JPWO2020254985A5 - - Google Patents

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Publication number
JPWO2020254985A5
JPWO2020254985A5 JP2021575482A JP2021575482A JPWO2020254985A5 JP WO2020254985 A5 JPWO2020254985 A5 JP WO2020254985A5 JP 2021575482 A JP2021575482 A JP 2021575482A JP 2021575482 A JP2021575482 A JP 2021575482A JP WO2020254985 A5 JPWO2020254985 A5 JP WO2020254985A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
administration
acceptable salt
agent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021575482A
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English (en)
Japanese (ja)
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JP2022537047A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2020/055653 external-priority patent/WO2020254985A1/en
Publication of JP2022537047A publication Critical patent/JP2022537047A/ja
Publication of JPWO2020254985A5 publication Critical patent/JPWO2020254985A5/ja
Pending legal-status Critical Current

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JP2021575482A 2019-06-19 2020-06-17 ヒト免疫不全ウイルス複製の阻害剤としてのピリド[2,3-d]ピリミジン誘導体 Pending JP2022537047A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962863406P 2019-06-19 2019-06-19
US62/863,406 2019-06-19
PCT/IB2020/055653 WO2020254985A1 (en) 2019-06-19 2020-06-17 Pyrido[2,3-d]pyrimidine derivatives as inhibitors of human immunodeficiency virus replication

Publications (2)

Publication Number Publication Date
JP2022537047A JP2022537047A (ja) 2022-08-23
JPWO2020254985A5 true JPWO2020254985A5 (fi) 2023-06-21

Family

ID=71738195

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021575482A Pending JP2022537047A (ja) 2019-06-19 2020-06-17 ヒト免疫不全ウイルス複製の阻害剤としてのピリド[2,3-d]ピリミジン誘導体

Country Status (25)

Country Link
US (1) US20210323967A1 (fi)
EP (1) EP3986561B1 (fi)
JP (1) JP2022537047A (fi)
KR (1) KR20220024608A (fi)
CN (1) CN114245795A (fi)
AR (1) AR119174A1 (fi)
AU (1) AU2020295793B2 (fi)
BR (1) BR112021025655A2 (fi)
CA (1) CA3143136A1 (fi)
CL (1) CL2021003388A1 (fi)
CO (1) CO2021017479A2 (fi)
CR (1) CR20210664A (fi)
DK (1) DK3986561T3 (fi)
FI (1) FI3986561T3 (fi)
IL (1) IL288750A (fi)
LT (1) LT3986561T (fi)
MA (1) MA56526A (fi)
MX (1) MX2021016149A (fi)
PE (1) PE20220510A1 (fi)
PT (1) PT3986561T (fi)
RS (1) RS65304B1 (fi)
SI (1) SI3986561T1 (fi)
TW (1) TW202115055A (fi)
UY (1) UY38755A (fi)
WO (1) WO2020254985A1 (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7398448B2 (ja) 2018-10-24 2023-12-14 ヴィーブ ヘルスケア ユーケー(ナンバー5)リミテッド ヒト免疫不全ウイルス複製の阻害剤
CA3164528A1 (en) * 2019-12-09 2021-06-17 Viiv Healthcare Company Pharmaceutical compositions comprising cabotegravir
BR112022017832A2 (pt) * 2020-03-06 2022-11-01 Viiv Healthcare Uk No 5 Ltd Inibidores de replicação do vírus da imunodeficiência humana
CA3234219A1 (en) 2021-10-13 2023-04-20 Gautam Dalwadi Inhibitors of human immunodeficiency virus replication

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2212324B1 (en) * 2008-07-02 2014-03-26 Avexa Limited Compounds having antiviral properties
CN102464654B (zh) 2010-11-12 2016-01-13 上海泓博智源医药技术有限公司 抗病毒化合物
PT2729448E (pt) 2011-07-06 2015-12-02 Gilead Sciences Inc Compostos para o tratamento de vih
CN102863512B (zh) 2011-07-07 2016-04-20 上海泓博智源医药技术有限公司 抗病毒化合物
AU2014205317B2 (en) 2013-01-09 2016-11-24 Gilead Sciences, Inc. 5-membered heteroaryls and their use as antiviral agents
ES2642265T3 (es) 2013-01-09 2017-11-16 Gilead Sciences, Inc. Compuestos terapéuticos para el tratamiento de infecciones virales
TW201443037A (zh) * 2013-01-09 2014-11-16 Gilead Sciences Inc 治療用化合物
TWI694071B (zh) 2013-03-01 2020-05-21 美商基利科學股份有限公司 治療反轉錄病毒科(Retroviridae)病毒感染之治療性化合物
WO2015130966A1 (en) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Antiviral agents
US10202353B2 (en) 2014-02-28 2019-02-12 Gilead Sciences, Inc. Therapeutic compounds
WO2016033243A1 (en) 2014-08-29 2016-03-03 Gilead Sciences, Inc. Antiretroviral agents
CN109890808B (zh) * 2016-08-19 2020-08-07 吉利德科学公司 用于预防性或治疗性治疗hiv病毒感染的治疗性化合物
ES2826748T3 (es) * 2016-09-02 2021-05-19 Gilead Sciences Inc Derivados de 4,6-diamino-pirido[3,2-d]pirimidina como moduladores de receptores de tipo Toll
TW201906834A (zh) * 2017-05-02 2019-02-16 英商Viiv醫療保健英國(No.5)有限公司 人類免疫不全病毒複製之抑制劑
UY38559A (es) * 2019-02-01 2020-07-31 Viiv Healthcare Uk No 5 Ltd Inhibidores de la replicación del virus de la inmunodeficiencia humana

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