JPS55122716A - - Google Patents

Info

Publication number
JPS55122716A
JPS55122716A JP1086680A JP1086680A JPS55122716A JP S55122716 A JPS55122716 A JP S55122716A JP 1086680 A JP1086680 A JP 1086680A JP 1086680 A JP1086680 A JP 1086680A JP S55122716 A JPS55122716 A JP S55122716A
Authority
JP
Japan
Prior art keywords
carbonic anhydrase
anhydrase inhibitors
intraocular pressure
hosts
normotensive
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1086680A
Other languages
English (en)
Japanese (ja)
Inventor
Eru Sumisu Robaato
Efu Hirushuman Rarufu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of JPS55122716A publication Critical patent/JPS55122716A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP1086680A 1979-02-02 1980-02-02 Pending JPS55122716A (enExample)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US890379A 1979-02-02 1979-02-02

Publications (1)

Publication Number Publication Date
JPS55122716A true JPS55122716A (enExample) 1980-09-20

Family

ID=21734364

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1086680A Pending JPS55122716A (enExample) 1979-02-02 1980-02-02

Country Status (9)

Country Link
EP (1) EP0014642B1 (enExample)
JP (1) JPS55122716A (enExample)
AT (1) ATE6738T1 (enExample)
AU (1) AU536438B2 (enExample)
DE (1) DE3067081D1 (enExample)
DK (1) DK43280A (enExample)
FI (1) FI800205A7 (enExample)
IE (1) IE49507B1 (enExample)
NZ (1) NZ192673A (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018500331A (ja) * 2014-12-19 2018-01-11 ドン−ア エスティ カンパニー リミテッド 茯苓皮抽出物を含有する退行性神経疾患の予防、改善または治療用組成物

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE50901B1 (en) * 1980-03-04 1986-08-06 Merck & Co Inc Ophthalmic compositions of carbonic anhydrase inhibitors for topical application in the treatment of elevated intraocular pressure
GB8822285D0 (en) * 1988-09-22 1988-10-26 Ddsa Pharmaceuticals Ltd Opthalmic preparations
EP1507513A1 (de) * 2002-05-24 2005-02-23 Dr. GERHARD MANN chem.-pharm. Fabrik GmbH Tropfbares ophthalmisches gelpräparat mit diclofenamid und timolol
EP2847175A4 (en) * 2012-05-08 2016-04-20 Cellix Bio Private Ltd COMPOSITIONS AND METHODS INHIBITING THE ACTIVITY OF CARBONIC ANHYDRASE

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB860371A (en) * 1958-07-03 1961-02-01 Pfizer & Co C Di-sulfonamides and compositions containing them
NL7508856A (nl) * 1974-08-16 1976-02-18 Merck & Co Inc Werkwijze voor het bereiden van preparaten tegen hypertensie.
NZ182022A (en) * 1975-09-26 1978-12-18 Merck & Co Inc Antiglaucoma compositions comprising 1-t butylamino-3-(4-morpholino-1,2,5-thiadiazol-3-yloxy)-2-prodanol hydogen maleate
US4077407A (en) * 1975-11-24 1978-03-07 Alza Corporation Osmotic devices having composite walls

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018500331A (ja) * 2014-12-19 2018-01-11 ドン−ア エスティ カンパニー リミテッド 茯苓皮抽出物を含有する退行性神経疾患の予防、改善または治療用組成物

Also Published As

Publication number Publication date
IE800207L (en) 1980-08-02
DK43280A (da) 1980-08-03
EP0014642A2 (en) 1980-08-20
ATE6738T1 (de) 1984-04-15
AU5487980A (en) 1980-08-07
AU536438B2 (en) 1984-05-10
IE49507B1 (en) 1985-10-16
NZ192673A (en) 1984-07-06
EP0014642A3 (en) 1981-01-07
EP0014642B1 (en) 1984-03-21
DE3067081D1 (en) 1984-04-26
FI800205A7 (fi) 1981-01-01

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