JPWO2023106310A5 - - Google Patents

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Publication number
JPWO2023106310A5
JPWO2023106310A5 JP2023566327A JP2023566327A JPWO2023106310A5 JP WO2023106310 A5 JPWO2023106310 A5 JP WO2023106310A5 JP 2023566327 A JP2023566327 A JP 2023566327A JP 2023566327 A JP2023566327 A JP 2023566327A JP WO2023106310 A5 JPWO2023106310 A5 JP WO2023106310A5
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JP
Japan
Prior art keywords
substituted
unsubstituted
pharmaceutically acceptable
acceptable salt
alkyl
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Pending
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JP2023566327A
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English (en)
Japanese (ja)
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JPWO2023106310A1 (https=
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Priority claimed from PCT/JP2022/045016 external-priority patent/WO2023106310A1/ja
Publication of JPWO2023106310A1 publication Critical patent/JPWO2023106310A1/ja
Publication of JPWO2023106310A5 publication Critical patent/JPWO2023106310A5/ja
Pending legal-status Critical Current

Links

JP2023566327A 2021-12-07 2022-12-07 Pending JPWO2023106310A1 (https=)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2021198891 2021-12-07
JP2022148916 2022-09-20
PCT/JP2022/045016 WO2023106310A1 (ja) 2021-12-07 2022-12-07 Glp-1受容体アゴニスト活性を有する芳香族複素環誘導体

Publications (2)

Publication Number Publication Date
JPWO2023106310A1 JPWO2023106310A1 (https=) 2023-06-15
JPWO2023106310A5 true JPWO2023106310A5 (https=) 2025-11-18

Family

ID=86730498

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023566327A Pending JPWO2023106310A1 (https=) 2021-12-07 2022-12-07

Country Status (2)

Country Link
JP (1) JPWO2023106310A1 (https=)
WO (1) WO2023106310A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT4408840T (pt) 2021-09-27 2025-10-07 Terns Pharmaceuticals Inc Ácidos benzimidazolocarboxílicos como agonistas de glp-1r
CN118401519A (zh) 2021-10-25 2024-07-26 拓臻制药公司 作为glp-1r激动剂的化合物
CN119095843A (zh) 2022-02-23 2024-12-06 拓臻制药公司 作为glp-1r激动剂的化合物
EP4568664B1 (en) 2023-04-07 2026-04-01 Terns Pharmaceuticals, Inc. Combination comprising a thr-beta agonist and a glp-1r agonist for use in treating obesity
CN120981457A (zh) 2023-09-14 2025-11-18 歌礼制药(中国)有限公司 Glp-1r激动剂及其治疗方法
TW202521534A (zh) 2023-11-24 2025-06-01 香港商歌禮製藥(中國)有限公司 Glp-1r 激動劑及其治療方法
TW202600132A (zh) 2024-03-08 2026-01-01 美商安尼波那生物公司 用於治療肥胖症及提高減重之方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102314286B1 (ko) * 2016-12-16 2021-10-21 화이자 인코포레이티드 Glp-1 수용체 작용제 및 이의 용도
AR111199A1 (es) * 2017-03-31 2019-06-12 Takeda Pharmaceuticals Co Compuesto aromático agonista de gpr40
WO2018181847A1 (ja) * 2017-03-31 2018-10-04 武田薬品工業株式会社 芳香環化合物
US10934279B2 (en) * 2018-06-13 2021-03-02 Pfizer Inc. GLP-1 receptor agonists and uses thereof
EP3953344A4 (en) * 2019-04-12 2023-08-09 Qilu Regor Therapeutics Inc. GLP-IR AGONISTS AND THEIR USES
JP2023537501A (ja) * 2020-08-06 2023-09-01 ガシャーブラム・バイオ・インコーポレイテッド ヘテロ環glp-1アゴニスト
JP7772778B2 (ja) * 2021-03-24 2025-11-18 塩野義製薬株式会社 縮合環を有するglp-1受容体作動薬を含有する医薬組成物
WO2022219495A1 (en) * 2021-04-12 2022-10-20 Novartis Ag 2-((4-((s)-2-(4-chloro-2-fluorophenyl)-2-methylbenzo[d][1,3]dioxol-4-yl)piperidin-1-yl)methyl)-1-(((s)-oxetan-2-yl)methyl)-1h-imidazole derivatives as activators of the glp1 receptor for the treatment of obesity
CN117177970A (zh) * 2021-04-30 2023-12-05 上海翰森生物医药科技有限公司 多环类衍生物调节剂、其制备方法和应用

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