MX9606179A - Agonistas y antagonistas de los receptores del acido acetilcolina nicotinico de insectos para el control de endoparasitos. - Google Patents

Agonistas y antagonistas de los receptores del acido acetilcolina nicotinico de insectos para el control de endoparasitos.

Info

Publication number
MX9606179A
MX9606179A MX9606179A MX9606179A MX9606179A MX 9606179 A MX9606179 A MX 9606179A MX 9606179 A MX9606179 A MX 9606179A MX 9606179 A MX9606179 A MX 9606179A MX 9606179 A MX9606179 A MX 9606179A
Authority
MX
Mexico
Prior art keywords
insects
agonists
antagonists
nicotinic acetylcholine
acetylcholine receptors
Prior art date
Application number
MX9606179A
Other languages
English (en)
Other versions
MXPA96006179A (es
Inventor
Norbert Mencke
Achim Harder
Terence Hopkins
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MXPA96006179A publication Critical patent/MXPA96006179A/es
Publication of MX9606179A publication Critical patent/MX9606179A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)

Abstract

Empleo de agonistas y antagonistas de los receptores nicotinérgicos de la acetilcolina de los insectos para la lucha contra los endoparásitos.
MX9606179A 1994-06-07 1995-05-26 Agonistas y antagonistas de los receptores del acido acetilcolina nicotinico de insectos para el control de endoparasitos. MX9606179A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE4419814A DE4419814A1 (de) 1994-06-07 1994-06-07 Endoparasitizide
DEP4419814.0 1994-06-07
PCT/EP1995/002014 WO1995033453A1 (de) 1994-06-07 1995-05-26 Agonisten und antagonisten der nicotinergen acetylcholinrezeptoren von insekten als endoparasitizide

Publications (2)

Publication Number Publication Date
MXPA96006179A MXPA96006179A (es) 1998-01-01
MX9606179A true MX9606179A (es) 1998-01-31

Family

ID=6519954

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9606179A MX9606179A (es) 1994-06-07 1995-05-26 Agonistas y antagonistas de los receptores del acido acetilcolina nicotinico de insectos para el control de endoparasitos.

Country Status (15)

Country Link
US (1) US5712295A (es)
EP (1) EP0764022B1 (es)
JP (1) JP3978227B2 (es)
KR (1) KR100372348B1 (es)
CN (1) CN1100537C (es)
AT (1) ATE348604T1 (es)
AU (1) AU704092B2 (es)
BR (1) BR9507926A (es)
CA (1) CA2192093C (es)
DE (2) DE4419814A1 (es)
DK (1) DK0764022T3 (es)
ES (1) ES2279513T3 (es)
MX (1) MX9606179A (es)
WO (1) WO1995033453A1 (es)
ZA (1) ZA954643B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4443888A1 (de) * 1994-12-09 1996-06-13 Bayer Ag Dermal applizierbare Formulierungen von Parasitiziden
US6426333B1 (en) * 1996-09-19 2002-07-30 Merial Spot-on formulations for combating parasites
DE19654079A1 (de) * 1996-12-23 1998-06-25 Bayer Ag Endo-ekto-parasitizide Mittel
FR2761232B1 (fr) * 1997-03-26 2000-03-10 Rhone Merieux Procede et moyens d'eradication des puces dans les locaux habites par les petits mammiferes
DE19734665A1 (de) * 1997-08-11 1999-02-18 Bayer Ag Mittel gegen holzzerstörende Insekten
DE19807630A1 (de) * 1998-02-23 1999-08-26 Bayer Ag Wasserhaltige Mittel zur Bekämpfung parasitierender Insekten und Milben an Menschen
US6727228B2 (en) * 2001-04-25 2004-04-27 Johnson & Johnson Consumer Companies, Inc. Pediculicidal and ovacidal treatment compositions and methods for killing head lice and their eggs
DK1941798T3 (da) * 2004-12-17 2012-08-27 Devgen Nv Nematicide præparater
US8110608B2 (en) 2008-06-05 2012-02-07 Ecolab Usa Inc. Solid form sodium lauryl sulfate (SLS) pesticide composition
US9820977B2 (en) * 2008-10-03 2017-11-21 Bayer Healthcare Llc Systemic treatment of blood-sucking and blood-consuming parasites by oral administration of a parasiticidal agent
US8968757B2 (en) * 2010-10-12 2015-03-03 Ecolab Usa Inc. Highly wettable, water dispersible, granules including two pesticides
CA2989391C (en) 2014-06-24 2023-03-14 John O'halloran Fish feed compositions containing a neonicotinoid for preventing and treating parasite infections

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA689474A (en) * 1964-06-23 Clarence H. Gleason Nicotine pamoate
JPS60172976A (ja) * 1984-02-16 1985-09-06 Nippon Tokushu Noyaku Seizo Kk ニトロメチレン誘導体,その製法及び殺虫,殺ダニ,殺センチユウ剤
ZW5085A1 (en) * 1984-04-13 1985-09-18 Nihon Tokushu Noyaku Seizo Kk Nitromethylene derivatives,intermediates thereof,processes for production thereof,and insecticides
ATE67493T1 (de) * 1985-02-04 1991-10-15 Bayer Agrochem Kk Heterocyclische verbindungen.
JPH07121909B2 (ja) * 1986-09-10 1995-12-25 日本バイエルアグロケム株式会社 新規複素環式化合物及び殺虫剤
JP3023794B2 (ja) * 1989-05-17 2000-03-21 日本バイエルアグロケム株式会社 殺虫性ニトロ置換ヘテロ環式化合物
DE4232561A1 (de) * 1992-09-29 1994-03-31 Bayer Ag Bekämpfung von Fischparasiten

Also Published As

Publication number Publication date
EP0764022B1 (de) 2006-12-20
WO1995033453A1 (de) 1995-12-14
EP0764022A1 (de) 1997-03-26
CN1100537C (zh) 2003-02-05
AU2736495A (en) 1996-01-04
ATE348604T1 (de) 2007-01-15
KR100372348B1 (ko) 2003-05-12
CA2192093C (en) 2007-05-22
CN1149827A (zh) 1997-05-14
JP3978227B2 (ja) 2007-09-19
ES2279513T3 (es) 2007-08-16
JPH10500699A (ja) 1998-01-20
AU704092B2 (en) 1999-04-15
ZA954643B (en) 1996-01-26
DE59511073D1 (de) 2007-02-01
DE4419814A1 (de) 1995-12-14
BR9507926A (pt) 1997-11-11
CA2192093A1 (en) 1995-12-14
DK0764022T3 (da) 2007-04-10
US5712295A (en) 1998-01-27

Similar Documents

Publication Publication Date Title
DE69528823D1 (en) Morpholinwirkstoffvorläufer als tachykininreceptorantagonisten
IL122464A0 (en) N-heteroaryl-pyridinesulonamide derivatives and their use as endothelin antagonists
AU3642795A (en) Endothelin receptor antagonists for the treatment of emesis
AU4422293A (en) Substituted 2-amidotetralins as melatonin agonists and antagonists
LV11460A (lv) Estrogenu agonisti un antagonisti
ZA964383B (en) Hepatocyte growth factor receptor antagonists and uses thereof.
AU1228792A (en) Substituted pyridinones and pyrimidinones as angiotensin ii antagonists
IL128003A0 (en) Therapeutic multispecific compounds comprised of anti-fcalpha receptor antibodies
AU8374491A (en) Angiotensin II receptor antagonists
AU5873594A (en) Endothelin receptor antagonists
DK0877734T3 (da) Quinolin- og quinazolinforbindelser, der er egnede i terapi
DE69327720D1 (de) Endothelin rezeptor antagonisten
HU9600256D0 (en) Substituted diphenyl-sulfonamides, antagonists of endothelin
CY2242B1 (en) Benzonitriles and -fluorides as 5-ht agonists and antagonists
AU9064991A (en) Use of angiotensin ii receptor antagonists in the treatment of diabetic retinopathy
BR9406572A (pt) Antagonistas receptores do endotelin
MX9606179A (es) Agonistas y antagonistas de los receptores del acido acetilcolina nicotinico de insectos para el control de endoparasitos.
AU3629595A (en) Endothelin antagonists bearing pyridyl amides
AU9058591A (en) Use of angiotensin ii receptor antagonists in the treatment of diabetic nephropathy
ID19245A (id) Antagonis reseptor vitronektin, pembuatannya dan pemakaiannya
IS4803A (is) Oxa- og þía- díazól sveppaeitrunar viðtaka mótlyf
IL113050A0 (en) Antagonists of endothelin receptors
AU3745795A (en) Use of CCK-B receptor antagonists for the treatment of sleepdisorders
EP0714295A4 (es)
PL331882A1 (en) Substituted 1,2,3,4-tetrahydro-2-dibenzofurane amines and 2-amino cyclohepta[b]benzofuranes

Legal Events

Date Code Title Description
FG Grant or registration
GB Transfer or rights
PD Change of proprietorship

Owner name: BAYER ANIMAL HEALTH GMBH

MM Annulment or lapse due to non-payment of fees