PL392436A1 - Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego - Google Patents

Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego

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Publication number
PL392436A1
PL392436A1 PL39243610A PL39243610A PL392436A1 PL 392436 A1 PL392436 A1 PL 392436A1 PL 39243610 A PL39243610 A PL 39243610A PL 39243610 A PL39243610 A PL 39243610A PL 392436 A1 PL392436 A1 PL 392436A1
Authority
PL
Poland
Prior art keywords
diseases
treating
nervous system
central nervous
arylsulphonamide
Prior art date
Application number
PL39243610A
Other languages
English (en)
Inventor
Marcin Kołaczkowski
Piotr Kowalski
Jolanta Jaśkowska
Katarzyna Mitka
Monika Jagodzińska
Adam Bucki
Anna Wesołowska
Maciej Pawłowski
Original Assignee
Adamed Spółka Z Ograniczoną Odpowiedzialnością
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adamed Spółka Z Ograniczoną Odpowiedzialnością filed Critical Adamed Spółka Z Ograniczoną Odpowiedzialnością
Priority to PL39243610A priority Critical patent/PL392436A1/pl
Priority to KR20137009661A priority patent/KR20130143569A/ko
Priority to EA201390398A priority patent/EA022776B1/ru
Priority to AU2011303807A priority patent/AU2011303807B2/en
Priority to CN201180044733XA priority patent/CN103108864A/zh
Priority to CA2808246A priority patent/CA2808246A1/en
Priority to JP2013528677A priority patent/JP5899218B2/ja
Priority to PCT/EP2011/066054 priority patent/WO2012035123A1/en
Priority to EP11767950.6A priority patent/EP2616440A1/en
Priority to BR112013006313A priority patent/BR112013006313A2/pt
Priority to US13/824,066 priority patent/US8822517B2/en
Priority to CN201410638124.2A priority patent/CN104529999A/zh
Priority to UAA201304643A priority patent/UA109793C2/uk
Priority to MX2013002956A priority patent/MX2013002956A/es
Priority to NZ607031A priority patent/NZ607031A/en
Publication of PL392436A1 publication Critical patent/PL392436A1/pl
Priority to ZA2013/02390A priority patent/ZA201302390B/en
Priority to ZA2013/05970A priority patent/ZA201305970B/en
Priority to US14/338,704 priority patent/US9120767B2/en

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • C07D209/04—Indoles; Hydrogenated indoles
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    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
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    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
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  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL39243610A 2010-09-17 2010-09-17 Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego PL392436A1 (pl)

Priority Applications (18)

Application Number Priority Date Filing Date Title
PL39243610A PL392436A1 (pl) 2010-09-17 2010-09-17 Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego
BR112013006313A BR112013006313A2 (pt) 2010-09-17 2011-09-16 arisulfonamidas para o tratamento de enfermidades do cns
US13/824,066 US8822517B2 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of CNS diseases
AU2011303807A AU2011303807B2 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of CNS diseases
CN201180044733XA CN103108864A (zh) 2010-09-17 2011-09-16 用于治疗cns疾病的芳基磺酰胺
CA2808246A CA2808246A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases
JP2013528677A JP5899218B2 (ja) 2010-09-17 2011-09-16 Ｃｎｓ疾患の処置のためのアリールスルホンアミド
PCT/EP2011/066054 WO2012035123A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases
EP11767950.6A EP2616440A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases
KR20137009661A KR20130143569A (ko) 2010-09-17 2011-09-16 중추신경계 질환의 치료를 위한 아릴술폰아미드
EA201390398A EA022776B1 (ru) 2010-09-17 2011-09-16 Арилсульфонамиды для лечения заболеваний цнс
CN201410638124.2A CN104529999A (zh) 2010-09-17 2011-09-16 用于治疗cns疾病的芳基磺酰胺
UAA201304643A UA109793C2 (uk) 2010-09-17 2011-09-16 Арилсульфонаміди для лікування захворювань центральної нервової системи (цнс)
MX2013002956A MX2013002956A (es) 2010-09-17 2011-09-16 Arilsulfonamidas para el tratamiento de enfermedades del sistema nervioso central.
NZ607031A NZ607031A (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases
ZA2013/02390A ZA201302390B (en) 2010-09-17 2013-04-03 Arylosulfonamides for the treatment of cns diseases
ZA2013/05970A ZA201305970B (en) 2010-09-17 2013-08-07 Arylosulfonami for the treatment of cns diseases
US14/338,704 US9120767B2 (en) 2010-09-17 2014-07-23 Arylosulfonamides for the treatment of CNS diseases

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CN106749219A (zh) * 2015-11-20 2017-05-31 江苏恩华药业股份有限公司 一种内酰胺类衍生物及其应用
CN107602446B (zh) * 2016-07-12 2020-04-07 中国科学院上海药物研究所 1,4-双取代-1,2,3,6-四氢吡啶类化合物、其制备方法、药物组合物及其应用
PT4082616T (pt) 2019-12-24 2025-12-02 Sumitomo Pharma Co Ltd Derivado de amida ácida alifática
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WO2021241875A1 (ko) * 2020-05-29 2021-12-02 재단법인 대구경북첨단의료산업진흥재단 설폰아미드 유도체 및 이를 유효성분으로 함유하는 정신질환의 예방 또는 치료용 약학적 조성물

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US9120767B2 (en) 2015-09-01
UA109793C2 (uk) 2015-10-12
EP2616440A1 (en) 2013-07-24
KR20130143569A (ko) 2013-12-31
BR112013006313A2 (pt) 2016-06-07
AU2011303807B2 (en) 2014-07-17
CN103108864A (zh) 2013-05-15
CN104529999A (zh) 2015-04-22
EA022776B1 (ru) 2016-02-29
AU2011303807A1 (en) 2013-02-28
US8822517B2 (en) 2014-09-02
CA2808246A1 (en) 2012-03-22
US20130172365A1 (en) 2013-07-04
EA201390398A1 (ru) 2013-07-30
NZ607031A (en) 2014-06-27
JP5899218B2 (ja) 2016-04-06
MX2013002956A (es) 2013-05-09
ZA201302390B (en) 2013-12-23
ZA201305970B (en) 2014-04-30
US20140336200A1 (en) 2014-11-13
WO2012035123A1 (en) 2012-03-22

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