BE849919A - Derives cycliques de la 1,4-benzoxazine et de la 1,4-benzothiazine et procede pour les preparer - Google Patents

Derives cycliques de la 1,4-benzoxazine et de la 1,4-benzothiazine et procede pour les preparer

Info

Publication number
BE849919A
BE849919A BE173691A BE173691A BE849919A BE 849919 A BE849919 A BE 849919A BE 173691 A BE173691 A BE 173691A BE 173691 A BE173691 A BE 173691A BE 849919 A BE849919 A BE 849919A
Authority
BE
Belgium
Prior art keywords
benzothiazine
benzoxazine
preparing
cyclic derivatives
cyclic
Prior art date
Application number
BE173691A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE849919A publication Critical patent/BE849919A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/36—Oxygen or sulfur atoms
    • C07D207/40—2,5-Pyrrolidine-diones
    • C07D207/404—2,5-Pyrrolidine-diones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms, e.g. succinimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/27—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups
    • C07C205/35—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/36—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/37—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
BE173691A 1975-12-30 1976-12-28 Derives cycliques de la 1,4-benzoxazine et de la 1,4-benzothiazine et procede pour les preparer BE849919A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT30829/75A IT1052009B (it) 1975-12-30 1975-12-30 Imidazo 4.3 c 1.4 benzossazino imidazo 4.3 c 1.4 benzotiazino pirazo 2.1 c 1.4 benzossazino e pirazo 2.1 c 1.4 benzotiazino derivati

Publications (1)

Publication Number Publication Date
BE849919A true BE849919A (fr) 1977-04-15

Family

ID=11232353

Family Applications (1)

Application Number Title Priority Date Filing Date
BE173691A BE849919A (fr) 1975-12-30 1976-12-28 Derives cycliques de la 1,4-benzoxazine et de la 1,4-benzothiazine et procede pour les preparer

Country Status (22)

Country Link
US (1) US4134974A (fr)
JP (1) JPS5283397A (fr)
AT (1) AT351041B (fr)
AU (1) AU504565B2 (fr)
BE (1) BE849919A (fr)
CA (1) CA1099267A (fr)
CH (1) CH630383A5 (fr)
CS (1) CS197301B2 (fr)
DE (1) DE2658806A1 (fr)
DK (1) DK587476A (fr)
FI (1) FI61902C (fr)
FR (1) FR2336929A1 (fr)
GB (1) GB1533020A (fr)
HU (1) HU176510B (fr)
IL (1) IL51091A (fr)
IT (1) IT1052009B (fr)
NL (1) NL7614445A (fr)
NO (1) NO150882C (fr)
NZ (1) NZ182952A (fr)
SE (1) SE7613778L (fr)
SU (1) SU812181A3 (fr)
ZA (1) ZA767588B (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5364854A (en) * 1992-06-12 1994-11-15 Farmitalia Carlo Erba S.R.L. Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation
WO1995011903A1 (fr) * 1993-10-25 1995-05-04 Ortho Pharmaceutical Corporation Composes tricycliques ayant une affinite pour le recepteur de 5-ht1a

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4049422A (en) * 1976-03-29 1977-09-20 United States Borax & Chemical Corporation Herbicidal morpholinobenzimidazoles
SE444319B (sv) * 1977-11-18 1986-04-07 Roussel Uclaf Nya imidazobensoxazinderivat, forfarande for framstellning derav och farmaceutiska kompositioner innehallande dessa foreningar
US4254121A (en) * 1979-08-13 1981-03-03 Ayerst, Mckenna & Harrison Inc. 3-Oxo-5H-pyrimido[2,1-c][1,4 ]benzoxazines
US4254118A (en) * 1979-08-13 1981-03-03 Ayerst, Mckenna & Harrison Inc. 1-Oxo-5H-pyrimido[2,1-c][1,4]benzthiazine-2-carboxylic acid esters
US5166343A (en) * 1988-02-05 1992-11-24 Riker Laboratories, Inc. Triazolo[1,5-c]pyrimido[1,4]-azines as bronchodilators
US5089493A (en) * 1988-02-05 1992-02-18 Riker Laboratories, Inc. Triazolo[1,5-C]pyrimido[1,4]azines as bronchodilators
WO1993016082A1 (fr) * 1992-02-13 1993-08-19 The Upjohn Company Benzoxazines 4-oxo et 4h-imidazo(5,1-c)(1,4) utiles comme agents de liaison de recepteurs de benzodiazepine
GB9410469D0 (en) * 1994-05-25 1994-07-13 Erba Farmitalia Imidazolylalkyl derivatives of imidazo (5,1-c) (1,4) benzoxazin-1-one and process for their preparation
WO1996023789A1 (fr) * 1995-02-03 1996-08-08 Sankyo Company, Limited Derives d'hexahydropyrazinoquinoline
CA2636043A1 (fr) * 2006-01-23 2007-08-02 Amira Pharmaceuticals, Inc. Inhibiteurs tricycliques de la 5-lipoxygenase
WO2014089904A1 (fr) 2012-12-10 2014-06-19 Abbvie Inc. Composés triazinones

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3929783A (en) * 1974-12-06 1975-12-30 Squibb & Sons Inc 1-Substituted-4-phenyl-4H-{8 1,2,4{9 triazolo{8 3,4-C{9 {8 1,4{9 {0 benzothiazines or benzoxazines
US4035495A (en) * 1975-02-10 1977-07-12 Ayerst Mckenna And Harrison Ltd. Pyrrolobenzoxazines, pyrrolobenzothiazines and process therefor

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5364854A (en) * 1992-06-12 1994-11-15 Farmitalia Carlo Erba S.R.L. Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation
WO1995011903A1 (fr) * 1993-10-25 1995-05-04 Ortho Pharmaceutical Corporation Composes tricycliques ayant une affinite pour le recepteur de 5-ht1a

Also Published As

Publication number Publication date
DE2658806A1 (de) 1977-07-14
NO764395L (fr) 1977-07-01
DK587476A (da) 1977-07-01
NL7614445A (nl) 1977-07-04
FR2336929B1 (fr) 1980-04-18
ATA985776A (de) 1978-12-15
IT1052009B (it) 1981-06-20
CH630383A5 (de) 1982-06-15
NO150882B (no) 1984-09-24
FI61902C (fi) 1982-10-11
HU176510B (en) 1981-03-28
AU2086376A (en) 1978-06-29
JPS5283397A (en) 1977-07-12
IL51091A0 (en) 1977-02-28
FR2336929A1 (fr) 1977-07-29
SU812181A3 (ru) 1981-03-07
US4134974A (en) 1979-01-16
CS197301B2 (en) 1980-04-30
SE7613778L (sv) 1977-07-01
ZA767588B (en) 1977-11-30
NZ182952A (en) 1980-05-08
AT351041B (de) 1979-07-10
AU504565B2 (en) 1979-10-18
IL51091A (en) 1984-01-31
GB1533020A (en) 1978-11-22
FI763752A (fr) 1977-07-01
CA1099267A (fr) 1981-04-14
NO150882C (no) 1985-01-09
FI61902B (fi) 1982-06-30

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: CARLO ERBA S.P.A.

Effective date: 19901231