JPS63115822A - 生理活性ポリペプチド類の経鼻投与用粉末状組成物 - Google Patents
生理活性ポリペプチド類の経鼻投与用粉末状組成物Info
- Publication number
- JPS63115822A JPS63115822A JP61260636A JP26063686A JPS63115822A JP S63115822 A JPS63115822 A JP S63115822A JP 61260636 A JP61260636 A JP 61260636A JP 26063686 A JP26063686 A JP 26063686A JP S63115822 A JPS63115822 A JP S63115822A
- Authority
- JP
- Japan
- Prior art keywords
- water
- composition according
- absorbing
- composition
- soluble
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
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- VMSNAUAEKXEYGP-YEUHZSMFSA-M sodium glycodeoxycholate Chemical compound [Na+].C([C@H]1CC2)[C@H](O)CC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CC[C@H]([C@@H](CCC(=O)NCC([O-])=O)C)[C@@]2(C)[C@@H](O)C1 VMSNAUAEKXEYGP-YEUHZSMFSA-M 0.000 description 1
- NNMHYFLPFNGQFZ-UHFFFAOYSA-M sodium polyacrylate Chemical compound [Na+].[O-]C(=O)C=C NNMHYFLPFNGQFZ-UHFFFAOYSA-M 0.000 description 1
- 229960004025 sodium salicylate Drugs 0.000 description 1
- 159000000000 sodium salts Chemical class 0.000 description 1
- HJHVQCXHVMGZNC-JCJNLNMISA-M sodium;(2z)-2-[(3r,4s,5s,8s,9s,10s,11r,13r,14s,16s)-16-acetyloxy-3,11-dihydroxy-4,8,10,14-tetramethyl-2,3,4,5,6,7,9,11,12,13,15,16-dodecahydro-1h-cyclopenta[a]phenanthren-17-ylidene]-6-methylhept-5-enoate Chemical compound [Na+].O[C@@H]([C@@H]12)C[C@H]3\C(=C(/CCC=C(C)C)C([O-])=O)[C@@H](OC(C)=O)C[C@]3(C)[C@@]2(C)CC[C@@H]2[C@]1(C)CC[C@@H](O)[C@H]2C HJHVQCXHVMGZNC-JCJNLNMISA-M 0.000 description 1
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- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
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- 229960001322 trypsin Drugs 0.000 description 1
- VBEQCZHXXJYVRD-GACYYNSASA-N uroanthelone Chemical compound C([C@@H](C(=O)N[C@H](C(=O)N[C@@H](CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CS)C(=O)N[C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)NCC(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CS)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O)C(C)C)[C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CC=1NC=NC=1)NC(=O)[C@H](CCSC)NC(=O)[C@H](CS)NC(=O)[C@@H](NC(=O)CNC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CS)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)CNC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](CS)NC(=O)CNC(=O)[C@H]1N(CCC1)C(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(N)=O)C(C)C)[C@@H](C)CC)C1=CC=C(O)C=C1 VBEQCZHXXJYVRD-GACYYNSASA-N 0.000 description 1
- 210000003462 vein Anatomy 0.000 description 1
- OENHQHLEOONYIE-JLTXGRSLSA-N β-Carotene Chemical compound CC=1CCCC(C)(C)C=1\C=C\C(\C)=C\C=C\C(\C)=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C OENHQHLEOONYIE-JLTXGRSLSA-N 0.000 description 1
Landscapes
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP61260636A JPS63115822A (ja) | 1986-11-04 | 1986-11-04 | 生理活性ポリペプチド類の経鼻投与用粉末状組成物 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP61260636A JPS63115822A (ja) | 1986-11-04 | 1986-11-04 | 生理活性ポリペプチド類の経鼻投与用粉末状組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS63115822A true JPS63115822A (ja) | 1988-05-20 |
| JPH0480008B2 JPH0480008B2 (enrdf_load_html_response) | 1992-12-17 |
Family
ID=17350671
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP61260636A Granted JPS63115822A (ja) | 1986-11-04 | 1986-11-04 | 生理活性ポリペプチド類の経鼻投与用粉末状組成物 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS63115822A (enrdf_load_html_response) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1990005535A1 (en) * | 1988-11-14 | 1990-05-31 | Otsuka Pharmaceutical Co., Ltd. | Interferon preparation for nasal administration |
| GB2218098B (en) * | 1988-04-30 | 1991-11-20 | Sandoz Ltd | Acid addition salts of amidated taurine or glycine,their preparation and use |
| GB2303064A (en) * | 1995-07-12 | 1997-02-12 | Ltt Inst Co Ltd | Ion-exchange resin particles for nasal administration of vaccines and peptides |
| WO1998047490A1 (de) * | 1997-04-18 | 1998-10-29 | Roche Diagnostics Gmbh | Stabile pharmazeutische darreichungsform für peptide, proteine und nukleinsäuren |
| US6552074B2 (en) * | 2000-11-16 | 2003-04-22 | Fukumi Morishige | Arginine/ascorbic acid mixed powder as an oral supplement |
| WO2004078211A1 (ja) * | 2003-03-04 | 2004-09-16 | Tanabe Seiyaku Co., Ltd. | 粉末経鼻投与製剤 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56140924A (en) * | 1980-04-04 | 1981-11-04 | Teijin Ltd | Calcitonin pharmaceutical preparation |
| JPS60224616A (ja) * | 1984-04-24 | 1985-11-09 | Teijin Ltd | 経鼻投与用組成物 |
| JPS61118325A (ja) * | 1984-11-12 | 1986-06-05 | Yamanouchi Pharmaceut Co Ltd | 塩基性および／または中性アミノ酸を含有するカルシトニン経鼻剤 |
-
1986
- 1986-11-04 JP JP61260636A patent/JPS63115822A/ja active Granted
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56140924A (en) * | 1980-04-04 | 1981-11-04 | Teijin Ltd | Calcitonin pharmaceutical preparation |
| JPS60224616A (ja) * | 1984-04-24 | 1985-11-09 | Teijin Ltd | 経鼻投与用組成物 |
| JPS61118325A (ja) * | 1984-11-12 | 1986-06-05 | Yamanouchi Pharmaceut Co Ltd | 塩基性および／または中性アミノ酸を含有するカルシトニン経鼻剤 |
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2218098B (en) * | 1988-04-30 | 1991-11-20 | Sandoz Ltd | Acid addition salts of amidated taurine or glycine,their preparation and use |
| WO1990005535A1 (en) * | 1988-11-14 | 1990-05-31 | Otsuka Pharmaceutical Co., Ltd. | Interferon preparation for nasal administration |
| GB2303064A (en) * | 1995-07-12 | 1997-02-12 | Ltt Inst Co Ltd | Ion-exchange resin particles for nasal administration of vaccines and peptides |
| GB2303064B (en) * | 1995-07-12 | 1999-10-06 | Ltt Inst Co Ltd | Medicament for nasal administration |
| WO1998047490A1 (de) * | 1997-04-18 | 1998-10-29 | Roche Diagnostics Gmbh | Stabile pharmazeutische darreichungsform für peptide, proteine und nukleinsäuren |
| AU744777B2 (en) * | 1997-04-18 | 2002-03-07 | Roche Diagnostics Gmbh | Stable pharmaceutical administration forms of peptides, proteins and nucleic acids |
| US6552074B2 (en) * | 2000-11-16 | 2003-04-22 | Fukumi Morishige | Arginine/ascorbic acid mixed powder as an oral supplement |
| US7214709B2 (en) | 2000-11-16 | 2007-05-08 | Eiji Kimoto | Arginine/ascorbic acid mixed powder as an oral supplement |
| WO2004078211A1 (ja) * | 2003-03-04 | 2004-09-16 | Tanabe Seiyaku Co., Ltd. | 粉末経鼻投与製剤 |
| US7591999B2 (en) | 2003-03-04 | 2009-09-22 | Mitsubishi Tanabe Pharma Corporation | Powdery preparation for nasal administration |
Also Published As
| Publication number | Publication date |
|---|---|
| JPH0480008B2 (enrdf_load_html_response) | 1992-12-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EXPY | Cancellation because of completion of term |