JPH0140837B2 - - Google Patents

Info

Publication number
JPH0140837B2
JPH0140837B2 JP55067685A JP6768580A JPH0140837B2 JP H0140837 B2 JPH0140837 B2 JP H0140837B2 JP 55067685 A JP55067685 A JP 55067685A JP 6768580 A JP6768580 A JP 6768580A JP H0140837 B2 JPH0140837 B2 JP H0140837B2
Authority
JP
Japan
Prior art keywords
acid
water
solution
mixture
ether
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP55067685A
Other languages
English (en)
Japanese (ja)
Other versions
JPS55154977A (en
Inventor
Fuon Daeene Berufu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Leo Pharma AS
Original Assignee
Leo Pharmaceutical Products Ltd AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharmaceutical Products Ltd AS filed Critical Leo Pharmaceutical Products Ltd AS
Publication of JPS55154977A publication Critical patent/JPS55154977A/ja
Publication of JPH0140837B2 publication Critical patent/JPH0140837B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP6768580A 1979-05-21 1980-05-20 Penicillanic acid derivative* its manufacture and use Granted JPS55154977A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB7917665 1979-05-21
GB7930819 1979-09-05
GB7941252 1979-11-29
GB8006681 1980-02-27

Publications (2)

Publication Number Publication Date
JPS55154977A JPS55154977A (en) 1980-12-02
JPH0140837B2 true JPH0140837B2 (en, 2012) 1989-08-31

Family

ID=27449123

Family Applications (1)

Application Number Title Priority Date Filing Date
JP6768580A Granted JPS55154977A (en) 1979-05-21 1980-05-20 Penicillanic acid derivative* its manufacture and use

Country Status (19)

Country Link
US (3) US4446144A (en, 2012)
JP (1) JPS55154977A (en, 2012)
AU (3) AU534754B2 (en, 2012)
BE (1) BE883390A (en, 2012)
CA (1) CA1265787A (en, 2012)
DE (3) DE3019244A1 (en, 2012)
DK (2) DK158669C (en, 2012)
FI (1) FI801618A7 (en, 2012)
FR (2) FR2457294A1 (en, 2012)
GR (1) GR68372B (en, 2012)
IE (2) IE49770B1 (en, 2012)
IL (1) IL59948A0 (en, 2012)
IT (1) IT1133091B (en, 2012)
LU (1) LU82468A1 (en, 2012)
NL (1) NL8002911A (en, 2012)
NZ (1) NZ193597A (en, 2012)
PH (2) PH17959A (en, 2012)
PT (1) PT71273A (en, 2012)
SE (3) SE452465B (en, 2012)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51846B1 (en) * 1980-11-17 1987-04-15 Leo Pharm Prod Ltd Pharmaceutical preparation for veterinary use and an appliance containing it
US4521533A (en) * 1984-07-12 1985-06-04 Pfizer Inc. Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics
GB8522156D0 (en) * 1985-09-06 1985-10-09 Leo Pharm Prod Ltd Producing chemical compounds
US5589354A (en) * 1994-12-20 1996-12-31 Biopure Corporation Halogenation of cephalexin with haloperoxidase from Rathayibacter biopuresis
US5695951A (en) * 1994-12-20 1997-12-09 Biopure Corporation Chlorination of cephalexin with chloroperoxidase from Rathayibacter biopuresis
PT971690E (pt) 1996-12-18 2002-12-31 Bimeda Res And Dev Ltd Composicao veterinaria intramamaria sem anti-infectantes
US20020035107A1 (en) * 2000-06-20 2002-03-21 Stefan Henke Highly concentrated stable meloxicam solutions
BRPI0315513B1 (pt) * 2002-10-25 2017-11-28 Intervet International B.V. Pharmaceutical composition preparation, and use of crystalline in a vehicle with prolonged release
EP1568369A1 (en) 2004-02-23 2005-08-31 Boehringer Ingelheim Vetmedica Gmbh Use of meloxicam for the treatment of respiratory diseases in pigs
DE102004025324A1 (de) * 2004-05-19 2005-12-08 Boehringer Ingelheim Vetmedica Gmbh Flüssige Zubereitung für die Veterinärmedizin, Verfahren zu deren Herstellung und deren Verwendung
HUE046427T2 (hu) * 2012-07-17 2020-03-30 Bayer New Zealand Ltd Injektálható antibiotikus készítmények és azok alkalmazása
EP2874623B1 (en) 2012-07-17 2018-12-12 Bayer New Zealand Limited Injectable antibiotic formulations and their methods of use
EP2934524B1 (en) * 2012-12-20 2019-03-27 Alleva Animal Health Limited Penethamate veterinary injectable formulations
EP4265241A1 (en) * 2022-04-20 2023-10-25 Bilim Ilac Sanayii Ve Ticaret A.S. Tablet formulations for the treatment of urinary system infections and method for the preparation of such formulations

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3206469A (en) * 1961-08-15 1965-09-14 Lepetit Spa 6-halopenicillanic acid
GB1297555A (en, 2012) * 1970-09-22 1972-11-22
GB1377817A (en) * 1971-06-09 1974-12-18 Beecham Group Ltd Penicillins and cephalosporins
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IN149747B (en, 2012) * 1977-06-07 1982-04-03 Pfizer
US4180506A (en) * 1978-01-18 1979-12-25 Rex Pratt 6β-Bromo penicillanic acid
CA1158639A (en) 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
US4203992A (en) * 1978-12-11 1980-05-20 E. R. Squibb & Sons, Inc. β-Bromopenicillanic acid sulfone
IL59081A0 (en) * 1979-01-10 1980-05-30 Schering Corp 2-penem compounds and a method for preparing them
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
US4397783A (en) 1979-03-05 1983-08-09 Pfizer Inc. Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
US4518530A (en) * 1979-03-05 1985-05-21 Pfizer Inc. 6-β-Substituted penicillanic acids as β-lactamase inhibitors
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
J. ORG. CHEM.=1978 *

Also Published As

Publication number Publication date
DK562589D0 (da) 1989-11-10
LU82468A1 (fr) 1980-12-16
FR2499575B1 (en, 2012) 1985-03-01
PT71273A (en) 1980-06-01
FR2457294B1 (en, 2012) 1984-01-13
NL8002911A (nl) 1980-11-25
IE49770B1 (en) 1985-12-11
SE8406201L (sv) 1984-12-06
GR68372B (en, 2012) 1981-12-28
AU1848683A (en) 1983-12-22
JPS55154977A (en) 1980-12-02
SE462097B (sv) 1990-05-07
AU5858480A (en) 1980-11-27
BE883390A (fr) 1980-11-20
DE3051038A1 (en, 2012) 1986-03-20
IE49768B1 (en) 1985-12-11
SE452465B (sv) 1987-11-30
IE800868L (en) 1980-11-21
DK158670B (da) 1990-07-02
AU541323B2 (en) 1985-01-03
DK218580A (da) 1980-11-22
DK158669B (da) 1990-07-02
FR2457294A1 (fr) 1980-12-19
DE3019244A1 (de) 1980-12-04
IL59948A0 (en) 1980-06-30
IE842559L (en) 1980-11-21
AU541322B2 (en) 1985-01-03
US4594246A (en) 1986-06-10
FI801618A7 (fi) 1981-01-01
DK158670C (da) 1991-01-07
SE462096B (sv) 1990-05-07
FR2499575A1 (fr) 1982-08-13
IT8067790A0 (it) 1980-05-20
CA1265787A (en) 1990-02-13
US4446144A (en) 1984-05-01
PH19005A (en) 1985-12-03
PH17959A (en) 1985-02-20
DE3019244C2 (en, 2012) 1989-04-06
SE8406201D0 (sv) 1984-12-06
SE8406202D0 (sv) 1984-12-06
NZ193597A (en) 1985-04-30
DE3051038C2 (en, 2012) 1989-04-13
DE3051037C2 (en, 2012) 1989-03-30
SE8003722L (sv) 1980-11-22
DK158669C (da) 1991-01-21
DK562589A (da) 1989-11-10
AU534754B2 (en) 1984-02-16
AU1848783A (en) 1983-12-22
SE8406202L (sv) 1984-12-06
IT1133091B (it) 1986-07-09
US4672114A (en) 1987-06-09

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