JPH10500699A - 内部寄生生物を防除するための昆虫のニコチン性アセチルコリン受容体のアゴニスト及びアンタゴニスト - Google Patents
内部寄生生物を防除するための昆虫のニコチン性アセチルコリン受容体のアゴニスト及びアンタゴニストInfo
- Publication number
- JPH10500699A JPH10500699A JP8500297A JP50029796A JPH10500699A JP H10500699 A JPH10500699 A JP H10500699A JP 8500297 A JP8500297 A JP 8500297A JP 50029796 A JP50029796 A JP 50029796A JP H10500699 A JPH10500699 A JP H10500699A
- Authority
- JP
- Japan
- Prior art keywords
- group
- antagonists
- nicotinic acetylcholine
- active compound
- agonists
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Abstract
Description
Claims (1)
- 【特許請求の範囲】 1.内部寄生生物を防除するための昆虫のニコチン性アセチルコリン受容体のア ゴニスト及びアンタゴニストの使用。 2.少なくとも1つのニコチン性アセチルコリン受容体のアゴニスト及びアンタ ゴニストを含んでなる殺内部寄生生物組成物。 3.増量剤及び/または界面活性剤と混合することを特徴とする、殺内部寄生生 物組成物の製造方法。 4.殺内部寄生生物組成物を製造するための殺内部寄生生物組成物の使用。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4419814A DE4419814A1 (de) | 1994-06-07 | 1994-06-07 | Endoparasitizide |
DE4419814.0 | 1994-06-07 | ||
PCT/EP1995/002014 WO1995033453A1 (de) | 1994-06-07 | 1995-05-26 | Agonisten und antagonisten der nicotinergen acetylcholinrezeptoren von insekten als endoparasitizide |
Publications (2)
Publication Number | Publication Date |
---|---|
JPH10500699A true JPH10500699A (ja) | 1998-01-20 |
JP3978227B2 JP3978227B2 (ja) | 2007-09-19 |
Family
ID=6519954
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP50029796A Expired - Lifetime JP3978227B2 (ja) | 1994-06-07 | 1995-05-26 | 内部寄生生物を防除するための昆虫のニコチン性アセチルコリン受容体のアゴニスト及びアンタゴニスト |
Country Status (15)
Country | Link |
---|---|
US (1) | US5712295A (ja) |
EP (1) | EP0764022B1 (ja) |
JP (1) | JP3978227B2 (ja) |
KR (1) | KR100372348B1 (ja) |
CN (1) | CN1100537C (ja) |
AT (1) | ATE348604T1 (ja) |
AU (1) | AU704092B2 (ja) |
BR (1) | BR9507926A (ja) |
CA (1) | CA2192093C (ja) |
DE (2) | DE4419814A1 (ja) |
DK (1) | DK0764022T3 (ja) |
ES (1) | ES2279513T3 (ja) |
MX (1) | MX9606179A (ja) |
WO (1) | WO1995033453A1 (ja) |
ZA (1) | ZA954643B (ja) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2002503682A (ja) * | 1998-02-23 | 2002-02-05 | バイエル・アクチエンゲゼルシヤフト | 人間への寄生昆虫及び寄生ダニ類を防除するための水性薬剤 |
JP2012504636A (ja) * | 2008-10-03 | 2012-02-23 | バイエル ビー. ブイ. | 血を吸うおよび血を消費する寄生生物の、殺寄生生物剤の経口投与による全身処置 |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4443888A1 (de) * | 1994-12-09 | 1996-06-13 | Bayer Ag | Dermal applizierbare Formulierungen von Parasitiziden |
US6426333B1 (en) * | 1996-09-19 | 2002-07-30 | Merial | Spot-on formulations for combating parasites |
DE19654079A1 (de) * | 1996-12-23 | 1998-06-25 | Bayer Ag | Endo-ekto-parasitizide Mittel |
FR2761232B1 (fr) * | 1997-03-26 | 2000-03-10 | Rhone Merieux | Procede et moyens d'eradication des puces dans les locaux habites par les petits mammiferes |
DE19734665A1 (de) * | 1997-08-11 | 1999-02-18 | Bayer Ag | Mittel gegen holzzerstörende Insekten |
US6727228B2 (en) * | 2001-04-25 | 2004-04-27 | Johnson & Johnson Consumer Companies, Inc. | Pediculicidal and ovacidal treatment compositions and methods for killing head lice and their eggs |
EP1969940A3 (en) * | 2004-12-17 | 2008-12-10 | Devgen NV | Nematicidal compositions |
US8110608B2 (en) | 2008-06-05 | 2012-02-07 | Ecolab Usa Inc. | Solid form sodium lauryl sulfate (SLS) pesticide composition |
US8968757B2 (en) * | 2010-10-12 | 2015-03-03 | Ecolab Usa Inc. | Highly wettable, water dispersible, granules including two pesticides |
CA2989391C (en) | 2014-06-24 | 2023-03-14 | John O'halloran | Fish feed compositions containing a neonicotinoid for preventing and treating parasite infections |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA689474A (en) * | 1964-06-23 | Clarence H. Gleason | Nicotine pamoate | |
JPS60172976A (ja) * | 1984-02-16 | 1985-09-06 | Nippon Tokushu Noyaku Seizo Kk | ニトロメチレン誘導体,その製法及び殺虫,殺ダニ,殺センチユウ剤 |
ZW5085A1 (en) * | 1984-04-13 | 1985-09-18 | Nihon Tokushu Noyaku Seizo Kk | Nitromethylene derivatives,intermediates thereof,processes for production thereof,and insecticides |
ATE67493T1 (de) * | 1985-02-04 | 1991-10-15 | Bayer Agrochem Kk | Heterocyclische verbindungen. |
JPH07121909B2 (ja) * | 1986-09-10 | 1995-12-25 | 日本バイエルアグロケム株式会社 | 新規複素環式化合物及び殺虫剤 |
JP3023794B2 (ja) * | 1989-05-17 | 2000-03-21 | 日本バイエルアグロケム株式会社 | 殺虫性ニトロ置換ヘテロ環式化合物 |
DE4232561A1 (de) * | 1992-09-29 | 1994-03-31 | Bayer Ag | Bekämpfung von Fischparasiten |
-
1994
- 1994-06-07 DE DE4419814A patent/DE4419814A1/de not_active Withdrawn
-
1995
- 1995-05-26 AT AT95922486T patent/ATE348604T1/de not_active IP Right Cessation
- 1995-05-26 JP JP50029796A patent/JP3978227B2/ja not_active Expired - Lifetime
- 1995-05-26 DE DE59511073T patent/DE59511073D1/de not_active Expired - Fee Related
- 1995-05-26 DK DK95922486T patent/DK0764022T3/da active
- 1995-05-26 CA CA002192093A patent/CA2192093C/en not_active Expired - Fee Related
- 1995-05-26 KR KR1019960706908A patent/KR100372348B1/ko not_active IP Right Cessation
- 1995-05-26 CN CN95193465A patent/CN1100537C/zh not_active Expired - Fee Related
- 1995-05-26 MX MX9606179A patent/MX9606179A/es not_active IP Right Cessation
- 1995-05-26 ES ES95922486T patent/ES2279513T3/es not_active Expired - Lifetime
- 1995-05-26 BR BR9507926A patent/BR9507926A/pt not_active Application Discontinuation
- 1995-05-26 EP EP95922486A patent/EP0764022B1/de not_active Expired - Lifetime
- 1995-05-26 WO PCT/EP1995/002014 patent/WO1995033453A1/de active IP Right Grant
- 1995-05-26 AU AU27364/95A patent/AU704092B2/en not_active Ceased
- 1995-05-26 US US08/750,012 patent/US5712295A/en not_active Expired - Lifetime
- 1995-06-06 ZA ZA954643A patent/ZA954643B/xx unknown
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2002503682A (ja) * | 1998-02-23 | 2002-02-05 | バイエル・アクチエンゲゼルシヤフト | 人間への寄生昆虫及び寄生ダニ類を防除するための水性薬剤 |
JP2012504636A (ja) * | 2008-10-03 | 2012-02-23 | バイエル ビー. ブイ. | 血を吸うおよび血を消費する寄生生物の、殺寄生生物剤の経口投与による全身処置 |
JP2016179983A (ja) * | 2008-10-03 | 2016-10-13 | バイエル ビー. ブイ. | 血を吸うおよび血を消費する寄生生物の、殺寄生生物剤の経口投与による全身処置 |
US9820977B2 (en) | 2008-10-03 | 2017-11-21 | Bayer Healthcare Llc | Systemic treatment of blood-sucking and blood-consuming parasites by oral administration of a parasiticidal agent |
Also Published As
Publication number | Publication date |
---|---|
ATE348604T1 (de) | 2007-01-15 |
ES2279513T3 (es) | 2007-08-16 |
DE4419814A1 (de) | 1995-12-14 |
US5712295A (en) | 1998-01-27 |
CA2192093C (en) | 2007-05-22 |
AU2736495A (en) | 1996-01-04 |
EP0764022B1 (de) | 2006-12-20 |
DK0764022T3 (da) | 2007-04-10 |
CN1149827A (zh) | 1997-05-14 |
DE59511073D1 (de) | 2007-02-01 |
ZA954643B (en) | 1996-01-26 |
WO1995033453A1 (de) | 1995-12-14 |
CN1100537C (zh) | 2003-02-05 |
MX9606179A (es) | 1998-01-31 |
JP3978227B2 (ja) | 2007-09-19 |
EP0764022A1 (de) | 1997-03-26 |
AU704092B2 (en) | 1999-04-15 |
BR9507926A (pt) | 1997-11-11 |
CA2192093A1 (en) | 1995-12-14 |
KR100372348B1 (ko) | 2003-05-12 |
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