JPWO2022014680A5 - - Google Patents

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Publication number
JPWO2022014680A5
JPWO2022014680A5 JP2022536446A JP2022536446A JPWO2022014680A5 JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5 JP 2022536446 A JP2022536446 A JP 2022536446A JP 2022536446 A JP2022536446 A JP 2022536446A JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5
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JP
Japan
Prior art keywords
octan
azabicyclo
represented
formula
fluoropyrimidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2022536446A
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English (en)
Japanese (ja)
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JPWO2022014680A1 (cg-RX-API-DMAC7.html
JP7190612B2 (ja
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Priority claimed from PCT/JP2021/026649 external-priority patent/WO2022014680A1/ja
Publication of JPWO2022014680A1 publication Critical patent/JPWO2022014680A1/ja
Application granted granted Critical
Publication of JP7190612B2 publication Critical patent/JP7190612B2/ja
Publication of JPWO2022014680A5 publication Critical patent/JPWO2022014680A5/ja
Active legal-status Critical Current
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JP2022536446A 2020-07-17 2021-07-15 置換ピペリジン化合物及びその用途 Active JP7190612B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2020122864 2020-07-17
JP2020122864 2020-07-17
PCT/JP2021/026649 WO2022014680A1 (ja) 2020-07-17 2021-07-15 置換ピペリジン化合物及びその用途

Publications (3)

Publication Number Publication Date
JPWO2022014680A1 JPWO2022014680A1 (cg-RX-API-DMAC7.html) 2022-01-20
JP7190612B2 JP7190612B2 (ja) 2022-12-15
JPWO2022014680A5 true JPWO2022014680A5 (cg-RX-API-DMAC7.html) 2022-12-16

Family

ID=79291962

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022536446A Active JP7190612B2 (ja) 2020-07-17 2021-07-15 置換ピペリジン化合物及びその用途

Country Status (19)

Country Link
US (1) US11479552B2 (cg-RX-API-DMAC7.html)
EP (1) EP4151277A4 (cg-RX-API-DMAC7.html)
JP (1) JP7190612B2 (cg-RX-API-DMAC7.html)
KR (1) KR20230040953A (cg-RX-API-DMAC7.html)
CN (3) CN115884971B (cg-RX-API-DMAC7.html)
AR (1) AR122973A1 (cg-RX-API-DMAC7.html)
AU (1) AU2021308053A1 (cg-RX-API-DMAC7.html)
BR (1) BR112022026161A2 (cg-RX-API-DMAC7.html)
CA (1) CA3187835A1 (cg-RX-API-DMAC7.html)
CL (1) CL2022003666A1 (cg-RX-API-DMAC7.html)
CO (1) CO2022018446A2 (cg-RX-API-DMAC7.html)
IL (1) IL299125B1 (cg-RX-API-DMAC7.html)
MX (1) MX2022016388A (cg-RX-API-DMAC7.html)
PE (1) PE20231103A1 (cg-RX-API-DMAC7.html)
PH (1) PH12022553488A1 (cg-RX-API-DMAC7.html)
TW (1) TWI888599B (cg-RX-API-DMAC7.html)
UA (1) UA129636C2 (cg-RX-API-DMAC7.html)
WO (1) WO2022014680A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA202213562B (cg-RX-API-DMAC7.html)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK4065585T3 (da) 2019-11-25 2025-09-08 Alkermes Inc Substituerede makrocykliske forbindelser og relaterede behandlingsfremgangsmåder
US11760747B2 (en) 2020-12-21 2023-09-19 Alkermes, Inc. Substituted piperidino compounds and related methods of treatment
US12006330B2 (en) 2020-12-21 2024-06-11 Alkermes, Inc. Substituted macrocyclic compounds and related methods of treatment
JP7591592B2 (ja) * 2022-01-14 2024-11-28 エーザイ・アール・アンド・ディー・マネジメント株式会社 置換ピペリジン化合物を含有する医薬
CN118451076A (zh) * 2022-01-14 2024-08-06 卫材R&D管理有限公司 经取代的哌啶化合物的晶体、经取代的哌啶化合物的盐及其晶体
TW202423404A (zh) * 2022-10-07 2024-06-16 日商橘生藥品工業股份有限公司 環戊烷化合物
TW202432109A (zh) * 2022-10-31 2024-08-16 日商武田藥品工業股份有限公司 食慾素2型受體促效劑之給藥
KR20250112793A (ko) 2022-12-16 2025-07-24 다이이찌 산쿄 가부시키가이샤 2-아자비시클로[3.1.1]헵탄 화합물
TW202502342A (zh) 2023-06-02 2025-01-16 日商武田藥品工業股份有限公司 食慾素2受體促效劑用於改善睡眠期間之呼吸功能的用途
WO2025124698A1 (en) 2023-12-12 2025-06-19 Idorsia Pharmaceuticals Ltd Aryl sulfone and sulfanone derivatives as orexin receptor modulators
WO2025132542A1 (en) 2023-12-19 2025-06-26 Idorsia Pharmaceuticals Ltd Macrocyclic orexin agonists
WO2025137359A1 (en) 2023-12-20 2025-06-26 Eisai R&D Management Co., Ltd. Assay methods to identify a disease
WO2025229493A1 (en) 2024-04-29 2025-11-06 Takeda Pharmaceutical Company Limited Dosing of orexin type 2 receptor agonists

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG34208A1 (en) 1995-03-01 1996-12-06 Guy Andrew Vaz Blast and fragment resistant polyurethane boot sole for safety footwear
WO1996034877A1 (en) 1995-05-05 1996-11-07 Human Genome Sciences, Inc. Human neuropeptide receptor
US6309854B1 (en) 1996-12-17 2001-10-30 Smithkline Beecham Corporation Polynucleotides encoding ligands of the neuropeptide receptor HFGAN72
US6159605A (en) 1997-02-18 2000-12-12 Dainichiseika Color & Chemicals Mfg. Co., Ltd. Ink-jet recording sheet
US6020157A (en) 1997-04-30 2000-02-01 Smithkline Beecham Corporation Polynucleotides encoding HFGAN72X receptor
US5935814A (en) 1997-04-30 1999-08-10 Smithkline Beecham Corporation Polynucleotides encoding HFGAN72Y receptor
US6166193A (en) 1997-07-25 2000-12-26 Board Of Regents, University Of Texas System Polynucleotides encoding MY1 receptor
KR100327888B1 (ko) 1999-07-14 2002-03-09 정숭렬 도로포장 파손촉진 시험장치의 무선제어 시스템
US7547693B2 (en) 2003-09-22 2009-06-16 Banyu Pharmaceutical Co. Ltd. Piperidine derivative
MX2007004269A (es) 2004-10-20 2007-06-15 Neurosearch As Derivados de arilo diazabiciclico nuevos y su uso medico.
JP2009184924A (ja) 2006-05-31 2009-08-20 Eisai R & D Management Co Ltd 生物学的試薬用化合物
TW201444849A (zh) * 2013-03-13 2014-12-01 Janssen Pharmaceutica Nv 經取代的7-氮雜雙環類及其作為食慾激素受體調節劑之用途

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