JPS57209296A - Tylosin derivative - Google Patents
Tylosin derivativeInfo
- Publication number
- JPS57209296A JPS57209296A JP56093782A JP9378281A JPS57209296A JP S57209296 A JPS57209296 A JP S57209296A JP 56093782 A JP56093782 A JP 56093782A JP 9378281 A JP9378281 A JP 9378281A JP S57209296 A JPS57209296 A JP S57209296A
- Authority
- JP
- Japan
- Prior art keywords
- lower alkyl
- compound
- tetrazol
- deoxy
- thio
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:The compound of formulaI[R1 is (lower alkyl) thiomethyloxy, mono- or di-(lower alkyl)amino(lower alkyl)-thio, or (substituted) heterocyclic- thio; R2 is H or OH].
EXAMPLE: 23-Deoxy-23-(1-methyl-1H-tetrazol-5-ylthio)mycaminosyl tylonolide.
USE: Antibacterial agent.
PROCESS: The compound of formulaIcan be prepared, e.g. by reacting the compound of formula II (R5 is protected aldehyde group; X is halogen) (e.g. 23- deoxy-23-iodomycaminosyl tylonolide diethylacetal) with the compound of formula R7-SH[R7 is mono- or di-(lower alkyl)amino(lower alkyl), or (substituted) heterocyclic group](e.g. 1-methyl-1H-tetrazol-5-ylthiol), and removing the aldehyde-protecting group.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP56093782A JPS57209296A (en) | 1981-06-19 | 1981-06-19 | Tylosin derivative |
US06/285,747 US4438109A (en) | 1980-07-25 | 1981-07-22 | Tylosin derivatives |
GB8122796A GB2081711B (en) | 1980-07-25 | 1981-07-23 | Tylosin derivatives |
DE19813129112 DE3129112A1 (en) | 1980-07-25 | 1981-07-23 | TYLOSIN DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
CA000382401A CA1202621A (en) | 1980-07-25 | 1981-07-23 | Process for producing tylosin derivatives |
CH4830/81A CH650513A5 (en) | 1980-07-25 | 1981-07-24 | TYLOSIN DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF. |
FR8114456A FR2495620A1 (en) | 1980-07-25 | 1981-07-24 | DERIVATIVES OF TYLOSINE |
ES514430A ES514430A0 (en) | 1980-11-06 | 1982-07-27 | A PROCEDURE FOR THE PRODUCTION OF A THYLOSINE DERIVATIVE. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP56093782A JPS57209296A (en) | 1981-06-19 | 1981-06-19 | Tylosin derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS57209296A true JPS57209296A (en) | 1982-12-22 |
Family
ID=14091978
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP56093782A Pending JPS57209296A (en) | 1980-07-25 | 1981-06-19 | Tylosin derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS57209296A (en) |
-
1981
- 1981-06-19 JP JP56093782A patent/JPS57209296A/en active Pending
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