JPWO2020181050A5 - - Google Patents

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Publication number
JPWO2020181050A5
JPWO2020181050A5 JP2021552747A JP2021552747A JPWO2020181050A5 JP WO2020181050 A5 JPWO2020181050 A5 JP WO2020181050A5 JP 2021552747 A JP2021552747 A JP 2021552747A JP 2021552747 A JP2021552747 A JP 2021552747A JP WO2020181050 A5 JPWO2020181050 A5 JP WO2020181050A5
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JP
Japan
Prior art keywords
disease
syndrome
compound
item
alkylenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021552747A
Other languages
English (en)
Japanese (ja)
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JP2022525010A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/021120 external-priority patent/WO2020181050A1/en
Publication of JP2022525010A publication Critical patent/JP2022525010A/ja
Publication of JPWO2020181050A5 publication Critical patent/JPWO2020181050A5/ja
Pending legal-status Critical Current

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JP2021552747A 2019-03-05 2020-03-05 疾患の治療のための化合物、組成物、及び方法 Pending JP2022525010A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962814025P 2019-03-05 2019-03-05
US62/814,025 2019-03-05
US201962879178P 2019-07-26 2019-07-26
US62/879,178 2019-07-26
PCT/US2020/021120 WO2020181050A1 (en) 2019-03-05 2020-03-05 Compounds, compositions, and methods for the treatment of disease

Publications (2)

Publication Number Publication Date
JP2022525010A JP2022525010A (ja) 2022-05-11
JPWO2020181050A5 true JPWO2020181050A5 (ko) 2023-03-13

Family

ID=72338059

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021552747A Pending JP2022525010A (ja) 2019-03-05 2020-03-05 疾患の治療のための化合物、組成物、及び方法

Country Status (20)

Country Link
US (1) US20220168309A1 (ko)
EP (1) EP3934652A4 (ko)
JP (1) JP2022525010A (ko)
KR (1) KR20210135544A (ko)
CN (1) CN113645977A (ko)
AU (1) AU2020232761A1 (ko)
BR (1) BR112021017583A2 (ko)
CA (1) CA3131620A1 (ko)
CL (1) CL2021002294A1 (ko)
CO (1) CO2021012586A2 (ko)
CR (1) CR20210508A (ko)
DO (1) DOP2021000184A (ko)
EC (1) ECSP21073266A (ko)
IL (1) IL285782A (ko)
JO (1) JOP20210244A1 (ko)
MA (1) MA55214A (ko)
MX (1) MX2021010701A (ko)
PE (1) PE20220166A1 (ko)
SG (1) SG11202109452SA (ko)
WO (1) WO2020181050A1 (ko)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113490668A (zh) 2018-10-05 2021-10-08 安娜普尔纳生物股份有限公司 用于治疗与apj受体活性有关的疾病的化合物和组合物
BR112021016620A2 (pt) 2019-02-27 2021-11-03 Univ California Azepino-indóis e outros heterociclos para o tratamento de distúrbios cerebrais
JP2022543086A (ja) 2019-08-02 2022-10-07 メルサナ セラピューティクス インコーポレイテッド がんの処置用のSTING(インターフェロン遺伝子刺激因子)アゴニストとしてのビス-[N-((5-カルバモイル)-1H-ベンゾ[d]イミダゾール-2-イル)-ピラゾール-5-カルボキサミド]誘導体および関連化合物
WO2021226261A1 (en) 2020-05-06 2021-11-11 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
WO2022034474A1 (en) * 2020-08-10 2022-02-17 Novartis Ag Treatments for retinal degenerative diseases
US11767321B2 (en) 2020-10-05 2023-09-26 Enliven Inc. 5- and 6-azaindole compounds for inhibition of BCR-ABL tyrosine kinases
CN114478715B (zh) * 2020-10-26 2023-12-22 南京吉芮康生物科技研究院有限公司 一种减毒沙门氏菌分泌表达s2结构域蛋白的新型冠状病毒疫苗递呈系统及其应用
US11964978B2 (en) * 2021-03-18 2024-04-23 Pfizer Inc. Modulators of STING (stimulator of interferon genes)
WO2022266711A1 (en) * 2021-06-23 2022-12-29 Aculeus Therapeutics Pty Ltd Substituted amidobenzimidazole dimers as sting modulators
AU2022388555A1 (en) 2021-11-09 2024-05-02 Ajax Therapeutics, Inc. 6-he tero aryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
WO2024118785A2 (en) 2022-11-30 2024-06-06 Regeneron Pharmaceuticals, Inc. Tlr7 agonists and antibody-drug-conjugates thereof
CN115624616B (zh) * 2022-12-21 2023-03-14 上海市东方医院(同济大学附属东方医院) 接头蛋白pinch在诊断血管发育异常相关疾病中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6110923A (en) * 1994-06-22 2000-08-29 Biochem Pharma Inc. Method for treating cancer using novel substituted purinyl derivatives with immunomodulating activity
US6770651B2 (en) * 2001-06-29 2004-08-03 Venkata Palle A2B adenosine receptor antagonists
WO2010017248A2 (en) * 2008-08-04 2010-02-11 University Of Miami Sting (stimulator of interferon genes), a regulator of innate immune responses
SG11201607586UA (en) * 2014-03-13 2016-10-28 Agency Science Tech & Res Fused pyrimidine-based hydroxamate derivatives
GB201501462D0 (en) * 2015-01-29 2015-03-18 Glaxosmithkline Ip Dev Ltd Novel compounds

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