JPH0798813B2 - １，５―ベンゾチアゼピン誘導体の製法 - Google Patents

１，５―ベンゾチアゼピン誘導体の製法

Info

Publication number
JPH0798813B2
JPH0798813B2 JP1109795A JP10979589A JPH0798813B2 JP H0798813 B2 JPH0798813 B2 JP H0798813B2 JP 1109795 A JP1109795 A JP 1109795A JP 10979589 A JP10979589 A JP 10979589A JP H0798813 B2 JPH0798813 B2 JP H0798813B2
Authority
JP
Japan
Prior art keywords
alkyl group
lower alkyl
compound
producing
iii
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP1109795A
Other languages
English (en)
Japanese (ja)
Other versions
JPH02286672A (ja
Inventor
宏徳 林
茂 西本
保 奥野
雅資 北野
貞夫 前田
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tanabe Seiyaku Co Ltd
Original Assignee
Tanabe Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co Ltd filed Critical Tanabe Seiyaku Co Ltd
Priority to JP1109795A priority Critical patent/JPH0798813B2/ja
Priority to ES90304299T priority patent/ES2106018T3/es
Priority to EP90304299A priority patent/EP0395323B1/de
Priority to DK90304299.2T priority patent/DK0395323T3/da
Priority to DE69030897T priority patent/DE69030897T2/de
Priority to SG1996001748A priority patent/SG47004A1/en
Priority to AT90304299T priority patent/ATE154348T1/de
Priority to FI902030A priority patent/FI109533B/fi
Priority to CA 2015182 priority patent/CA2015182C/en
Priority to IL94208A priority patent/IL94208A0/xx
Priority to AU53856/90A priority patent/AU616351B2/en
Priority to FR9005323A priority patent/FR2646424B1/fr
Priority to HU902607A priority patent/HU203882B/hu
Priority to CN90102552A priority patent/CN1031708C/zh
Priority to KR1019900006059A priority patent/KR970002466B1/ko
Publication of JPH02286672A publication Critical patent/JPH02286672A/ja
Priority to US07/722,497 priority patent/US5128469A/en
Priority to CN94120033A priority patent/CN1052479C/zh
Publication of JPH0798813B2 publication Critical patent/JPH0798813B2/ja
Priority to GR970401275T priority patent/GR3023767T3/el
Priority to HK98102939A priority patent/HK1003789A1/xx
Priority to CNB991017072A priority patent/CN1136205C/zh
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP1109795A 1989-04-28 1989-04-28 １，５―ベンゾチアゼピン誘導体の製法 Expired - Lifetime JPH0798813B2 (ja)

Priority Applications (20)

Application Number Priority Date Filing Date Title
JP1109795A JPH0798813B2 (ja) 1989-04-28 1989-04-28 １，５―ベンゾチアゼピン誘導体の製法
ES90304299T ES2106018T3 (es) 1989-04-28 1990-04-20 Procedimiento para la preparacion de derivados de 1,5-benzotiazepina.
EP90304299A EP0395323B1 (de) 1989-04-28 1990-04-20 Verfahren zur Herstellung von 1,5-Benzothiazepin-Derivaten
DK90304299.2T DK0395323T3 (da) 1989-04-28 1990-04-20 Fremgangsmåde til fremstilling af 1,5-benzothiazepinderivater
DE69030897T DE69030897T2 (de) 1989-04-28 1990-04-20 Verfahren zur Herstellung von 1,5-Benzothiazepin-Derivaten
SG1996001748A SG47004A1 (en) 1989-04-28 1990-04-20 Process for preparin 1 5-benzothiazepine derivatives
AT90304299T ATE154348T1 (de) 1989-04-28 1990-04-20 Verfahren zur herstellung von 1,5-benzothiazepin- derivaten
FI902030A FI109533B (fi) 1989-04-28 1990-04-23 Menetelmä 1,5-bentsotiatsepiinijohdannaisten valmistamiseksi
CA 2015182 CA2015182C (en) 1989-04-28 1990-04-23 Processes for preparing 1,5-benzothiazepine derivatives
IL94208A IL94208A0 (en) 1989-04-28 1990-04-25 Preparation of 1,5-benzothiazepine derivatives
FR9005323A FR2646424B1 (fr) 1989-04-28 1990-04-26 Procede de preparation de derives de la 1,5-benzothiazepine
AU53856/90A AU616351B2 (en) 1989-04-28 1990-04-26 Processes for preparing 1,5-benzothiazepine derivatives
HU902607A HU203882B (en) 1989-04-28 1990-04-27 New process for producing 1,5-benzothiazepine derivatives
CN90102552A CN1031708C (zh) 1989-04-28 1990-04-28 1,5－苯并硫氮杂䓬衍生物的制备方法
KR1019900006059A KR970002466B1 (ko) 1989-04-28 1990-04-28 1,5-벤조티아제핀 유도체의 제조방법
US07/722,497 US5128469A (en) 1989-04-28 1991-06-26 Process for preparing 1,5-benzothiazepine derivatives
CN94120033A CN1052479C (zh) 1989-04-28 1994-12-28 1,5苯并硫氮杂䓬衍生物的制备方法
GR970401275T GR3023767T3 (en) 1989-04-28 1997-06-12 Process for preparing 1,5-benzothiazepine derivatives
HK98102939A HK1003789A1 (en) 1989-04-28 1998-04-08 Process for preparing 1.5- benzothiazepine derivatives 1-5
CNB991017072A CN1136205C (zh) 1989-04-28 1999-01-28 1,5苯并硫氮杂�衍生物的制备方法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1109795A JPH0798813B2 (ja) 1989-04-28 1989-04-28 １，５―ベンゾチアゼピン誘導体の製法

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP6181894A Division JP2676720B2 (ja) 1994-03-31 1994-03-31 １，５−ベンゾチアゼピン誘導体の製法

Publications (2)

Publication Number Publication Date
JPH02286672A JPH02286672A (ja) 1990-11-26
JPH0798813B2 true JPH0798813B2 (ja) 1995-10-25

Family

ID=14519414

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1109795A Expired - Lifetime JPH0798813B2 (ja) 1989-04-28 1989-04-28 １，５―ベンゾチアゼピン誘導体の製法

Country Status (16)

Country Link
EP (1) EP0395323B1 (de)
JP (1) JPH0798813B2 (de)
KR (1) KR970002466B1 (de)
CN (3) CN1031708C (de)
AT (1) ATE154348T1 (de)
AU (1) AU616351B2 (de)
DE (1) DE69030897T2 (de)
DK (1) DK0395323T3 (de)
ES (1) ES2106018T3 (de)
FI (1) FI109533B (de)
FR (1) FR2646424B1 (de)
GR (1) GR3023767T3 (de)
HK (1) HK1003789A1 (de)
HU (1) HU203882B (de)
IL (1) IL94208A0 (de)
SG (1) SG47004A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2069003T3 (es) * 1989-04-28 1995-05-01 Tanabe Seiyaku Co Procedimiento para preparar derivados de 1,5-benzotiazepina.
IT1234387B (it) * 1989-07-12 1992-05-18 Zambon Spa Processo di purificazione di intermedi utili nella preparazione del diltiazem
ZA906810B (en) * 1989-08-31 1991-10-30 Marion Merrell Dow Inc Heterogeneous synthesis of azepinones from esters
JPH085869B2 (ja) * 1990-03-08 1996-01-24 田辺製薬株式会社 １，５−ベンゾチアゼピン誘導体の製法
IT1249318B (it) * 1991-05-23 1995-02-22 Zambon Spa Processo per la preparazione di benzotiazepine per ciclizzazione con acidi fosfonici
DE4206714A1 (de) * 1992-03-04 1993-09-09 Sandoz Ag Wachsdispersionen, deren herstellung und verwendung
NL1002687C2 (nl) * 1996-03-22 1997-09-23 Dsm Nv Werkwijze voor de bereiding van een benzothiazepine.
IL123352A0 (en) 1997-02-27 1998-09-24 Tanabe Seiyaku Co Process for preparing an optically active trans-3-substituted glycidic acid ester
IT1295376B1 (it) * 1997-10-22 1999-05-12 Zambon Spa Processo per il riciclo di un sottoprodotto della sintesi del diltiazem
CN116143723A (zh) * 2022-12-07 2023-05-23 海南锦瑞制药有限公司 一种盐酸地尔硫卓的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE31309T1 (de) * 1982-07-07 1987-12-15 Siegfried Ag Verfahren zur herstellung von 4-hydroxy-2-methyln-2-pyridyl-2h-1,2-benzothiazin-3-carboxamid 1,1- dioxid.
US4552695A (en) * 1983-04-21 1985-11-12 Shionogi & Co., Ltd. Process for production of diltiazem hydrochloride
ZA893392B (en) * 1988-05-24 1990-01-31 Hoffmann La Roche Process for the manufacture of optically active naphthothiazepinones
FR2641535B1 (fr) * 1989-01-11 1991-03-15 Synthelabo Procede de preparation de (+) - (2s, 3s)-hydroxy-3 (methoxy-4 phenyl)-2 dihydro-2,3 5h-benzothiazepine-1,5 one-4
ES2069003T3 (es) * 1989-04-28 1995-05-01 Tanabe Seiyaku Co Procedimiento para preparar derivados de 1,5-benzotiazepina.
JPH085869B2 (ja) * 1990-03-08 1996-01-24 田辺製薬株式会社 １，５−ベンゾチアゼピン誘導体の製法

Also Published As

Publication number Publication date
AU616351B2 (en) 1991-10-24
SG47004A1 (en) 1998-03-20
CN1110684A (zh) 1995-10-25
AU5385690A (en) 1990-11-01
JPH02286672A (ja) 1990-11-26
DE69030897D1 (de) 1997-07-17
HU203882B (en) 1991-10-28
DK0395323T3 (da) 1997-09-08
HU902607D0 (en) 1990-09-28
FR2646424A1 (fr) 1990-11-02
HUT55373A (en) 1991-05-28
ES2106018T3 (es) 1997-11-01
FI902030A0 (fi) 1990-04-23
EP0395323A1 (de) 1990-10-31
KR970002466B1 (ko) 1997-03-05
CN1245802A (zh) 2000-03-01
CN1046901A (zh) 1990-11-14
IL94208A0 (en) 1991-01-31
CN1136205C (zh) 2004-01-28
DE69030897T2 (de) 1997-09-25
GR3023767T3 (en) 1997-09-30
FR2646424B1 (fr) 1994-05-20
EP0395323B1 (de) 1997-06-11
KR900016171A (ko) 1990-11-12
CN1031708C (zh) 1996-05-01
FI109533B (fi) 2002-08-30
HK1003789A1 (en) 1998-11-06
CN1052479C (zh) 2000-05-17
ATE154348T1 (de) 1997-06-15

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