JPS5962595A - 3,5,7―トリ置換―トリアゾロピリミジン誘導体 - Google Patents
3,5,7―トリ置換―トリアゾロピリミジン誘導体Info
- Publication number
- JPS5962595A JPS5962595A JP17117382A JP17117382A JPS5962595A JP S5962595 A JPS5962595 A JP S5962595A JP 17117382 A JP17117382 A JP 17117382A JP 17117382 A JP17117382 A JP 17117382A JP S5962595 A JPS5962595 A JP S5962595A
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituent
- groups
- formula
- following general
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17117382A JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17117382A JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5962595A true JPS5962595A (ja) | 1984-04-10 |
JPH0366310B2 JPH0366310B2 (en, 2012) | 1991-10-16 |
Family
ID=15918347
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP17117382A Granted JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5962595A (en, 2012) |
Cited By (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5204353A (en) * | 1987-04-07 | 1993-04-20 | Ciba-Geigy Corporation | 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith |
US6124300A (en) * | 1996-03-26 | 2000-09-26 | Dupont Pharmaceuticals | Aryloxy- and arylthio- fused pyridines and pyrimidines and derivatives |
EP0901476A4 (en) * | 1996-03-26 | 2001-08-16 | Du Pont Pharm Co | PYRIDINES AND PYRIMIDINES FUSION ARYLOXY AND ARYLTHIO AND DERIVATIVES THEREOF |
WO2004018473A3 (en) * | 2002-08-23 | 2004-05-21 | Inst Of Ex Botany Ascr | Azapurine derivatives |
US7141575B2 (en) | 2001-01-10 | 2006-11-28 | Vernalis Research Ltd. | Triazolo[4,5-d]pyrimidine derivatives and their use as purinergic receptor antagonists |
US7285550B2 (en) | 2003-04-09 | 2007-10-23 | Biogen Idec Ma Inc. | Triazolotriazines and pyrazolotriazines and methods of making and using the same |
US7674791B2 (en) | 2003-04-09 | 2010-03-09 | Biogen Idec Ma Inc. | Triazolopyrazines and methods of making and using the same |
US7834014B2 (en) | 2003-04-09 | 2010-11-16 | Biogen Idec Ma Inc. | A2a adenosine receptor antagonists |
US8236809B2 (en) | 2004-05-18 | 2012-08-07 | Vasopharm Gmbh | Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation |
US8450328B2 (en) | 2008-06-25 | 2013-05-28 | Vernalis (R&D) Limited | Triazolo[4,5-D]pyramidine derivatives and their use as purine receptor antagonists |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS56131587A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | 7-substituted triazolopyrimidine derivative and its preparation |
JPS56131586A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | Triazolopyrimidine derivative and its preparation |
-
1982
- 1982-09-30 JP JP17117382A patent/JPS5962595A/ja active Granted
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS56131587A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | 7-substituted triazolopyrimidine derivative and its preparation |
JPS56131586A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | Triazolopyrimidine derivative and its preparation |
Cited By (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5204353A (en) * | 1987-04-07 | 1993-04-20 | Ciba-Geigy Corporation | 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith |
US6124300A (en) * | 1996-03-26 | 2000-09-26 | Dupont Pharmaceuticals | Aryloxy- and arylthio- fused pyridines and pyrimidines and derivatives |
US6258809B1 (en) | 1996-03-26 | 2001-07-10 | Dupont Pharmaceuticals Company | 6-aryloxy and arylthiopurines |
EP0901476A4 (en) * | 1996-03-26 | 2001-08-16 | Du Pont Pharm Co | PYRIDINES AND PYRIMIDINES FUSION ARYLOXY AND ARYLTHIO AND DERIVATIVES THEREOF |
US7405219B2 (en) | 2001-01-10 | 2008-07-29 | Vernalis Research Limited | Triazolo [4,5-d] pyrimidine derivatives and their use as purinergic receptor antagonists |
US7141575B2 (en) | 2001-01-10 | 2006-11-28 | Vernalis Research Ltd. | Triazolo[4,5-d]pyrimidine derivatives and their use as purinergic receptor antagonists |
US7589097B2 (en) | 2001-01-10 | 2009-09-15 | Vernalis Research Limited | Triazol[4,5-d] pyramidine derivatives and their use as purinergic receptor antagonists |
US7816350B2 (en) | 2002-08-23 | 2010-10-19 | Institute Of Experimental Botany Ascr | Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors |
WO2004018473A3 (en) * | 2002-08-23 | 2004-05-21 | Inst Of Ex Botany Ascr | Azapurine derivatives |
US7285550B2 (en) | 2003-04-09 | 2007-10-23 | Biogen Idec Ma Inc. | Triazolotriazines and pyrazolotriazines and methods of making and using the same |
US7674791B2 (en) | 2003-04-09 | 2010-03-09 | Biogen Idec Ma Inc. | Triazolopyrazines and methods of making and using the same |
US7834014B2 (en) | 2003-04-09 | 2010-11-16 | Biogen Idec Ma Inc. | A2a adenosine receptor antagonists |
US8236809B2 (en) | 2004-05-18 | 2012-08-07 | Vasopharm Gmbh | Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation |
US8987279B2 (en) | 2008-06-25 | 2015-03-24 | Vernalis (R&D) Limited | Triazolo [4, 5-D] pyramidine derivatives and their use as purine receptor antagonists |
US8450328B2 (en) | 2008-06-25 | 2013-05-28 | Vernalis (R&D) Limited | Triazolo[4,5-D]pyramidine derivatives and their use as purine receptor antagonists |
US9376443B2 (en) | 2008-06-25 | 2016-06-28 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US9765080B2 (en) | 2008-06-25 | 2017-09-19 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10106547B2 (en) | 2008-06-25 | 2018-10-23 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10538526B2 (en) | 2008-06-25 | 2020-01-21 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10875868B2 (en) | 2008-06-25 | 2020-12-29 | Vernalis (R&D) Limited | Triazolo[4,5-d] pyramidine derivatives and their use as purine receptor antagonists |
US11466019B2 (en) | 2008-06-25 | 2022-10-11 | Vernalis (R&D) Limited | Triazolo[4,5-d] pyramidine derivatives and their use as purine receptor antagonists |
Also Published As
Publication number | Publication date |
---|---|
JPH0366310B2 (en, 2012) | 1991-10-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CN105026400A (zh) | 用于制备药物的方法和中间体 | |
JPS5962595A (ja) | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 | |
EP0009384A1 (en) | Processes for the preparation of triazinones and condensed triazinones, and compounds so obtained | |
JPS634544B2 (en, 2012) | ||
JPS58192872A (ja) | 含窒素化合物、その製法および該化合物を含有する、降圧作用を有する製薬組成物 | |
JPS634543B2 (en, 2012) | ||
WO1984000957A1 (en) | 4-amino-tetrahydro-2-naphthoic acid derivatives | |
Santana et al. | Synthesis of 1, 2-disubstituted carbocyclic analogs of pyrimidine and purine nucleosides | |
CN112778317A (zh) | 一种[1,2,4]三氮唑并[1,5-a]嘧啶类化合物的合成方法 | |
SU564809A3 (ru) | Способ получени 6-аза-1,2дигидро-3н-1,4-бензодиазепинов или их солей | |
JPS5962593A (ja) | 3―置換―5,7―ジクロルトリアゾロピリミジン誘導体 | |
JP4138883B2 (ja) | アクリドン誘導体及び8―ヒドロキシイミダゾアクリジノン誘導体の製造方法 | |
JPS5962594A (ja) | 3,5―ジ置換―トリアゾロピリミジン誘導体 | |
US3205236A (en) | Process of preparation of /j-alkylated tryptamines | |
CN112142663B (zh) | (s)-1-苯基-1,2,3,4-四氢异喹啉的合成方法 | |
CN112250533B (zh) | (s)-1-(3-乙氧基-4-甲氧基苯基)-2-(甲磺酰基)乙胺的合成方法 | |
JPS5951288A (ja) | 新規な9−ニトロカンプトテシン及びその製造法 | |
JPS623150B2 (en, 2012) | ||
SU492517A1 (ru) | Способ получени 1-/ -аминофенил/-3 -/ -аминофенил/-7н-пирмдо-/2,3-с/карбазола | |
SU595312A1 (ru) | Способ получени 2,4,6-замещенных перхлоратов пиримидини | |
CN118580235A (zh) | 一种内磺酰胺化合物的制备方法 | |
BE535830A (en, 2012) | ||
CN120112512A (zh) | 制备(z)-3-(2-(5-溴-1h-吲哚-3-基)-2-氰基乙烯基)-4-甲氧基苯甲腈的方法 | |
JPS595147A (ja) | 2−アミノ−1−フエニル−1−プロパノ−ル誘導体の製造法 | |
FR2606017A1 (fr) | Derives cycliques condenses du triazole, procede de preparation, compositions pharmaceutiques les contenant et leur utilisation comme sedatif et tranquilisant |