JPS55145689A - Pyrimidoo and imidazoopyridoindole derivative - Google Patents
Pyrimidoo and imidazoopyridoindole derivativeInfo
- Publication number
- JPS55145689A JPS55145689A JP300380A JP300380A JPS55145689A JP S55145689 A JPS55145689 A JP S55145689A JP 300380 A JP300380 A JP 300380A JP 300380 A JP300380 A JP 300380A JP S55145689 A JPS55145689 A JP S55145689A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- pyrimidoo
- imidazoopyridoindole
- derivative
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Psychiatry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7910653A FR2455039A1 (fr) | 1979-04-26 | 1979-04-26 | Pyrimido et imidazo-pyrido-indole-diones et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS55145689A true JPS55145689A (en) | 1980-11-13 |
Family
ID=9224796
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP300380A Pending JPS55145689A (en) | 1979-04-26 | 1980-01-14 | Pyrimidoo and imidazoopyridoindole derivative |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4358451A (enExample) |
| EP (1) | EP0018857B1 (enExample) |
| JP (1) | JPS55145689A (enExample) |
| AT (1) | ATE2253T1 (enExample) |
| AU (1) | AU528634B2 (enExample) |
| CA (1) | CA1129854A (enExample) |
| DE (1) | DE3061648D1 (enExample) |
| DK (1) | DK16980A (enExample) |
| ES (1) | ES487713A1 (enExample) |
| FR (1) | FR2455039A1 (enExample) |
| GR (1) | GR74394B (enExample) |
| IL (1) | IL59128A (enExample) |
| NO (1) | NO794271L (enExample) |
| PT (1) | PT70698A (enExample) |
| ZA (1) | ZA80242B (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005531585A (ja) * | 2002-05-24 | 2005-10-20 | エックス−セプター セラピューティクス, インコーポレイテッド | 薬剤としてのアゼピノインドールおよびピリドインドール誘導体 |
| US8524704B2 (en) | 2002-05-24 | 2013-09-03 | Exelixis, Inc. | Azepinoindole derivatives as pharmaceutical agents |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3246932A1 (de) * | 1982-12-16 | 1984-06-20 | Schering AG, 1000 Berlin und 4709 Bergkamen | Substituierte 5h-pyrimido(5,4-b)indole |
| EP2147679B1 (en) | 2001-07-25 | 2014-06-25 | Raptor Pharmaceutical, Inc. | Compositions for blood-brain barrier transport |
| CA2789262C (en) | 2005-04-28 | 2016-10-04 | Proteus Digital Health, Inc. | Pharma-informatics system |
| FR2901795A1 (fr) * | 2006-05-30 | 2007-12-07 | Fourtillan Snc | Derives de pyrimidino[1',6'-1,2]pyrido[3,4-b]indoles et leur utilisation en therapeutique |
| MX2009002893A (es) | 2006-09-18 | 2009-07-10 | Raptor Pharmaceutical Inc | Tratamiento de trastornos hepaticos mediante la administracion de conjugados de la proteina asociada al receptor (rap). |
| DK2398500T3 (da) | 2009-02-20 | 2019-05-13 | 2 Bbb Medicines B V | Glutathion-baseret lægemiddelafgivelsessystem |
| CA2760945A1 (en) | 2009-05-06 | 2010-11-11 | Laboratory Skin Care, Inc. | Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1076114A (en) * | 1975-02-10 | 1980-04-22 | Mitsubishi Chemical Industries Limited | 1,5-alkylene-3-aryl hydantoin derivatives |
-
1979
- 1979-04-26 FR FR7910653A patent/FR2455039A1/fr active Granted
- 1979-12-27 NO NO794271A patent/NO794271L/no unknown
-
1980
- 1980-01-14 JP JP300380A patent/JPS55145689A/ja active Pending
- 1980-01-15 GR GR60963A patent/GR74394B/el unknown
- 1980-01-15 ZA ZA00800242A patent/ZA80242B/xx unknown
- 1980-01-15 CA CA343,698A patent/CA1129854A/en not_active Expired
- 1980-01-15 US US06/112,238 patent/US4358451A/en not_active Expired - Lifetime
- 1980-01-15 EP EP80400050A patent/EP0018857B1/fr not_active Expired
- 1980-01-15 ES ES487713A patent/ES487713A1/es not_active Expired
- 1980-01-15 AT AT80400050T patent/ATE2253T1/de not_active IP Right Cessation
- 1980-01-15 AU AU54630/80A patent/AU528634B2/en not_active Ceased
- 1980-01-15 DE DE8080400050T patent/DE3061648D1/de not_active Expired
- 1980-01-15 PT PT70698A patent/PT70698A/pt unknown
- 1980-01-15 IL IL59128A patent/IL59128A/xx unknown
- 1980-01-15 DK DK16980A patent/DK16980A/da not_active Application Discontinuation
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005531585A (ja) * | 2002-05-24 | 2005-10-20 | エックス−セプター セラピューティクス, インコーポレイテッド | 薬剤としてのアゼピノインドールおよびピリドインドール誘導体 |
| US8133992B2 (en) | 2002-05-24 | 2012-03-13 | Exelixis, Inc. | Azepinoindole and pyridoindole derivatives as pharmaceutical agents |
| US8524704B2 (en) | 2002-05-24 | 2013-09-03 | Exelixis, Inc. | Azepinoindole derivatives as pharmaceutical agents |
Also Published As
| Publication number | Publication date |
|---|---|
| DE3061648D1 (en) | 1983-02-24 |
| FR2455039B1 (enExample) | 1983-05-13 |
| GR74394B (enExample) | 1984-06-28 |
| ZA80242B (en) | 1980-12-31 |
| IL59128A (en) | 1982-07-30 |
| ES487713A1 (es) | 1980-06-16 |
| EP0018857A1 (fr) | 1980-11-12 |
| PT70698A (fr) | 1980-02-01 |
| NO794271L (no) | 1980-10-28 |
| FR2455039A1 (fr) | 1980-11-21 |
| CA1129854A (en) | 1982-08-17 |
| IL59128A0 (en) | 1980-05-30 |
| DK16980A (da) | 1980-10-27 |
| EP0018857B1 (fr) | 1983-01-19 |
| AU5463080A (en) | 1980-10-30 |
| AU528634B2 (en) | 1983-05-05 |
| US4358451A (en) | 1982-11-09 |
| ATE2253T1 (de) | 1983-02-15 |
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