JPS5962595A - 3,5,7―トリ置換―トリアゾロピリミジン誘導体 - Google Patents
3,5,7―トリ置換―トリアゾロピリミジン誘導体Info
- Publication number
- JPS5962595A JPS5962595A JP17117382A JP17117382A JPS5962595A JP S5962595 A JPS5962595 A JP S5962595A JP 17117382 A JP17117382 A JP 17117382A JP 17117382 A JP17117382 A JP 17117382A JP S5962595 A JPS5962595 A JP S5962595A
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- substituent
- groups
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17117382A JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17117382A JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5962595A true JPS5962595A (ja) | 1984-04-10 |
JPH0366310B2 JPH0366310B2 (US07943777-20110517-C00090.png) | 1991-10-16 |
Family
ID=15918347
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP17117382A Granted JPS5962595A (ja) | 1982-09-30 | 1982-09-30 | 3,5,7―トリ置換―トリアゾロピリミジン誘導体 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5962595A (US07943777-20110517-C00090.png) |
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5204353A (en) * | 1987-04-07 | 1993-04-20 | Ciba-Geigy Corporation | 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith |
WO1997035539A2 (en) * | 1996-03-27 | 1997-10-02 | Du Pont Pharmaceuticals Company | Arylamino fused pyridines and pyrimidines |
EP0901476A1 (en) * | 1996-03-26 | 1999-03-17 | Du Pont Pharmaceuticals Company | Aryloxy- and arylthio-fused pyridines and pyrimidines and derivatives |
US6124300A (en) * | 1996-03-26 | 2000-09-26 | Dupont Pharmaceuticals | Aryloxy- and arylthio- fused pyridines and pyrimidines and derivatives |
WO2004018473A3 (en) * | 2002-08-23 | 2004-05-21 | Inst Of Ex Botany Ascr | Azapurine derivatives |
US7141575B2 (en) | 2001-01-10 | 2006-11-28 | Vernalis Research Ltd. | Triazolo[4,5-d]pyrimidine derivatives and their use as purinergic receptor antagonists |
US7285550B2 (en) | 2003-04-09 | 2007-10-23 | Biogen Idec Ma Inc. | Triazolotriazines and pyrazolotriazines and methods of making and using the same |
US7674791B2 (en) | 2003-04-09 | 2010-03-09 | Biogen Idec Ma Inc. | Triazolopyrazines and methods of making and using the same |
US7834014B2 (en) | 2003-04-09 | 2010-11-16 | Biogen Idec Ma Inc. | A2a adenosine receptor antagonists |
US8236809B2 (en) | 2004-05-18 | 2012-08-07 | Vasopharm Gmbh | Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation |
US8450328B2 (en) | 2008-06-25 | 2013-05-28 | Vernalis (R&D) Limited | Triazolo[4,5-D]pyramidine derivatives and their use as purine receptor antagonists |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS56131587A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | 7-substituted triazolopyrimidine derivative and its preparation |
JPS56131586A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | Triazolopyrimidine derivative and its preparation |
-
1982
- 1982-09-30 JP JP17117382A patent/JPS5962595A/ja active Granted
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS56131587A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | 7-substituted triazolopyrimidine derivative and its preparation |
JPS56131586A (en) * | 1980-03-18 | 1981-10-15 | Ss Pharmaceut Co Ltd | Triazolopyrimidine derivative and its preparation |
Cited By (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5204353A (en) * | 1987-04-07 | 1993-04-20 | Ciba-Geigy Corporation | 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith |
EP0901476A1 (en) * | 1996-03-26 | 1999-03-17 | Du Pont Pharmaceuticals Company | Aryloxy- and arylthio-fused pyridines and pyrimidines and derivatives |
US6124300A (en) * | 1996-03-26 | 2000-09-26 | Dupont Pharmaceuticals | Aryloxy- and arylthio- fused pyridines and pyrimidines and derivatives |
US6258809B1 (en) | 1996-03-26 | 2001-07-10 | Dupont Pharmaceuticals Company | 6-aryloxy and arylthiopurines |
EP0901476A4 (en) * | 1996-03-26 | 2001-08-16 | Du Pont Pharm Co | PYRIDINES AND PYRIMIDINES FUSION ARYLOXY AND ARYLTHIO AND DERIVATIVES THEREOF |
WO1997035539A2 (en) * | 1996-03-27 | 1997-10-02 | Du Pont Pharmaceuticals Company | Arylamino fused pyridines and pyrimidines |
US7589097B2 (en) | 2001-01-10 | 2009-09-15 | Vernalis Research Limited | Triazol[4,5-d] pyramidine derivatives and their use as purinergic receptor antagonists |
US7141575B2 (en) | 2001-01-10 | 2006-11-28 | Vernalis Research Ltd. | Triazolo[4,5-d]pyrimidine derivatives and their use as purinergic receptor antagonists |
US7405219B2 (en) | 2001-01-10 | 2008-07-29 | Vernalis Research Limited | Triazolo [4,5-d] pyrimidine derivatives and their use as purinergic receptor antagonists |
WO2004018473A3 (en) * | 2002-08-23 | 2004-05-21 | Inst Of Ex Botany Ascr | Azapurine derivatives |
US7816350B2 (en) | 2002-08-23 | 2010-10-19 | Institute Of Experimental Botany Ascr | Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors |
US7285550B2 (en) | 2003-04-09 | 2007-10-23 | Biogen Idec Ma Inc. | Triazolotriazines and pyrazolotriazines and methods of making and using the same |
US7674791B2 (en) | 2003-04-09 | 2010-03-09 | Biogen Idec Ma Inc. | Triazolopyrazines and methods of making and using the same |
US7834014B2 (en) | 2003-04-09 | 2010-11-16 | Biogen Idec Ma Inc. | A2a adenosine receptor antagonists |
US8236809B2 (en) | 2004-05-18 | 2012-08-07 | Vasopharm Gmbh | Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation |
US8450328B2 (en) | 2008-06-25 | 2013-05-28 | Vernalis (R&D) Limited | Triazolo[4,5-D]pyramidine derivatives and their use as purine receptor antagonists |
US8987279B2 (en) | 2008-06-25 | 2015-03-24 | Vernalis (R&D) Limited | Triazolo [4, 5-D] pyramidine derivatives and their use as purine receptor antagonists |
US9376443B2 (en) | 2008-06-25 | 2016-06-28 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US9765080B2 (en) | 2008-06-25 | 2017-09-19 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10106547B2 (en) | 2008-06-25 | 2018-10-23 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10538526B2 (en) | 2008-06-25 | 2020-01-21 | Vernalis (R&D) Limited | Triazolo[4,5-D] pyramidine derivatives and their use as purine receptor antagonists |
US10875868B2 (en) | 2008-06-25 | 2020-12-29 | Vernalis (R&D) Limited | Triazolo[4,5-d] pyramidine derivatives and their use as purine receptor antagonists |
US11466019B2 (en) | 2008-06-25 | 2022-10-11 | Vernalis (R&D) Limited | Triazolo[4,5-d] pyramidine derivatives and their use as purine receptor antagonists |
Also Published As
Publication number | Publication date |
---|---|
JPH0366310B2 (US07943777-20110517-C00090.png) | 1991-10-16 |
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