JPWO2022014680A5 - - Google Patents
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- Publication number
- JPWO2022014680A5 JPWO2022014680A5 JP2022536446A JP2022536446A JPWO2022014680A5 JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5 JP 2022536446 A JP2022536446 A JP 2022536446A JP 2022536446 A JP2022536446 A JP 2022536446A JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5
- Authority
- JP
- Japan
- Prior art keywords
- octan
- azabicyclo
- represented
- formula
- fluoropyrimidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- DLFVBJFMPXGRIB-UHFFFAOYSA-N thioacetamide Natural products CC(N)=O DLFVBJFMPXGRIB-UHFFFAOYSA-N 0.000 claims 6
- 150000003839 salts Chemical class 0.000 claims 5
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020122864 | 2020-07-17 | ||
| JP2020122864 | 2020-07-17 | ||
| PCT/JP2021/026649 WO2022014680A1 (ja) | 2020-07-17 | 2021-07-15 | 置換ピペリジン化合物及びその用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2022014680A1 JPWO2022014680A1 (cg-RX-API-DMAC7.html) | 2022-01-20 |
| JP7190612B2 JP7190612B2 (ja) | 2022-12-15 |
| JPWO2022014680A5 true JPWO2022014680A5 (cg-RX-API-DMAC7.html) | 2022-12-16 |
Family
ID=79291962
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022536446A Active JP7190612B2 (ja) | 2020-07-17 | 2021-07-15 | 置換ピペリジン化合物及びその用途 |
Country Status (19)
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK4065585T3 (da) | 2019-11-25 | 2025-09-08 | Alkermes Inc | Substituerede makrocykliske forbindelser og relaterede behandlingsfremgangsmåder |
| US11760747B2 (en) | 2020-12-21 | 2023-09-19 | Alkermes, Inc. | Substituted piperidino compounds and related methods of treatment |
| US12006330B2 (en) | 2020-12-21 | 2024-06-11 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| JP7591592B2 (ja) * | 2022-01-14 | 2024-11-28 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 置換ピペリジン化合物を含有する医薬 |
| CN118451076A (zh) * | 2022-01-14 | 2024-08-06 | 卫材R&D管理有限公司 | 经取代的哌啶化合物的晶体、经取代的哌啶化合物的盐及其晶体 |
| TW202423404A (zh) * | 2022-10-07 | 2024-06-16 | 日商橘生藥品工業股份有限公司 | 環戊烷化合物 |
| TW202432109A (zh) * | 2022-10-31 | 2024-08-16 | 日商武田藥品工業股份有限公司 | 食慾素2型受體促效劑之給藥 |
| KR20250112793A (ko) | 2022-12-16 | 2025-07-24 | 다이이찌 산쿄 가부시키가이샤 | 2-아자비시클로[3.1.1]헵탄 화합물 |
| TW202502342A (zh) | 2023-06-02 | 2025-01-16 | 日商武田藥品工業股份有限公司 | 食慾素2受體促效劑用於改善睡眠期間之呼吸功能的用途 |
| WO2025124698A1 (en) | 2023-12-12 | 2025-06-19 | Idorsia Pharmaceuticals Ltd | Aryl sulfone and sulfanone derivatives as orexin receptor modulators |
| WO2025132542A1 (en) | 2023-12-19 | 2025-06-26 | Idorsia Pharmaceuticals Ltd | Macrocyclic orexin agonists |
| WO2025137359A1 (en) | 2023-12-20 | 2025-06-26 | Eisai R&D Management Co., Ltd. | Assay methods to identify a disease |
| WO2025229493A1 (en) | 2024-04-29 | 2025-11-06 | Takeda Pharmaceutical Company Limited | Dosing of orexin type 2 receptor agonists |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG34208A1 (en) | 1995-03-01 | 1996-12-06 | Guy Andrew Vaz | Blast and fragment resistant polyurethane boot sole for safety footwear |
| WO1996034877A1 (en) | 1995-05-05 | 1996-11-07 | Human Genome Sciences, Inc. | Human neuropeptide receptor |
| US6309854B1 (en) | 1996-12-17 | 2001-10-30 | Smithkline Beecham Corporation | Polynucleotides encoding ligands of the neuropeptide receptor HFGAN72 |
| US6159605A (en) | 1997-02-18 | 2000-12-12 | Dainichiseika Color & Chemicals Mfg. Co., Ltd. | Ink-jet recording sheet |
| US6020157A (en) | 1997-04-30 | 2000-02-01 | Smithkline Beecham Corporation | Polynucleotides encoding HFGAN72X receptor |
| US5935814A (en) | 1997-04-30 | 1999-08-10 | Smithkline Beecham Corporation | Polynucleotides encoding HFGAN72Y receptor |
| US6166193A (en) | 1997-07-25 | 2000-12-26 | Board Of Regents, University Of Texas System | Polynucleotides encoding MY1 receptor |
| KR100327888B1 (ko) | 1999-07-14 | 2002-03-09 | 정숭렬 | 도로포장 파손촉진 시험장치의 무선제어 시스템 |
| US7547693B2 (en) | 2003-09-22 | 2009-06-16 | Banyu Pharmaceutical Co. Ltd. | Piperidine derivative |
| MX2007004269A (es) | 2004-10-20 | 2007-06-15 | Neurosearch As | Derivados de arilo diazabiciclico nuevos y su uso medico. |
| JP2009184924A (ja) | 2006-05-31 | 2009-08-20 | Eisai R & D Management Co Ltd | 生物学的試薬用化合物 |
| TW201444849A (zh) * | 2013-03-13 | 2014-12-01 | Janssen Pharmaceutica Nv | 經取代的7-氮雜雙環類及其作為食慾激素受體調節劑之用途 |
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2021
- 2021-07-15 JP JP2022536446A patent/JP7190612B2/ja active Active
- 2021-07-15 KR KR1020227044679A patent/KR20230040953A/ko active Pending
- 2021-07-15 US US17/376,452 patent/US11479552B2/en active Active
- 2021-07-15 AU AU2021308053A patent/AU2021308053A1/en active Pending
- 2021-07-15 WO PCT/JP2021/026649 patent/WO2022014680A1/ja not_active Ceased
- 2021-07-15 CN CN202180044081.3A patent/CN115884971B/zh active Active
- 2021-07-15 TW TW110126031A patent/TWI888599B/zh active
- 2021-07-15 CN CN202411459551.4A patent/CN119235864A/zh active Pending
- 2021-07-15 MX MX2022016388A patent/MX2022016388A/es unknown
- 2021-07-15 CA CA3187835A patent/CA3187835A1/en active Pending
- 2021-07-15 EP EP21842047.9A patent/EP4151277A4/en active Pending
- 2021-07-15 PE PE2022003006A patent/PE20231103A1/es unknown
- 2021-07-15 UA UAA202204882A patent/UA129636C2/uk unknown
- 2021-07-15 PH PH1/2022/553488A patent/PH12022553488A1/en unknown
- 2021-07-15 CN CN202411462171.6A patent/CN119258067A/zh active Pending
- 2021-07-15 BR BR112022026161A patent/BR112022026161A2/pt unknown
- 2021-07-15 AR ARP210101982A patent/AR122973A1/es unknown
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2022
- 2022-12-14 IL IL299125A patent/IL299125B1/en unknown
- 2022-12-14 ZA ZA2022/13562A patent/ZA202213562B/en unknown
- 2022-12-20 CO CONC2022/0018446A patent/CO2022018446A2/es unknown
- 2022-12-20 CL CL2022003666A patent/CL2022003666A1/es unknown