JPWO2022101633A5 - - Google Patents

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JPWO2022101633A5
JPWO2022101633A5 JP2023528449A JP2023528449A JPWO2022101633A5 JP WO2022101633 A5 JPWO2022101633 A5 JP WO2022101633A5 JP 2023528449 A JP2023528449 A JP 2023528449A JP 2023528449 A JP2023528449 A JP 2023528449A JP WO2022101633 A5 JPWO2022101633 A5 JP WO2022101633A5
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JP
Japan
Prior art keywords
seq
referred
acceptable salt
peptide ligand
pharma
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JP2023528449A
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English (en)
Japanese (ja)
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JP2023549229A (ja
JP2023549229A5 (https=
JP7848202B2 (ja
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Priority claimed from GBGB2017927.1A external-priority patent/GB202017927D0/en
Priority claimed from GBGB2106903.4A external-priority patent/GB202106903D0/en
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Priority claimed from PCT/GB2021/052927 external-priority patent/WO2022101633A1/en
Publication of JP2023549229A publication Critical patent/JP2023549229A/ja
Publication of JP2023549229A5 publication Critical patent/JP2023549229A5/ja
Publication of JPWO2022101633A5 publication Critical patent/JPWO2022101633A5/ja
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Publication of JP7848202B2 publication Critical patent/JP7848202B2/ja
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JP2023528449A 2020-11-13 2021-11-12 トランスフェリン受容体1(TfR1)に特異的な二環式ペプチドリガンド Active JP7848202B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB2017927.1 2020-11-13
GBGB2017927.1A GB202017927D0 (en) 2020-11-13 2020-11-13 Bicyclic peptide ligands specific for transferrin
GB2106903.4 2021-05-14
GBGB2106903.4A GB202106903D0 (en) 2021-05-14 2021-05-14 Bicycle peptide ligands specific for transferrin
US202163261820P 2021-09-29 2021-09-29
US63/261,820 2021-09-29
PCT/GB2021/052927 WO2022101633A1 (en) 2020-11-13 2021-11-12 BICYCLIC PEPTIDE LIGANDS SPECIFIC FOR TRANSFERRIN RECEPTOR 1 (TfR1)

Publications (4)

Publication Number Publication Date
JP2023549229A JP2023549229A (ja) 2023-11-22
JP2023549229A5 JP2023549229A5 (https=) 2024-11-21
JPWO2022101633A5 true JPWO2022101633A5 (https=) 2024-11-21
JP7848202B2 JP7848202B2 (ja) 2026-04-20

Family

ID=81600834

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023528449A Active JP7848202B2 (ja) 2020-11-13 2021-11-12 トランスフェリン受容体1(TfR1)に特異的な二環式ペプチドリガンド

Country Status (12)

Country Link
US (3) US11970555B2 (https=)
EP (1) EP4244235A1 (https=)
JP (1) JP7848202B2 (https=)
KR (1) KR20230107589A (https=)
CN (1) CN116802190A (https=)
AR (1) AR126029A1 (https=)
AU (1) AU2021376917A1 (https=)
CA (1) CA3201414A1 (https=)
IL (1) IL302713A (https=)
MX (1) MX2023005624A (https=)
SA (1) SA523440745B1 (https=)
WO (1) WO2022101633A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL302713A (en) 2020-11-13 2023-07-01 Bicycletx Ltd Bicyclic peptide ligands specific for transferrin receptor 1 (TfR1)
GB202206431D0 (en) * 2022-05-03 2022-06-15 Bicycletx Ltd Bicyclic peptide ligands specific for transferrin receptor 1 (TfR1)
KR20260021596A (ko) * 2023-04-05 2026-02-13 아이오니스 파마수티컬즈, 인코포레이티드 Pln 발현을 감소시키는 화합물 및 방법
WO2025073871A1 (en) 2023-10-03 2025-04-10 Bicycletx Limited Bicyclic peptide ligand complexes specific for tfr1
GB202316970D0 (en) * 2023-11-06 2023-12-20 Bicycletx Ltd Bicyclic peptide ligands specific for transferrin receptor 1 (TfR1)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2009211253B2 (en) 2008-02-05 2014-11-06 Bicyclerd Limited Methods and compositions
GB0914110D0 (en) * 2009-08-12 2009-09-16 Medical Res Council Peptide libraries
WO2016077840A2 (en) * 2014-11-14 2016-05-19 Ossianix, Inc. TfR SELECTIVE BINDING COMPOUNDS AND RELATED METHODS
CN104650186A (zh) 2015-03-09 2015-05-27 中国药科大学 一种能够与TfR1特异性结合的活性肽及其应用
GB201706477D0 (en) * 2017-04-24 2017-06-07 Bicycle Therapeutics Ltd Modification of polypeptides
WO2018197893A1 (en) 2017-04-27 2018-11-01 Bicycletx Limited Bicyclic peptide ligands and uses thereof
CN111183147B (zh) * 2017-08-04 2024-07-05 拜斯科技术开发有限公司 Cd137特异性的双环肽配体
CA3080351A1 (en) * 2017-11-02 2019-05-09 Ossianix, Inc. Improved tfr-selective binding peptides capable of crossing the blood brain barrier
JP2021514953A (ja) * 2018-02-23 2021-06-17 バイスクルテクス・リミテッド 多量体二環式ペプチドリガンド
WO2020084305A1 (en) * 2018-10-23 2020-04-30 Bicycletx Limited Bicyclic peptide ligands and uses thereof
JP2022514618A (ja) * 2018-12-21 2022-02-14 バイスクルテクス・リミテッド Pd-l1に特異的な二環式ペプチドリガンド
GB201912320D0 (en) * 2019-08-28 2019-10-09 Bicycletx Ltd PBP Binding Bicyclic Peptide Ligands
IL302713A (en) 2020-11-13 2023-07-01 Bicycletx Ltd Bicyclic peptide ligands specific for transferrin receptor 1 (TfR1)

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