JPS5913798A - チロシン誘導体、それらの製造方法およびそれらを含有する医薬組成物 - Google Patents

チロシン誘導体、それらの製造方法およびそれらを含有する医薬組成物

Info

Publication number
JPS5913798A
JPS5913798A JP58116819A JP11681983A JPS5913798A JP S5913798 A JPS5913798 A JP S5913798A JP 58116819 A JP58116819 A JP 58116819A JP 11681983 A JP11681983 A JP 11681983A JP S5913798 A JPS5913798 A JP S5913798A
Authority
JP
Japan
Prior art keywords
acyl
imino
tyrosine
formula
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP58116819A
Other languages
English (en)
Japanese (ja)
Inventor
アラン・ケイス・モ−ラムズ
アシト・クマル・ガングリ−
イ−ツン・リウ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Schering Plough Corp
Original Assignee
Schering Plough Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Plough Corp filed Critical Schering Plough Corp
Publication of JPS5913798A publication Critical patent/JPS5913798A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
JP58116819A 1982-06-30 1983-06-28 チロシン誘導体、それらの製造方法およびそれらを含有する医薬組成物 Pending JPS5913798A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/393,901 US4436729A (en) 1982-06-30 1982-06-30 23-Demycinosyltylosin compounds, pharmaceutical compositions and method of use
US393901 1982-06-30

Publications (1)

Publication Number Publication Date
JPS5913798A true JPS5913798A (ja) 1984-01-24

Family

ID=23556716

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58116819A Pending JPS5913798A (ja) 1982-06-30 1983-06-28 チロシン誘導体、それらの製造方法およびそれらを含有する医薬組成物

Country Status (16)

Country Link
US (1) US4436729A (Direct)
EP (1) EP0097925B1 (Direct)
JP (1) JPS5913798A (Direct)
AT (1) ATE24914T1 (Direct)
AU (1) AU555788B2 (Direct)
CA (1) CA1241952A (Direct)
DE (1) DE3369142D1 (Direct)
DK (1) DK297883D0 (Direct)
GR (1) GR77522B (Direct)
HU (1) HU194270B (Direct)
IE (1) IE55267B1 (Direct)
IL (1) IL69086A0 (Direct)
NZ (1) NZ204718A (Direct)
PH (1) PH18303A (Direct)
PT (1) PT76936B (Direct)
ZA (1) ZA834692B (Direct)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4452784A (en) * 1982-07-19 1984-06-05 Eli Lilly And Company C-23-Modified derivatives of DMT
US4820695A (en) * 1982-09-13 1989-04-11 Eli Lilly And Company C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
US4851518A (en) * 1985-12-23 1989-07-25 Schering Corporation Di and tri-O-acetyl-"O-iso-valeryl-23-O-demycinosyl tylosins, hydrazone derivatives thereof and processes for their preparation
US4920103A (en) * 1986-09-29 1990-04-24 Eli Lilly And Company Modifications of mycinose and 3-O-demethylmycinose in tylosin-type macrolides
US4919804A (en) * 1988-03-01 1990-04-24 University Of Florida Ultrasound driven synthesis of reversed and normal phase stationary phases for liquid chromatography
US4933439A (en) * 1988-06-21 1990-06-12 Sanraku Incorporated Tylosin derivatives and processes for producing the same
US6753415B2 (en) * 2002-04-19 2004-06-22 Enanta Pharmaceuticals, Inc. 23-O-substituted 5-O-mycaminosyltylonide derivatives
US6710034B2 (en) 2002-04-19 2004-03-23 Enanta Pharmaceuticals, Inc. 5-O-mycaminosyltylonide derivatives

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH630391A5 (en) * 1975-02-28 1982-06-15 Scherico Ltd Process for preparing derivatives of rosaramicin
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4321361A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company Demycinosyltylosin and process for its production
US4334019A (en) 1980-06-12 1982-06-08 Eli Lilly And Company Process for producing de(mycinosyloxy)tylosin
US4279896A (en) 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents
US4438109A (en) * 1980-07-25 1984-03-20 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Tylosin derivatives
US4299953A (en) 1980-07-29 1981-11-10 Eli Lilly And Company Mycarosyltylactone
US4341770A (en) * 1981-04-20 1982-07-27 Eli Lilly And Company Method of controlling ureaplasma infections
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58219197A (ja) * 1982-06-15 1983-12-20 Sanraku Inc マクロライド系抗生物質の誘導体
US4452784A (en) * 1982-07-19 1984-06-05 Eli Lilly And Company C-23-Modified derivatives of DMT

Also Published As

Publication number Publication date
PT76936B (en) 1986-04-09
PT76936A (en) 1983-07-01
IE831491L (en) 1983-12-30
DE3369142D1 (en) 1987-02-19
DK297883D0 (da) 1983-06-28
AU555788B2 (en) 1986-10-09
IL69086A0 (en) 1983-10-31
ATE24914T1 (de) 1987-01-15
CA1241952A (en) 1988-09-13
AU1630683A (en) 1984-01-05
PH18303A (en) 1985-05-29
EP0097925A1 (en) 1984-01-11
ZA834692B (en) 1984-03-28
HU194270B (en) 1988-01-28
EP0097925B1 (en) 1987-01-14
GR77522B (Direct) 1984-09-24
IE55267B1 (en) 1990-07-18
NZ204718A (en) 1986-05-09
US4436729A (en) 1984-03-13

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