylmethane protection agent |
| EP4056580A4 (en) | 2019-11-07 | 2023-12-06 | Chugai Seiyaku Kabushiki Kaisha | METHOD FOR PRODUCING A PEPTIDE COMPOUND COMPRISING A STERICALLY HINDERED AMINO ACID |
| KR20230097018A (ko) | 2020-11-05 | 2023-06-30 | 추가이 세이야쿠 가부시키가이샤 | 다이케토피페라진 형성에 의한 결손을 억제하는 펩타이드 합성 방법 |
| JP7063409B1 (ja) * | 2021-07-02 | 2022-05-09 | ペプチスター株式会社 | Ｆｍоｃ基を除去する方法 |
| JP7063408B1 (ja) * | 2021-07-02 | 2022-05-09 | ペプチスター株式会社 | 液相ペプチド製造方法 |
-
2023
- 2023-05-02 US US18/860,859 patent/US20250353875A1/en active Pending
- 2023-05-02 TW TW112116267A patent/TW202409059A/zh unknown
- 2023-05-02 EP EP23799506.3A patent/EP4509517A1/en active Pending
- 2023-05-02 KR KR1020247038699A patent/KR20250006193A/ko active Pending
- 2023-05-02 CN CN202380036194.8A patent/CN119213009A/zh active Pending
- 2023-05-02 JP JP2024519230A patent/JPWO2023214577A1/ja active Pending
- 2023-05-02 WO PCT/JP2023/017114 patent/WO2023214577A1/ja not_active Ceased
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