JPS62221665A - アゼチジノンの製造法及び中間体 - Google Patents

アゼチジノンの製造法及び中間体

Info

Publication number
JPS62221665A
JPS62221665A JP62056399A JP5639987A JPS62221665A JP S62221665 A JPS62221665 A JP S62221665A JP 62056399 A JP62056399 A JP 62056399A JP 5639987 A JP5639987 A JP 5639987A JP S62221665 A JPS62221665 A JP S62221665A
Authority
JP
Japan
Prior art keywords
formula
compound
phenyl
tables
formulas
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP62056399A
Other languages
English (en)
Japanese (ja)
Inventor
サムエル・チャッカラマニル
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Schering Plough Corp
Original Assignee
Schering Plough Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Plough Corp filed Critical Schering Plough Corp
Publication of JPS62221665A publication Critical patent/JPS62221665A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
JP62056399A 1986-03-13 1987-03-11 アゼチジノンの製造法及び中間体 Pending JPS62221665A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/839,307 US4740595A (en) 1986-03-13 1986-03-13 Preparation of azetidinones via N-protected oxirancecarboxamide intermediates
US839307 1986-03-13

Publications (1)

Publication Number Publication Date
JPS62221665A true JPS62221665A (ja) 1987-09-29

Family

ID=25279384

Family Applications (1)

Application Number Title Priority Date Filing Date
JP62056399A Pending JPS62221665A (ja) 1986-03-13 1987-03-11 アゼチジノンの製造法及び中間体

Country Status (7)

Country Link
US (1) US4740595A (enExample)
EP (1) EP0238252B1 (enExample)
JP (1) JPS62221665A (enExample)
AT (1) ATE76065T1 (enExample)
DE (1) DE3778946D1 (enExample)
ES (1) ES2032201T3 (enExample)
GR (1) GR3005360T3 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4876365A (en) * 1988-12-05 1989-10-24 Schering Corporation Intermediate compounds for preparing penems and carbapenems
US5075439A (en) * 1990-08-17 1991-12-24 Pfizer Inc. Processes for (3S,4R)-3-[1(R)-t-butyl-dimethylsilyloxy)-ethyl]-4-[1-oxo-3-thiolanylthio(thiocarbonyl)thio]azetidin-2-ones and intermediates therefor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0126709B1 (de) * 1983-03-28 1991-04-03 Ciba-Geigy Ag Verfahren zur Herstellung von optisch aktiven Azetidinonen
ATE93520T1 (de) * 1984-10-01 1993-09-15 Ciba Geigy Ag Verfahren zur herstellung von optisch aktiven acyloxyazetidinonen.

Also Published As

Publication number Publication date
ATE76065T1 (de) 1992-05-15
US4740595A (en) 1988-04-26
EP0238252B1 (en) 1992-05-13
EP0238252A3 (en) 1987-12-02
DE3778946D1 (de) 1992-06-17
EP0238252A2 (en) 1987-09-23
ES2032201T3 (es) 1993-01-16
GR3005360T3 (enExample) 1993-05-24

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