JPWO2021132311A1 - - Google Patents
Info
- Publication number
- JPWO2021132311A1 JPWO2021132311A1 JP2021567520A JP2021567520A JPWO2021132311A1 JP WO2021132311 A1 JPWO2021132311 A1 JP WO2021132311A1 JP 2021567520 A JP2021567520 A JP 2021567520A JP 2021567520 A JP2021567520 A JP 2021567520A JP WO2021132311 A1 JPWO2021132311 A1 JP WO2021132311A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019232927 | 2019-12-24 | ||
| JP2019232927 | 2019-12-24 | ||
| PCT/JP2020/048117 WO2021132311A1 (ja) | 2019-12-24 | 2020-12-23 | 脂肪族酸アミド誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2021132311A1 true JPWO2021132311A1 (https=) | 2021-07-01 |
| JPWO2021132311A5 JPWO2021132311A5 (https=) | 2023-12-12 |
| JP7662534B2 JP7662534B2 (ja) | 2025-04-15 |
Family
ID=76574184
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021567520A Active JP7662534B2 (ja) | 2019-12-24 | 2020-12-23 | 脂肪族酸アミド誘導体 |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US12503463B2 (https=) |
| EP (1) | EP4082616B1 (https=) |
| JP (1) | JP7662534B2 (https=) |
| KR (1) | KR20220120625A (https=) |
| CN (1) | CN114981264B (https=) |
| AU (1) | AU2020413284A1 (https=) |
| BR (1) | BR112022011844A2 (https=) |
| CA (1) | CA3161806A1 (https=) |
| ES (1) | ES3040677T3 (https=) |
| HU (1) | HUE072877T2 (https=) |
| MX (1) | MX2022007947A (https=) |
| PL (1) | PL4082616T3 (https=) |
| PT (1) | PT4082616T (https=) |
| WO (1) | WO2021132311A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20220120625A (ko) * | 2019-12-24 | 2022-08-30 | 스미토모 파마 가부시키가이샤 | 지방족 산 아미드 유도체 |
| JP7655885B2 (ja) * | 2021-06-30 | 2025-04-02 | 住友ファーマ株式会社 | 脂肪族酸アミド誘導体を含有する医薬組成物 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH01168677A (ja) * | 1987-11-30 | 1989-07-04 | Bristol Myers Co | 向精神性非環式アミド誘導体 |
| JPH093060A (ja) * | 1995-03-17 | 1997-01-07 | Hoechst Marion Roussel Inc | 置換されたベンゾチエニルピペラジン、医薬としてのその使用およびその製法 |
| JP2006508101A (ja) * | 2002-11-08 | 2006-03-09 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | フェニルアルキルおよびピリジルアルキルピペラジン誘導体 |
| JP2008539268A (ja) * | 2005-04-26 | 2008-11-13 | ハイプニオン・インコーポレイテッド | ベンズイソオキサゾールピペラジン化合物およびその使用方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5880121A (en) * | 1996-01-05 | 1999-03-09 | Hoechst Marion Roussel Inc. | 4,5-dihydronaphth (1,2-c) isoxazoles and derivatives thereof |
| JP4497815B2 (ja) | 2001-02-16 | 2010-07-07 | アベンティス・ファーマスーティカルズ・インコーポレイテツド | 新規な複素環式アミド誘導体およびドーパミンｄ３受容体リガンドとしてのその使用 |
| FR2827287B1 (fr) * | 2001-07-13 | 2003-10-31 | Servier Lab | Nouveaux derives de benzene sulfonamide, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| PL392436A1 (pl) | 2010-09-17 | 2012-03-26 | Adamed Spółka Z Ograniczoną Odpowiedzialnością | Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego |
| WO2014079155A1 (zh) * | 2012-11-26 | 2014-05-30 | 辽宁贝雷生物制药有限公司 | 苯并五元氮杂环基哌嗪或哌啶衍生物的用途 |
| KR20220120625A (ko) * | 2019-12-24 | 2022-08-30 | 스미토모 파마 가부시키가이샤 | 지방족 산 아미드 유도체 |
-
2020
- 2020-12-23 KR KR1020227025336A patent/KR20220120625A/ko active Pending
- 2020-12-23 PL PL20907330.3T patent/PL4082616T3/pl unknown
- 2020-12-23 CA CA3161806A patent/CA3161806A1/en active Pending
- 2020-12-23 JP JP2021567520A patent/JP7662534B2/ja active Active
- 2020-12-23 AU AU2020413284A patent/AU2020413284A1/en active Pending
- 2020-12-23 EP EP20907330.3A patent/EP4082616B1/en active Active
- 2020-12-23 MX MX2022007947A patent/MX2022007947A/es unknown
- 2020-12-23 US US17/612,099 patent/US12503463B2/en active Active
- 2020-12-23 HU HUE20907330A patent/HUE072877T2/hu unknown
- 2020-12-23 CN CN202080089588.6A patent/CN114981264B/zh active Active
- 2020-12-23 WO PCT/JP2020/048117 patent/WO2021132311A1/ja not_active Ceased
- 2020-12-23 PT PT209073303T patent/PT4082616T/pt unknown
- 2020-12-23 BR BR112022011844A patent/BR112022011844A2/pt unknown
- 2020-12-23 ES ES20907330T patent/ES3040677T3/es active Active
-
2021
- 2021-11-17 US US17/528,743 patent/US11339151B2/en active Active
-
2025
- 2025-11-18 US US19/392,712 patent/US20260078115A1/en active Pending
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH01168677A (ja) * | 1987-11-30 | 1989-07-04 | Bristol Myers Co | 向精神性非環式アミド誘導体 |
| JPH093060A (ja) * | 1995-03-17 | 1997-01-07 | Hoechst Marion Roussel Inc | 置換されたベンゾチエニルピペラジン、医薬としてのその使用およびその製法 |
| JP2006508101A (ja) * | 2002-11-08 | 2006-03-09 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | フェニルアルキルおよびピリジルアルキルピペラジン誘導体 |
| JP2008539268A (ja) * | 2005-04-26 | 2008-11-13 | ハイプニオン・インコーポレイテッド | ベンズイソオキサゾールピペラジン化合物およびその使用方法 |
Non-Patent Citations (2)
| Title |
|---|
| NORMAN, MARK H. ET AL.: "Synthesis and Evaluation of Heterocyclic Carboxamides as Potential Antipsychotic Agents", J. MED. CHEM., vol. 39, JPN6021004911, 1996, pages 4692 - 4703, XP055837896, ISSN: 0005452257, DOI: 10.1021/jm9603375 * |
| REGISTRY(STN)[ONLINE], JPN7024004569, 4 June 2019 (2019-06-04), pages 1, ISSN: 0005452258 * |
Also Published As
| Publication number | Publication date |
|---|---|
| US12503463B2 (en) | 2025-12-23 |
| TW202136235A (zh) | 2021-10-01 |
| KR20220120625A (ko) | 2022-08-30 |
| CA3161806A1 (en) | 2021-07-01 |
| EP4082616A1 (en) | 2022-11-02 |
| US20220073506A1 (en) | 2022-03-10 |
| US20260078115A1 (en) | 2026-03-19 |
| BR112022011844A2 (pt) | 2022-08-30 |
| WO2021132311A1 (ja) | 2021-07-01 |
| EP4082616B1 (en) | 2025-09-03 |
| US11339151B2 (en) | 2022-05-24 |
| JP7662534B2 (ja) | 2025-04-15 |
| CN114981264A (zh) | 2022-08-30 |
| PL4082616T3 (pl) | 2025-12-15 |
| MX2022007947A (es) | 2022-07-27 |
| EP4082616A4 (en) | 2024-01-03 |
| AU2020413284A1 (en) | 2022-08-18 |
| US20220213079A1 (en) | 2022-07-07 |
| PT4082616T (pt) | 2025-12-02 |
| HUE072877T2 (hu) | 2025-12-28 |
| CN114981264B (zh) | 2024-07-26 |
| ES3040677T3 (en) | 2025-11-04 |
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