EA201390398A1 - Арилсульфонамиды для лечения заболеваний цнс - Google Patents

Арилсульфонамиды для лечения заболеваний цнс

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Publication number
EA201390398A1
EA201390398A1 EA201390398A EA201390398A EA201390398A1 EA 201390398 A1 EA201390398 A1 EA 201390398A1 EA 201390398 A EA201390398 A EA 201390398A EA 201390398 A EA201390398 A EA 201390398A EA 201390398 A1 EA201390398 A1 EA 201390398A1
Authority
EA
Eurasian Patent Office
Prior art keywords
arylsulphonamides
treatment
cns diseases
arylsulfonamide
treat
Prior art date
Application number
EA201390398A
Other languages
English (en)
Other versions
EA022776B1 (ru
Inventor
Марцин Колачковский
Петр Ковальский
Йолянта Яськовская
Моника Марцинковская
Катажина Митка
Адам Буцкий
Анна Весоловская
Мацей Павловский
Original Assignee
Адамед Сп. З О.О.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Адамед Сп. З О.О. filed Critical Адамед Сп. З О.О.
Publication of EA201390398A1 publication Critical patent/EA201390398A1/ru
Publication of EA022776B1 publication Critical patent/EA022776B1/ru

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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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Abstract

Производные арилсульфонамида формулы (I) и их фармацевтически приемлемые соли. Эти соединения могут быть использованы для лечения и/или профилактики нарушений центральной нервной системы.
EA201390398A 2010-09-17 2011-09-16 Арилсульфонамиды для лечения заболеваний цнс EA022776B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PL39243610A PL392436A1 (pl) 2010-09-17 2010-09-17 Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego
PCT/EP2011/066054 WO2012035123A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases

Publications (2)

Publication Number Publication Date
EA201390398A1 true EA201390398A1 (ru) 2013-07-30
EA022776B1 EA022776B1 (ru) 2016-02-29

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Application Number Title Priority Date Filing Date
EA201390398A EA022776B1 (ru) 2010-09-17 2011-09-16 Арилсульфонамиды для лечения заболеваний цнс

Country Status (15)

Country Link
US (2) US8822517B2 (ru)
EP (1) EP2616440A1 (ru)
JP (1) JP5899218B2 (ru)
KR (1) KR20130143569A (ru)
CN (2) CN103108864A (ru)
AU (1) AU2011303807B2 (ru)
BR (1) BR112013006313A2 (ru)
CA (1) CA2808246A1 (ru)
EA (1) EA022776B1 (ru)
MX (1) MX2013002956A (ru)
NZ (1) NZ607031A (ru)
PL (1) PL392436A1 (ru)
UA (1) UA109793C2 (ru)
WO (1) WO2012035123A1 (ru)
ZA (2) ZA201302390B (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105085436B (zh) 2014-04-19 2019-08-16 广东东阳光药业有限公司 磺酰胺类衍生物及其在药物上的应用
CN106749219A (zh) * 2015-11-20 2017-05-31 江苏恩华药业股份有限公司 一种内酰胺类衍生物及其应用
CN107602446B (zh) * 2016-07-12 2020-04-07 中国科学院上海药物研究所 1,4-双取代-1,2,3,6-四氢吡啶类化合物、其制备方法、药物组合物及其应用
MX2022007947A (es) * 2019-12-24 2022-07-27 Sumitomo Pharma Co Ltd Derivado de amida de acido alifatico.
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WO2012035123A1 (en) 2012-03-22
BR112013006313A2 (pt) 2016-06-07
EP2616440A1 (en) 2013-07-24
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US9120767B2 (en) 2015-09-01
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AU2011303807A1 (en) 2013-02-28
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