JPS5283397A - 1*44benzoxazine and 1*44benzothiazine cyclic derivatives process for preparing same and medical composition having antiidepression activity containing same - Google Patents

1*44benzoxazine and 1*44benzothiazine cyclic derivatives process for preparing same and medical composition having antiidepression activity containing same

Info

Publication number
JPS5283397A
JPS5283397A JP16078076A JP16078076A JPS5283397A JP S5283397 A JPS5283397 A JP S5283397A JP 16078076 A JP16078076 A JP 16078076A JP 16078076 A JP16078076 A JP 16078076A JP S5283397 A JPS5283397 A JP S5283397A
Authority
JP
Japan
Prior art keywords
same
antiidepression
medical composition
cyclic derivatives
activity containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP16078076A
Other languages
English (en)
Japanese (ja)
Inventor
Meroni Piero
Mongeri Nikora
Rauriia Furanchiesuko
Rotsushi Aretsusandoro
Tomashiini Rafuaere
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Carlo Erba SpA filed Critical Carlo Erba SpA
Publication of JPS5283397A publication Critical patent/JPS5283397A/ja
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/36Oxygen or sulfur atoms
    • C07D207/402,5-Pyrrolidine-diones
    • C07D207/4042,5-Pyrrolidine-diones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms, e.g. succinimide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/27Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups
    • C07C205/35Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/36Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/37Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/341,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/361,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP16078076A 1975-12-30 1976-12-28 1*44benzoxazine and 1*44benzothiazine cyclic derivatives process for preparing same and medical composition having antiidepression activity containing same Pending JPS5283397A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT30829/75A IT1052009B (it) 1975-12-30 1975-12-30 Imidazo 4.3 c 1.4 benzossazino imidazo 4.3 c 1.4 benzotiazino pirazo 2.1 c 1.4 benzossazino e pirazo 2.1 c 1.4 benzotiazino derivati

Publications (1)

Publication Number Publication Date
JPS5283397A true JPS5283397A (en) 1977-07-12

Family

ID=11232353

Family Applications (1)

Application Number Title Priority Date Filing Date
JP16078076A Pending JPS5283397A (en) 1975-12-30 1976-12-28 1*44benzoxazine and 1*44benzothiazine cyclic derivatives process for preparing same and medical composition having antiidepression activity containing same

Country Status (22)

Country Link
US (1) US4134974A (US07494231-20090224-C00006.png)
JP (1) JPS5283397A (US07494231-20090224-C00006.png)
AT (1) AT351041B (US07494231-20090224-C00006.png)
AU (1) AU504565B2 (US07494231-20090224-C00006.png)
BE (1) BE849919A (US07494231-20090224-C00006.png)
CA (1) CA1099267A (US07494231-20090224-C00006.png)
CH (1) CH630383A5 (US07494231-20090224-C00006.png)
CS (1) CS197301B2 (US07494231-20090224-C00006.png)
DE (1) DE2658806A1 (US07494231-20090224-C00006.png)
DK (1) DK587476A (US07494231-20090224-C00006.png)
FI (1) FI61902C (US07494231-20090224-C00006.png)
FR (1) FR2336929A1 (US07494231-20090224-C00006.png)
GB (1) GB1533020A (US07494231-20090224-C00006.png)
HU (1) HU176510B (US07494231-20090224-C00006.png)
IL (1) IL51091A (US07494231-20090224-C00006.png)
IT (1) IT1052009B (US07494231-20090224-C00006.png)
NL (1) NL7614445A (US07494231-20090224-C00006.png)
NO (1) NO150882C (US07494231-20090224-C00006.png)
NZ (1) NZ182952A (US07494231-20090224-C00006.png)
SE (1) SE7613778L (US07494231-20090224-C00006.png)
SU (1) SU812181A3 (US07494231-20090224-C00006.png)
ZA (1) ZA767588B (US07494231-20090224-C00006.png)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996023789A1 (fr) * 1995-02-03 1996-08-08 Sankyo Company, Limited Derives d'hexahydropyrazinoquinoline

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4049422A (en) * 1976-03-29 1977-09-20 United States Borax & Chemical Corporation Herbicidal morpholinobenzimidazoles
SE444319B (sv) * 1977-11-18 1986-04-07 Roussel Uclaf Nya imidazobensoxazinderivat, forfarande for framstellning derav och farmaceutiska kompositioner innehallande dessa foreningar
US4254121A (en) * 1979-08-13 1981-03-03 Ayerst, Mckenna & Harrison Inc. 3-Oxo-5H-pyrimido[2,1-c][1,4 ]benzoxazines
US4254118A (en) * 1979-08-13 1981-03-03 Ayerst, Mckenna & Harrison Inc. 1-Oxo-5H-pyrimido[2,1-c][1,4]benzthiazine-2-carboxylic acid esters
US5089493A (en) * 1988-02-05 1992-02-18 Riker Laboratories, Inc. Triazolo[1,5-C]pyrimido[1,4]azines as bronchodilators
US5166343A (en) * 1988-02-05 1992-11-24 Riker Laboratories, Inc. Triazolo[1,5-c]pyrimido[1,4]-azines as bronchodilators
ES2177539T3 (es) * 1992-02-13 2002-12-16 Upjohn Co Benzoxacinas 4-oxo- y 4h-imidazo(5,1-c)(1,4) utilez como agentes de union de receptores de benzodiacepina.
GB9212486D0 (en) * 1992-06-12 1992-07-22 Erba Carlo Spa Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation
US5512566A (en) * 1993-10-25 1996-04-30 Ortho Pharmaceutical Corporation Tricyclic compounds having affinity for the 5-HT1A receptor
GB9410469D0 (en) * 1994-05-25 1994-07-13 Erba Farmitalia Imidazolylalkyl derivatives of imidazo (5,1-c) (1,4) benzoxazin-1-one and process for their preparation
WO2007087250A2 (en) 2006-01-23 2007-08-02 Amira Pharmaceuticals, Inc. Tricyclic inhibitors of 5-lipoxygenase
WO2014089904A1 (en) 2012-12-10 2014-06-19 Abbvie Inc. Triazinone compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3929783A (en) * 1974-12-06 1975-12-30 Squibb & Sons Inc 1-Substituted-4-phenyl-4H-{8 1,2,4{9 triazolo{8 3,4-C{9 {8 1,4{9 {0 benzothiazines or benzoxazines
US4035495A (en) * 1975-02-10 1977-07-12 Ayerst Mckenna And Harrison Ltd. Pyrrolobenzoxazines, pyrrolobenzothiazines and process therefor

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996023789A1 (fr) * 1995-02-03 1996-08-08 Sankyo Company, Limited Derives d'hexahydropyrazinoquinoline

Also Published As

Publication number Publication date
CH630383A5 (de) 1982-06-15
HU176510B (en) 1981-03-28
AU2086376A (en) 1978-06-29
NO764395L (US07494231-20090224-C00006.png) 1977-07-01
US4134974A (en) 1979-01-16
FI763752A (US07494231-20090224-C00006.png) 1977-07-01
BE849919A (fr) 1977-04-15
IT1052009B (it) 1981-06-20
IL51091A0 (en) 1977-02-28
ATA985776A (de) 1978-12-15
FI61902B (fi) 1982-06-30
FR2336929B1 (US07494231-20090224-C00006.png) 1980-04-18
CS197301B2 (en) 1980-04-30
SE7613778L (sv) 1977-07-01
DE2658806A1 (de) 1977-07-14
IL51091A (en) 1984-01-31
FI61902C (fi) 1982-10-11
DK587476A (da) 1977-07-01
CA1099267A (en) 1981-04-14
NO150882B (no) 1984-09-24
AU504565B2 (en) 1979-10-18
GB1533020A (en) 1978-11-22
NZ182952A (en) 1980-05-08
AT351041B (de) 1979-07-10
NO150882C (no) 1985-01-09
SU812181A3 (ru) 1981-03-07
FR2336929A1 (fr) 1977-07-29
ZA767588B (en) 1977-11-30
NL7614445A (nl) 1977-07-04

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