JPWO2020035779A5 - - Google Patents

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Publication number
JPWO2020035779A5
JPWO2020035779A5 JP2021507613A JP2021507613A JPWO2020035779A5 JP WO2020035779 A5 JPWO2020035779 A5 JP WO2020035779A5 JP 2021507613 A JP2021507613 A JP 2021507613A JP 2021507613 A JP2021507613 A JP 2021507613A JP WO2020035779 A5 JPWO2020035779 A5 JP WO2020035779A5
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JP
Japan
Prior art keywords
cancer
carcinoma
hydrogen
cell carcinoma
pharmaceutically acceptable
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JP2021507613A
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English (en)
Japanese (ja)
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JP2021534147A (ja
JP7328323B2 (ja
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Priority claimed from PCT/IB2019/056847 external-priority patent/WO2020035779A1/en
Publication of JP2021534147A publication Critical patent/JP2021534147A/ja
Publication of JPWO2020035779A5 publication Critical patent/JPWO2020035779A5/ja
Application granted granted Critical
Publication of JP7328323B2 publication Critical patent/JP7328323B2/ja
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JP2021507613A 2018-08-17 2019-08-12 SMARCA2/BRM ATPase阻害剤としての尿素化合物及び組成物 Active JP7328323B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862765138P 2018-08-17 2018-08-17
US62/765,138 2018-08-17
PCT/IB2019/056847 WO2020035779A1 (en) 2018-08-17 2019-08-12 Urea compounds and compositions as smarca2/brm atpase inhibitors

Publications (3)

Publication Number Publication Date
JP2021534147A JP2021534147A (ja) 2021-12-09
JPWO2020035779A5 true JPWO2020035779A5 (es) 2022-08-17
JP7328323B2 JP7328323B2 (ja) 2023-08-16

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ID=68072895

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021507613A Active JP7328323B2 (ja) 2018-08-17 2019-08-12 SMARCA2/BRM ATPase阻害剤としての尿素化合物及び組成物

Country Status (21)

Country Link
US (1) US11958846B2 (es)
EP (2) EP4219488A1 (es)
JP (1) JP7328323B2 (es)
KR (1) KR20210047313A (es)
CN (1) CN112585136B (es)
AU (1) AU2019322325B2 (es)
BR (1) BR112021002632A2 (es)
CA (1) CA3107097A1 (es)
CY (1) CY1126039T1 (es)
DK (1) DK3837256T3 (es)
ES (1) ES2946060T3 (es)
FI (1) FI3837256T3 (es)
HR (1) HRP20230477T1 (es)
HU (1) HUE061963T2 (es)
LT (1) LT3837256T (es)
MX (1) MX2021001804A (es)
PL (1) PL3837256T3 (es)
PT (1) PT3837256T (es)
RS (1) RS64238B1 (es)
SI (1) SI3837256T1 (es)
WO (1) WO2020035779A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11497752B2 (en) 2018-01-30 2022-11-15 Foghorn Therapeutics Inc. Compounds and uses thereof
BR112022015004A2 (pt) 2020-01-29 2022-09-20 Foghorn Therapeutics Inc Composto, composição farmacêutica, métodos para diminuir a atividade de um complexo baf, induzir apoptose, reduzir o crescimento tumoral, suprimir a progressão e a colonização metastática do câncer e reduzir o nível e/ou a atividade de brg1 e/ou brm em um câncer e métodos de tratamento e de inibição de brm e brg1
CN112979646B (zh) * 2021-03-08 2022-01-14 北京富龙康泰生物技术有限公司 一种咪唑并吡啶类衍生物

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US2779780A (en) 1955-03-01 1957-01-29 Du Pont 1, 4-diamino-2, 3-dicyano-1, 4-bis (substituted mercapto) butadienes and their preparation
AUPP003197A0 (en) 1997-09-03 1997-11-20 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
GB9823873D0 (en) * 1998-10-30 1998-12-30 Pharmacia & Upjohn Spa 2-ureido-thiazole derivatives,process for their preparation,and their use as antitumour agents
KR100609800B1 (ko) 1998-12-16 2006-08-09 워너-램버트 캄파니 엘엘씨 Mek 저해제를 사용한 관절염 치료 방법
US7217722B2 (en) * 2000-02-01 2007-05-15 Kirin Beer Kabushiki Kaisha Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same
PL203387B1 (pl) 2000-07-19 2009-09-30 Warner Lambert Co Utlenione estry kwasu 4-jodofenyloaminobenzhydroksamowego
US20020173507A1 (en) 2000-08-15 2002-11-21 Vincent Santora Urea compounds and methods of uses
ATE442362T1 (de) 2001-05-24 2009-09-15 Leo Pharma As Pyridylcyanoguanidin verbindungen
PL221491B1 (pl) 2002-03-08 2016-04-29 Eisai R&D Man Co Związki makrocykliczne, środek farmaceutyczny zawierający te związki oraz zastosowanie tych związków
ES2335276T3 (es) 2002-03-13 2010-03-24 Array Biopharma, Inc. Derivados de bencimidazol alquilado n3 como inhibidores de mek.
US20030236287A1 (en) 2002-05-03 2003-12-25 Piotrowski David W. Positive allosteric modulators of the nicotinic acetylcholine receptor
CA2744893A1 (en) 2002-06-27 2004-01-08 Novo Nordisk A/S Aryl carbonyl derivatives as glucokinase activators
CA2514733A1 (en) 2003-02-28 2004-09-16 Transform Pharmaceuticals, Inc. Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
WO2004085433A2 (en) 2003-03-28 2004-10-07 Pharmacia & Upjohn Company Llc Positive allosteric modulators of the nicotinic acetylcholine receptor
PT1912636E (pt) 2005-07-21 2014-07-24 Ardea Biosciences Inc Inibidores de n-(arilamino)-sulfonamida de mek
JO2660B1 (en) 2006-01-20 2012-06-17 نوفارتيس ايه جي Pi-3 inhibitors and methods of use
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TWI471134B (zh) 2007-09-12 2015-02-01 Genentech Inc 肌醇磷脂3-激酶抑制劑化合物及化療劑之組合及使用方法
WO2009055730A1 (en) 2007-10-25 2009-04-30 Genentech, Inc. Process for making thienopyrimidine compounds
CN101969949B (zh) 2008-03-14 2013-12-25 大塚制药株式会社 Mmp-2及/或mmp-9抑制剂
JP6665154B2 (ja) 2014-07-17 2020-03-13 ノース・アンド・サウス・ブラザー・ファーマシー・インベストメント・カンパニー・リミテッド 置換尿素誘導体及びその薬学的使用
MA41598A (fr) 2015-02-25 2018-01-02 Constellation Pharmaceuticals Inc Composés thérapeutiques de pyridazine et leurs utilisations
CN105481723B (zh) 2015-04-29 2017-08-25 中国农业大学 一种非均相催化的烷基/苄基/芳基脲类化合物的制备方法
WO2018187414A1 (en) 2017-04-05 2018-10-11 The Regents Of The University Of California Inhibitors of mtor-rictor interactions
WO2020126968A2 (en) 2018-12-20 2020-06-25 Bayer Aktiengesellschaft Urea derivatives

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