JPWO2021161105A5 - - Google Patents

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Publication number
JPWO2021161105A5
JPWO2021161105A5 JP2022548875A JP2022548875A JPWO2021161105A5 JP WO2021161105 A5 JPWO2021161105 A5 JP WO2021161105A5 JP 2022548875 A JP2022548875 A JP 2022548875A JP 2022548875 A JP2022548875 A JP 2022548875A JP WO2021161105 A5 JPWO2021161105 A5 JP WO2021161105A5
Authority
JP
Japan
Prior art keywords
alkyl
pharmaceutically acceptable
solvate
acceptable salt
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022548875A
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English (en)
Japanese (ja)
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JP2023513373A (ja
JP2023513373A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/000091 external-priority patent/WO2021161105A1/en
Publication of JP2023513373A publication Critical patent/JP2023513373A/ja
Publication of JPWO2021161105A5 publication Critical patent/JPWO2021161105A5/ja
Publication of JP2023513373A5 publication Critical patent/JP2023513373A5/ja
Ceased legal-status Critical Current

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JP2022548875A 2020-02-14 2021-02-12 P2x3修飾薬 Ceased JP2023513373A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062977008P 2020-02-14 2020-02-14
US62/977,008 2020-02-14
PCT/IB2021/000091 WO2021161105A1 (en) 2020-02-14 2021-02-12 P2x3 modulators

Publications (3)

Publication Number Publication Date
JP2023513373A JP2023513373A (ja) 2023-03-30
JPWO2021161105A5 true JPWO2021161105A5 (https=) 2024-02-20
JP2023513373A5 JP2023513373A5 (https=) 2024-02-20

Family

ID=77292083

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022548875A Ceased JP2023513373A (ja) 2020-02-14 2021-02-12 P2x3修飾薬

Country Status (11)

Country Link
US (1) US20230312557A1 (https=)
EP (1) EP4103564A4 (https=)
JP (1) JP2023513373A (https=)
KR (1) KR20220141331A (https=)
CN (2) CN119039290A (https=)
AU (1) AU2021219097A1 (https=)
BR (1) BR112022015858A2 (https=)
CA (1) CA3170664A1 (https=)
IL (1) IL295393A (https=)
MX (1) MX2022009762A (https=)
WO (1) WO2021161105A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2020228760A1 (en) 2019-02-25 2021-09-23 Glaxosmithkline Intellectual Property (No. 3) Limited Treatment with P2X3 modulators
EP4103572A4 (en) * 2020-02-14 2024-03-06 Bellus Health Cough Inc. MAKING A P2X3 ANTAGONIST
WO2021244634A1 (zh) * 2020-06-05 2021-12-09 武汉人福创新药物研发中心有限公司 咪唑并吡啶类化合物及其用途
CN114805237B (zh) * 2021-01-22 2026-04-21 武汉人福创新药物研发中心有限公司 杂环类化合物的制备方法及其中间体
CN114805340A (zh) * 2021-01-22 2022-07-29 武汉人福创新药物研发中心有限公司 咪唑并吡啶类化合物的制备方法及其中间体
CN116635389A (zh) * 2021-01-29 2023-08-22 上海海雁医药科技有限公司 吗啉衍生物及其药物组合物和用途
CN115043836B (zh) * 2021-08-20 2023-07-18 苏州璞正医药有限公司 一种咪唑并吡啶衍生物的p2x3受体选择性调节剂及其药物用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012011518B8 (pt) * 2009-11-18 2023-01-10 Astrazeneca Ab Compostos, composição farmacêutica, kit e usos de um composto
US9598409B2 (en) * 2013-01-31 2017-03-21 Neomed Institute Imidazopyridine compounds and uses thereof
US9907795B2 (en) * 2016-01-08 2018-03-06 Nerre Therapeutics Limited Method of treatment of chronic cough administering orvepitant in combination with other therapeutic agents
US10111883B1 (en) * 2017-09-18 2018-10-30 Bellus Health Cough Inc. Selective P2X3 modulators
CA3115939A1 (en) * 2018-10-10 2020-04-16 Bellus Health Cough Inc. Treatment of pruritus with p2x3 antagonists
WO2020135771A1 (zh) * 2018-12-29 2020-07-02 武汉朗来科技发展有限公司 杂环类化合物、中间体、其制备方法及应用
AU2020228760A1 (en) * 2019-02-25 2021-09-23 Glaxosmithkline Intellectual Property (No. 3) Limited Treatment with P2X3 modulators
CN112409331B (zh) * 2019-08-21 2024-02-20 上海翰森生物医药科技有限公司 杂环类衍生物抑制剂、其制备方法和应用

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