JPS5495592A - Cephalosporin derivative and manufacture - Google Patents

Cephalosporin derivative and manufacture

Info

Publication number
JPS5495592A
JPS5495592A JP15817278A JP15817278A JPS5495592A JP S5495592 A JPS5495592 A JP S5495592A JP 15817278 A JP15817278 A JP 15817278A JP 15817278 A JP15817278 A JP 15817278A JP S5495592 A JPS5495592 A JP S5495592A
Authority
JP
Japan
Prior art keywords
manufacture
cephalosporin derivative
cephalosporin
derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP15817278A
Other languages
English (en)
Other versions
JPH0132226B2 (ja
Inventor
Burumubatsuha Yurugen
Deyurutsukuhaimaa Warutaa
Shiyurinaa Erumaa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of JPS5495592A publication Critical patent/JPS5495592A/ja
Publication of JPH0132226B2 publication Critical patent/JPH0132226B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP15817278A 1977-12-24 1978-12-23 Cephalosporin derivative and manufacture Granted JPS5495592A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772758001 DE2758001A1 (de) 1977-12-24 1977-12-24 Cephalosporinderivate und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
JPS5495592A true JPS5495592A (en) 1979-07-28
JPH0132226B2 JPH0132226B2 (ja) 1989-06-29

Family

ID=6027279

Family Applications (1)

Application Number Title Priority Date Filing Date
JP15817278A Granted JPS5495592A (en) 1977-12-24 1978-12-23 Cephalosporin derivative and manufacture

Country Status (20)

Country Link
US (1) US4293550A (ja)
EP (1) EP0002765B1 (ja)
JP (1) JPS5495592A (ja)
AT (1) AT365599B (ja)
AU (1) AU534258B2 (ja)
CA (1) CA1109461A (ja)
DE (2) DE2758001A1 (ja)
DK (1) DK578978A (ja)
EG (1) EG13762A (ja)
ES (1) ES476109A1 (ja)
FI (1) FI66007C (ja)
GR (1) GR65234B (ja)
HU (1) HU184140B (ja)
IE (1) IE48147B1 (ja)
IL (1) IL56284A (ja)
NO (1) NO784366L (ja)
NZ (1) NZ189266A (ja)
PH (1) PH15925A (ja)
PT (1) PT68964A (ja)
ZA (1) ZA787209B (ja)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5547688A (en) * 1978-09-08 1980-04-04 Fujisawa Pharmaceut Co Ltd Novel cephem compound and its preparation
JPS5657790A (en) * 1979-10-02 1981-05-20 Glaxo Group Ltd Cephalosporin antibiotic
JPS56142289A (en) * 1980-02-23 1981-11-06 Hoechst Ag Cephalosporin derivative and manufacture
JPS57131794A (en) * 1980-12-31 1982-08-14 Fujisawa Pharmaceut Co Ltd Novel cephem compound or salt thereof, preparation of the same and preventing agent and remedy for microbism containing the same as active constituent

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4409214A (en) * 1979-11-19 1983-10-11 Fujisawa Pharmaceutical, Co., Ltd. 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
EP0055465B1 (en) 1980-12-31 1989-08-23 Fujisawa Pharmaceutical Co., Ltd. 7-acylaminocephalosporanic acid derivatives and processes for the preparation thereof
US4427677A (en) * 1980-12-31 1984-01-24 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4618606A (en) * 1982-11-17 1986-10-21 Toyama Chemical Co., Ltd. Antibiotic 7-(thiazolyl)-3-(pyrazinylmethyl) or (pyridazinylmethyl) cephalosporins
EP1059293A1 (en) * 1995-10-12 2000-12-13 Microcide Pharmaceuticals, Inc. Novel amino chlorothiazole compounds
IT1295935B1 (it) * 1997-10-30 1999-05-28 Acs Dobfar Spa Derivati aminotiazolici utili nella preparazione di antibiotici b -lattamici
TWI335332B (en) * 2001-10-12 2011-01-01 Theravance Inc Cross-linked vancomycin-cephalosporin antibiotics
CN102015591B (zh) 2008-03-04 2014-01-29 艾尼纳制药公司 制备与5-ht2c激动剂(r)-8-氯-1-甲基-2，3，4，5-四氢-1h-3-苯并氮杂卓相关的中间体的方法
WO2011153206A1 (en) 2010-06-02 2011-12-08 Arena Pharmaceuticals, Inc. Processes for the preparation of 5-ht2c receptor agonists
KR20140091458A (ko) 2010-09-01 2014-07-21 아레나 파마슈티칼스, 인크. 신장 손상을 갖는 개체에 대한 로카세린의 투여
CN103189359A (zh) 2010-09-01 2013-07-03 艾尼纳制药公司 5-ht2c激动剂的光学活性酸盐
AU2011296003B2 (en) 2010-09-01 2015-11-12 Arena Pharmaceuticals, Inc. Modified-release dosage forms of 5-HT2C agonist useful for weight management
KR20130101524A (ko) 2010-09-01 2013-09-13 아레나 파마슈티칼스, 인크. 5-ｈｔ2ｃ 아고니스트의 비-흡습성 염
CA2886875A1 (en) 2012-10-09 2014-04-17 Arena Pharmaceuticals, Inc. Method of weight management

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51149296A (en) * 1975-06-09 1976-12-22 Takeda Chem Ind Ltd Cephems or penams and their preparation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5168589A (ja) * 1974-12-06 1976-06-14 Shionogi Seiyaku Kk
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
DE2760123C2 (de) * 1976-01-23 1986-04-30 Roussel-Uclaf, Paris 7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporansäuren, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51149296A (en) * 1975-06-09 1976-12-22 Takeda Chem Ind Ltd Cephems or penams and their preparation

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5547688A (en) * 1978-09-08 1980-04-04 Fujisawa Pharmaceut Co Ltd Novel cephem compound and its preparation
JPH0121154B2 (ja) * 1978-09-08 1989-04-19 Fujisawa Pharmaceutical Co
JPS5657790A (en) * 1979-10-02 1981-05-20 Glaxo Group Ltd Cephalosporin antibiotic
JPS56142289A (en) * 1980-02-23 1981-11-06 Hoechst Ag Cephalosporin derivative and manufacture
JPS57131794A (en) * 1980-12-31 1982-08-14 Fujisawa Pharmaceut Co Ltd Novel cephem compound or salt thereof, preparation of the same and preventing agent and remedy for microbism containing the same as active constituent

Also Published As

Publication number Publication date
ZA787209B (en) 1979-12-27
IL56284A (en) 1983-03-31
AU4284878A (en) 1979-06-28
DK578978A (da) 1979-06-25
PH15925A (en) 1983-04-26
FI66007C (fi) 1984-08-10
GR65234B (en) 1980-07-30
IE782546L (en) 1979-06-24
CA1109461A (en) 1981-09-22
IL56284A0 (en) 1979-03-12
NO784366L (no) 1979-06-26
AU534258B2 (en) 1984-01-12
JPH0132226B2 (ja) 1989-06-29
AT365599B (de) 1982-01-25
US4293550A (en) 1981-10-06
PT68964A (de) 1979-01-01
EG13762A (en) 1982-09-30
EP0002765B1 (de) 1981-09-02
DE2861043D1 (en) 1981-11-26
FI783960A (fi) 1979-06-25
FI66007B (fi) 1984-04-30
DE2758001A1 (de) 1979-07-12
IE48147B1 (en) 1984-10-17
EP0002765A1 (de) 1979-07-11
ATA924178A (de) 1981-06-15
HU184140B (en) 1984-07-30
ES476109A1 (es) 1979-10-16
NZ189266A (en) 1981-12-15

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