BR112013006313A2 - arisulfonamidas para o tratamento de enfermidades do cns - Google Patents

arisulfonamidas para o tratamento de enfermidades do cns

Info

Publication number
BR112013006313A2
BR112013006313A2 BR112013006313A BR112013006313A BR112013006313A2 BR 112013006313 A2 BR112013006313 A2 BR 112013006313A2 BR 112013006313 A BR112013006313 A BR 112013006313A BR 112013006313 A BR112013006313 A BR 112013006313A BR 112013006313 A2 BR112013006313 A2 BR 112013006313A2
Authority
BR
Brazil
Prior art keywords
treatment
arisulfonamides
cns diseases
cns
diseases
Prior art date
Application number
BR112013006313A
Other languages
English (en)
Inventor
Adam Bucki
Anna Wesolowska
Jolanta Jaskowska
Kataryzna Mitka
Marcin Kolaczkowski
Maciej Pawlowski
Monika Marcinkowska
Piotr Kowalski
Original Assignee
Adamed Sp Zoo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adamed Sp Zoo filed Critical Adamed Sp Zoo
Publication of BR112013006313A2 publication Critical patent/BR112013006313A2/pt

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Abstract

arilsofonamidas para o tratamento de enfermidades do cns. expõem-se derivados de arilsulfonamidas da fórmula (i) e os seus sais farmaceuticamente aceitáveis. os compostos podem ser de utilidade para o tratamento e/ou prevenção de distúrbios do sistema nervoso central.
BR112013006313A 2010-09-17 2011-09-16 arisulfonamidas para o tratamento de enfermidades do cns BR112013006313A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PL39243610A PL392436A1 (pl) 2010-09-17 2010-09-17 Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego
PCT/EP2011/066054 WO2012035123A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases

Publications (1)

Publication Number Publication Date
BR112013006313A2 true BR112013006313A2 (pt) 2016-06-07

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BR112013006313A BR112013006313A2 (pt) 2010-09-17 2011-09-16 arisulfonamidas para o tratamento de enfermidades do cns

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US (2) US8822517B2 (pt)
EP (1) EP2616440A1 (pt)
JP (1) JP5899218B2 (pt)
KR (1) KR20130143569A (pt)
CN (2) CN103108864A (pt)
AU (1) AU2011303807B2 (pt)
BR (1) BR112013006313A2 (pt)
CA (1) CA2808246A1 (pt)
EA (1) EA022776B1 (pt)
MX (1) MX2013002956A (pt)
NZ (1) NZ607031A (pt)
PL (1) PL392436A1 (pt)
UA (1) UA109793C2 (pt)
WO (1) WO2012035123A1 (pt)
ZA (2) ZA201302390B (pt)

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WO2015158313A1 (en) 2014-04-19 2015-10-22 Sunshine Lake Pharma Co., Ltd. Sulfonamide derivatives and pharmaceutical applications thereof
CN106749219A (zh) * 2015-11-20 2017-05-31 江苏恩华药业股份有限公司 一种内酰胺类衍生物及其应用
CN107602446B (zh) * 2016-07-12 2020-04-07 中国科学院上海药物研究所 1,4-双取代-1,2,3,6-四氢吡啶类化合物、其制备方法、药物组合物及其应用
JPWO2021132311A1 (pt) * 2019-12-24 2021-07-01
KR102447231B1 (ko) * 2020-05-29 2022-09-27 재단법인 대구경북첨단의료산업진흥재단 설폰아미드 유도체 및 이를 유효성분으로 함유하는 정신질환의 예방 또는 치료용 약학적 조성물
JP2023528545A (ja) * 2020-05-29 2023-07-04 テグ－キョンプク メディカル イノベーション ファウンデーション スルホンアミド誘導体およびそれを有効成分とする精神病の予防または治療に使用するための医薬組成物

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WO2012035123A1 (en) 2012-03-22
CN104529999A (zh) 2015-04-22
AU2011303807A1 (en) 2013-02-28
JP2013540738A (ja) 2013-11-07
US20130172365A1 (en) 2013-07-04
CN103108864A (zh) 2013-05-15
CA2808246A1 (en) 2012-03-22
EA201390398A1 (ru) 2013-07-30
UA109793C2 (uk) 2015-10-12
AU2011303807B2 (en) 2014-07-17
US20140336200A1 (en) 2014-11-13
PL392436A1 (pl) 2012-03-26
ZA201305970B (en) 2014-04-30
MX2013002956A (es) 2013-05-09
JP5899218B2 (ja) 2016-04-06
EP2616440A1 (en) 2013-07-24
EA022776B1 (ru) 2016-02-29
NZ607031A (en) 2014-06-27
US9120767B2 (en) 2015-09-01
US8822517B2 (en) 2014-09-02
ZA201302390B (en) 2013-12-23
KR20130143569A (ko) 2013-12-31

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