JPWO2019145729A5 - - Google Patents

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Publication number
JPWO2019145729A5
JPWO2019145729A5 JP2020561950A JP2020561950A JPWO2019145729A5 JP WO2019145729 A5 JPWO2019145729 A5 JP WO2019145729A5 JP 2020561950 A JP2020561950 A JP 2020561950A JP 2020561950 A JP2020561950 A JP 2020561950A JP WO2019145729 A5 JPWO2019145729 A5 JP WO2019145729A5
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JP
Japan
Prior art keywords
disease
cancer
arthritis
syndrome
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2020561950A
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English (en)
Japanese (ja)
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JP2021512158A (ja
Publication date
Priority claimed from GBGB1801226.0A external-priority patent/GB201801226D0/en
Application filed filed Critical
Publication of JP2021512158A publication Critical patent/JP2021512158A/ja
Publication of JPWO2019145729A5 publication Critical patent/JPWO2019145729A5/ja
Priority to JP2023200631A priority Critical patent/JP2024026193A/ja
Pending legal-status Critical Current

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JP2020561950A 2018-01-25 2019-01-25 Rho関連プロテインキナーゼのモジュレーター Pending JP2021512158A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023200631A JP2024026193A (ja) 2018-01-25 2023-11-28 Rho関連プロテインキナーゼのモジュレーター

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1801226.0 2018-01-25
GBGB1801226.0A GB201801226D0 (en) 2018-01-25 2018-01-25 Modulators of Rho-associated protein kinase
PCT/GB2019/050215 WO2019145729A1 (en) 2018-01-25 2019-01-25 Heterocyclylamino-substituted triazoles as modulators of rho-associated protein kinase

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023200631A Division JP2024026193A (ja) 2018-01-25 2023-11-28 Rho関連プロテインキナーゼのモジュレーター

Publications (2)

Publication Number Publication Date
JP2021512158A JP2021512158A (ja) 2021-05-13
JPWO2019145729A5 true JPWO2019145729A5 (es) 2022-01-31

Family

ID=61558335

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020561950A Pending JP2021512158A (ja) 2018-01-25 2019-01-25 Rho関連プロテインキナーゼのモジュレーター
JP2023200631A Pending JP2024026193A (ja) 2018-01-25 2023-11-28 Rho関連プロテインキナーゼのモジュレーター

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023200631A Pending JP2024026193A (ja) 2018-01-25 2023-11-28 Rho関連プロテインキナーゼのモジュレーター

Country Status (25)

Country Link
US (2) US11497751B2 (es)
EP (2) EP3743420B1 (es)
JP (2) JP2021512158A (es)
KR (1) KR20200113216A (es)
CN (1) CN111655681B (es)
AU (1) AU2019213214B2 (es)
BR (1) BR112020013759A2 (es)
CA (1) CA3088330A1 (es)
CY (1) CY1125017T1 (es)
DK (1) DK3743420T3 (es)
EA (1) EA202091711A1 (es)
ES (1) ES2907833T3 (es)
GB (1) GB201801226D0 (es)
HR (1) HRP20220269T8 (es)
HU (1) HUE058940T2 (es)
IL (1) IL275988B2 (es)
LT (1) LT3743420T (es)
MX (1) MX2020007898A (es)
PH (1) PH12020550986A1 (es)
PL (1) PL3743420T3 (es)
PT (1) PT3743420T (es)
SG (1) SG11202006087UA (es)
SI (1) SI3743420T1 (es)
WO (1) WO2019145729A1 (es)
ZA (1) ZA202003983B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201801226D0 (en) 2018-01-25 2018-03-14 Redx Pharma Plc Modulators of Rho-associated protein kinase
CN111718310B (zh) * 2019-08-19 2021-06-11 中国药科大学 苯基取代的五元杂环类化合物及其制备方法、用途和药物组合物
CN110845410B (zh) * 2019-10-29 2021-02-26 暨明医药科技(苏州)有限公司 一种一锅法制备6,7-二甲氧基-3,4-二氢异喹啉盐酸盐的方法
IL310209A (en) * 2021-07-26 2024-03-01 Harvard College ROCK2 inhibitors and their uses
CN113999211B (zh) * 2021-11-23 2022-11-29 郑州大学 一类特异性抗前列腺癌活性的含1,2,3-三氮唑的吲唑骨架衍生物
GB202200735D0 (en) * 2022-01-20 2022-03-09 Redx Pharma Plc Compounds
WO2023182856A1 (ko) * 2022-03-24 2023-09-28 서울대학교산학협력단 로-키나제 억제제를 포함하는 켈로이드 등 피부 섬유화 질환의 예방 또는 치료용 약학적 조성물 및 그의 용도
CN116891460A (zh) * 2023-07-12 2023-10-17 浙江大学 一种吲唑类衍生物或其药用盐及应用

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9207396D0 (en) 1992-04-03 1992-05-13 Merck Sharp & Dohme Therapeutic agents
DE60120193T2 (de) * 2000-09-15 2007-03-29 Vertex Pharmaceuticals Inc., Cambridge Pyrazolverbindungen als protein-kinasehemmer
CL2003002353A1 (es) * 2002-11-15 2005-02-04 Vertex Pharma Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condic
AU2003293376A1 (en) * 2002-12-10 2004-06-30 Imclone Systems Incorporated Anti-angiogenic compounds and their use in cancer treatment
EP1730124A4 (en) * 2004-03-26 2009-04-01 Amphora Discovery Corp Certain compounds based on triazole, compositions and applications thereof
WO2006135383A2 (en) * 2004-08-04 2006-12-21 Myriad Genetics, Inc. Indazoles
AU2007267859B2 (en) 2006-05-25 2012-04-12 Synta Pharmaceuticals Corp. Triazole compounds that modulate Hsp90 activity
DE102007022565A1 (de) * 2007-05-14 2008-11-20 Merck Patent Gmbh Heterocyclische Indazolderivate
CA2727928A1 (en) * 2008-06-18 2009-12-23 Merck Sharp & Dohme Corp. Inhibitors of janus kinases
AU2011232372B2 (en) * 2010-03-24 2016-06-30 Amitech Therapeutic Solutions, Inc. Heterocyclic compounds useful for kinase inhibition
US9061966B2 (en) 2010-10-08 2015-06-23 Oryzon Genomics S.A. Cyclopropylamine inhibitors of oxidases
SI2655357T1 (sl) 2010-12-20 2016-10-28 Merck Serono S.A. Derivati indazolil triazola kot zaviralci IRAK
EP2824099A4 (en) * 2012-03-09 2015-11-11 Carna Biosciences Inc NOVEL TRIAZINE DERIVATIVE
EP3262041A4 (en) * 2015-02-27 2018-08-01 Lycera Corporation Indazolyl thiadiazolamines and related compounds for inhibition of rho-associated protein kinase and the treatment of disease
CO2018006164A2 (es) 2015-12-16 2018-09-20 Loxo Oncology Inc Compuestos útiles como inhibidores de cinasa
EP3421464B1 (en) * 2017-06-30 2021-11-24 Beijing Tide Pharmaceutical Co., Ltd. Rho-associated protein kinase inhibitor, pharmaceutical composition comprising the same, as well as preparation method and use thereof
GB201801226D0 (en) 2018-01-25 2018-03-14 Redx Pharma Plc Modulators of Rho-associated protein kinase

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