JPS6284082A - ２−オキソ−１−〔〔（置換スルホニル）アミノ〕カルボニル〕アゼチジン類 - Google Patents

２−オキソ−１−〔〔（置換スルホニル）アミノ〕カルボニル〕アゼチジン類

Info

Publication number
JPS6284082A
JPS6284082A JP61229474A JP22947486A JPS6284082A JP S6284082 A JPS6284082 A JP S6284082A JP 61229474 A JP61229474 A JP 61229474A JP 22947486 A JP22947486 A JP 22947486A JP S6284082 A JPS6284082 A JP S6284082A
Authority
JP
Japan
Prior art keywords
amino
oxo
formulas
tables
carbonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP61229474A
Other languages
English (en)
Japanese (ja)
Inventor
ヘルマン・ブロイエル
ウウエ・デー・トロイネル
ウィリアム・エイチ・コスター
ロバート・ザーラー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of JPS6284082A publication Critical patent/JPS6284082A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
JP61229474A 1985-09-26 1986-09-26 ２−オキソ−１−〔〔（置換スルホニル）アミノ〕カルボニル〕アゼチジン類 Pending JPS6284082A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78047985A 1985-09-26 1985-09-26
US780479 1985-09-26

Publications (1)

Publication Number Publication Date
JPS6284082A true JPS6284082A (ja) 1987-04-17

Family

ID=25119699

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61229474A Pending JPS6284082A (ja) 1985-09-26 1986-09-26 ２−オキソ−１−〔〔（置換スルホニル）アミノ〕カルボニル〕アゼチジン類

Country Status (31)

Country Link
JP (1) JPS6284082A (sv)
KR (1) KR900001013B1 (sv)
CN (1) CN86106980A (sv)
AT (1) ATA257986A (sv)
AU (1) AU600912B2 (sv)
BE (1) BE905502A (sv)
CA (1) CA1308719C (sv)
CH (1) CH670828A5 (sv)
DD (1) DD250121A5 (sv)
DE (1) DE3632876A1 (sv)
DK (1) DK460386A (sv)
EG (1) EG18314A (sv)
ES (1) ES2001995A6 (sv)
FI (1) FI863890A (sv)
FR (1) FR2587700B1 (sv)
GB (1) GB2181130B (sv)
GR (1) GR862449B (sv)
HU (1) HU198044B (sv)
IE (1) IE59686B1 (sv)
IL (1) IL80160A (sv)
IT (1) IT1214533B (sv)
LU (1) LU86611A1 (sv)
NL (1) NL8602446A (sv)
NO (1) NO863837L (sv)
NZ (1) NZ217704A (sv)
PH (1) PH23315A (sv)
PL (1) PL151546B1 (sv)
PT (1) PT83440B (sv)
SE (1) SE8604089L (sv)
YU (1) YU46177B (sv)
ZA (1) ZA867373B (sv)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013073577A1 (ja) * 2011-11-15 2013-05-23 アステラス製薬株式会社 ジヒドロキシ芳香族へテロ環化合物
US9180122B2 (en) 2011-07-07 2015-11-10 Takeda Pharmaceutical Company Limited 5- or 6-substituted 3-hydroxy-2 (1 H)-pyridinones as D-amino acid oxidase (DAAO) inhibitors in therapy of diseases such as schizophrenia, cognitive disorder and pain
US9290456B2 (en) 2011-08-22 2016-03-22 Takeda Pharmaceutical Company Limited Pyridazinone compounds and their use as DAAO inhibitors
US9750748B2 (en) 2012-12-17 2017-09-05 Takeda Pharmaceutical Company Limited Pyridazinones as DAAO enzyme inhibitors
US10085986B2 (en) 2011-07-07 2018-10-02 Takeda Pharmaceutical Company Limited Pyrimidinone compounds and their use

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU7541487A (en) * 1986-05-23 1987-12-22 Upjohn Company, The N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams
US5006650A (en) * 1987-02-11 1991-04-09 The Upjohn Company Novel N-1 substituted beta-lactams as antibiotics
WO1988006156A1 (en) * 1987-02-11 1988-08-25 The Upjohn Company NOVEL N-1 SUBSTITUTED beta-LACTAMS AS ANTIBIOTICS
WO1988006587A1 (en) * 1987-02-27 1988-09-07 The Upjohn Company ANTIBIOTIC beta-LACTAMS CONTAINING A PYRIDONE CARBOXYLIC ACID OR ACID DERIVATIVE
CA1317298C (en) * 1987-03-03 1993-05-04 Upjohn Company (The) Antibiotic sulfonylaminocarbonyl activated .beta.-lactams
US4762922A (en) * 1987-07-01 1988-08-09 Squibb Corporation 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4772693A (en) * 1987-07-01 1988-09-20 E. R. Squibb & Sons, Inc. 2-oxo-1-((Substituted sulfonyl)amino)-carbonyl)azetidines
EP0368908A1 (en) * 1987-07-22 1990-05-23 The Upjohn Company THERAPEUTICALLY USEFUL $g(b)-LACTAMS
US5015737A (en) * 1987-07-22 1991-05-14 The Upjohn Company Therapeutically useful beta-lactams
US4777252A (en) * 1987-08-13 1988-10-11 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4889930A (en) * 1987-12-21 1989-12-26 E. R. Squibb & Sons, Inc. Process for making 2-oxo-1-((substituted sulfonyl)amino)carbonzyl)azetidines and intermediates used therein
US4871841A (en) * 1987-12-23 1989-10-03 E. R. Squibb & Sons, Inc. 2-Oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
EP0336667A3 (en) * 1988-04-04 1991-04-10 E.R. Squibb & Sons, Inc. [3S(Z)]-3-[[(2-amino-4-thiazolyl)[[2-(hydroxyamino)-2-oxoethoxy]imino]acetyl]-amino]-2,2-dimethyl-4-oxo-1-azetidinyl sulfate
US4959470A (en) * 1988-08-17 1990-09-25 E. R. Squibb & Sons, Inc. 2-oxo-[[(substituted sulfonyl)-amino]carbonyl]-azetidines
EP0604365B1 (en) * 1992-12-23 1999-05-26 Novartis AG Imidazole derivatives and their use as agrochemical agents
DE69405535T2 (de) * 1994-03-11 1998-04-02 Agfa Gevaert Nv Photographisches Material, das einen neuen Typ eines Hydrazides enthält
US7511159B2 (en) * 2003-12-25 2009-03-31 Ono Pharmaceutical Co., Ltd. Azetidine ring compounds and drugs comprising the same
CN106986820B (zh) * 2017-02-24 2019-05-21 浙江工商大学 多功能的羟基吡啶酮衍生物及其水合物的制备法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
CA1272726C (en) * 1982-01-04 1990-08-14 2-oxo-1-(aminocarbonylaminosulfonyl- aminocarbonyl)azetidines
US4939253A (en) * 1982-08-04 1990-07-03 E. R. Squibb & Sons, Inc. 2-oxoazetidin-1-yloxy acetic acids and analogs
US4801705A (en) * 1986-06-23 1989-01-31 E. R. Squibb & Sons, Inc. 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9180122B2 (en) 2011-07-07 2015-11-10 Takeda Pharmaceutical Company Limited 5- or 6-substituted 3-hydroxy-2 (1 H)-pyridinones as D-amino acid oxidase (DAAO) inhibitors in therapy of diseases such as schizophrenia, cognitive disorder and pain
US10085986B2 (en) 2011-07-07 2018-10-02 Takeda Pharmaceutical Company Limited Pyrimidinone compounds and their use
US9290456B2 (en) 2011-08-22 2016-03-22 Takeda Pharmaceutical Company Limited Pyridazinone compounds and their use as DAAO inhibitors
US9931340B2 (en) 2011-08-22 2018-04-03 Takeda Pharmaceutical Company Limited Pyridazinone compounds and their use as DAAO inhibitors
US10463663B2 (en) 2011-08-22 2019-11-05 Takeda Pharmaceutical Company Limited Pyridazinone compounds and their use as DAAO inhibitors
US11129828B2 (en) 2011-08-22 2021-09-28 Takeda Pharmaceutical Company Limited Pyridazinone compounds and their use as DAAO inhibitors
WO2013073577A1 (ja) * 2011-11-15 2013-05-23 アステラス製薬株式会社 ジヒドロキシ芳香族へテロ環化合物
US9212147B2 (en) 2011-11-15 2015-12-15 Takeda Pharmaceutical Company Limited Dihydroxy aromatic heterocyclic compound
US9562020B2 (en) 2011-11-15 2017-02-07 Takeda Pharmaceutical Company Limited Dihydroxy aromatic heterocyclic compound
US10202399B2 (en) 2011-11-15 2019-02-12 Takeda Pharmaceutical Company Limited Dihydroxy aromatic heterocyclic compound
US9750748B2 (en) 2012-12-17 2017-09-05 Takeda Pharmaceutical Company Limited Pyridazinones as DAAO enzyme inhibitors

Also Published As

Publication number Publication date
FI863890A (fi) 1987-03-27
FI863890A0 (fi) 1986-09-26
DE3632876A1 (de) 1987-04-02
KR900001013B1 (ko) 1990-02-24
CH670828A5 (sv) 1989-07-14
AU6315686A (en) 1987-04-02
NL8602446A (nl) 1987-04-16
FR2587700B1 (fr) 1988-09-16
DK460386A (da) 1987-03-27
ATA257986A (de) 1994-07-15
IE59686B1 (en) 1994-03-23
NO863837L (no) 1987-03-27
HU198044B (en) 1989-07-28
CA1308719C (en) 1992-10-13
IT1214533B (it) 1990-01-18
DK460386D0 (da) 1986-09-26
BE905502A (fr) 1987-01-16
SE8604089L (sv) 1987-03-27
HUT44535A (en) 1988-03-28
EG18314A (en) 1993-02-28
GB2181130B (en) 1989-09-20
LU86611A1 (fr) 1987-04-02
GR862449B (en) 1987-01-27
ZA867373B (en) 1987-05-27
ES2001995A6 (es) 1988-07-01
YU46177B (sh) 1993-05-28
YU165986A (en) 1988-06-30
PT83440B (pt) 1989-05-12
CN86106980A (zh) 1987-04-08
NO863837D0 (no) 1986-09-26
DD250121A5 (de) 1987-09-30
IT8621834A0 (it) 1986-09-26
GB8623151D0 (en) 1986-10-29
IL80160A0 (en) 1986-12-31
PH23315A (en) 1989-07-14
PT83440A (pt) 1986-10-01
PL261575A1 (en) 1988-07-21
NZ217704A (en) 1989-02-24
PL151546B1 (en) 1990-09-28
KR870003101A (ko) 1987-04-15
FR2587700A1 (fr) 1987-03-27
IE862547L (en) 1987-03-26
GB2181130A (en) 1987-04-15
IL80160A (en) 1991-04-15
AU600912B2 (en) 1990-08-30
SE8604089D0 (sv) 1986-09-26

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