JPS55145625A - Preparation of alkynyl alcohol - Google Patents
Preparation of alkynyl alcoholInfo
- Publication number
- JPS55145625A JPS55145625A JP5373379A JP5373379A JPS55145625A JP S55145625 A JPS55145625 A JP S55145625A JP 5373379 A JP5373379 A JP 5373379A JP 5373379 A JP5373379 A JP 5373379A JP S55145625 A JPS55145625 A JP S55145625A
- Authority
- JP
- Japan
- Prior art keywords
- aldehyde
- acetylide
- alkynyl alcohol
- preparation
- hight
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PURPOSE: To obtain the title compound, useful as an intermediate for the synthesis of prostaglandin, vitamin E, pheromone, etc., by the reaction of an acetylide with an aldehyde, in the presence of a specific ligand.
CONSTITUTION: An aldehyde, e.g. benzaldehyde, is reacted with an acetylide of formula R'-C≡C-X (R' is H or silyl; X is alkali metal), e.g. lithium trimethylsilyl acetylide, in the presence of asymmetric 2-hydroxymethyl-1-[(1-methylpyrrolidin-2-yl)methyl]pyrrolidine or its salt in a molar amount of about 2W10 times that of the aldehyde, to give an optically active alkynyl alcohol, e.g. 1-phenyl-2- propyn-1-ol.
EFFECT: Hight optical purity of the product.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5373379A JPS55145625A (en) | 1979-05-01 | 1979-05-01 | Preparation of alkynyl alcohol |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5373379A JPS55145625A (en) | 1979-05-01 | 1979-05-01 | Preparation of alkynyl alcohol |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS55145625A true JPS55145625A (en) | 1980-11-13 |
Family
ID=12951023
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP5373379A Pending JPS55145625A (en) | 1979-05-01 | 1979-05-01 | Preparation of alkynyl alcohol |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55145625A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996037457A1 (en) * | 1995-05-25 | 1996-11-28 | Merck & Co., Inc. | Asymmetric synthesis of (-) 6-chloro-4-cyclopropyl-ethynyl-4-trifluoromethyl-1,4-dihydro-2h-3,1-benzoxazin-2-one |
-
1979
- 1979-05-01 JP JP5373379A patent/JPS55145625A/en active Pending
Non-Patent Citations (2)
Title |
---|
CHEMISTRY LETTERS=1978 * |
CHEMISTRY=1978 * |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996037457A1 (en) * | 1995-05-25 | 1996-11-28 | Merck & Co., Inc. | Asymmetric synthesis of (-) 6-chloro-4-cyclopropyl-ethynyl-4-trifluoromethyl-1,4-dihydro-2h-3,1-benzoxazin-2-one |
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