AU5873594A - Endothelin receptor antagonists - Google Patents

Endothelin receptor antagonists

Info

Publication number
AU5873594A
AU5873594A AU58735/94A AU5873594A AU5873594A AU 5873594 A AU5873594 A AU 5873594A AU 58735/94 A AU58735/94 A AU 58735/94A AU 5873594 A AU5873594 A AU 5873594A AU 5873594 A AU5873594 A AU 5873594A
Authority
AU
Australia
Prior art keywords
receptor antagonists
endothelin receptor
endothelin
antagonists
receptor
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU58735/94A
Inventor
John Duncan Elliott
Jack Dale Leber
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of AU5873594A publication Critical patent/AU5873594A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
AU58735/94A 1992-12-22 1993-12-21 Endothelin receptor antagonists Abandoned AU5873594A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US99546692A 1992-12-22 1992-12-22
US995466 1992-12-22
PCT/US1993/012435 WO1994014434A1 (en) 1992-12-22 1993-12-21 Endothelin receptor antagonists

Publications (1)

Publication Number Publication Date
AU5873594A true AU5873594A (en) 1994-07-19

Family

ID=25541843

Family Applications (1)

Application Number Title Priority Date Filing Date
AU58735/94A Abandoned AU5873594A (en) 1992-12-22 1993-12-21 Endothelin receptor antagonists

Country Status (7)

Country Link
EP (1) EP0676959A4 (en)
JP (1) JPH08504826A (en)
CN (1) CN1096513A (en)
AU (1) AU5873594A (en)
MX (1) MX9400071A (en)
WO (1) WO1994014434A1 (en)
ZA (1) ZA939516B (en)

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DE60221391T2 (en) 2001-06-20 2008-04-17 Wyeth SUBSTITUTED INDOLESE DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1)
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CA2043741C (en) * 1990-06-07 2003-04-01 Kiyofumi Ishikawa Endothelin antagonistic peptide derivatives

Also Published As

Publication number Publication date
EP0676959A1 (en) 1995-10-18
ZA939516B (en) 1994-06-06
MX9400071A (en) 1994-07-29
JPH08504826A (en) 1996-05-28
EP0676959A4 (en) 1996-01-03
WO1994014434A1 (en) 1994-07-07
CN1096513A (en) 1994-12-21

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