JPS6259709B2 - - Google Patents

Info

Publication number
JPS6259709B2
JPS6259709B2 JP55017197A JP1719780A JPS6259709B2 JP S6259709 B2 JPS6259709 B2 JP S6259709B2 JP 55017197 A JP55017197 A JP 55017197A JP 1719780 A JP1719780 A JP 1719780A JP S6259709 B2 JPS6259709 B2 JP S6259709B2
Authority
JP
Japan
Prior art keywords
formula
amino
acid
ester
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP55017197A
Other languages
English (en)
Japanese (ja)
Other versions
JPS55113790A (en
Inventor
Ore Gotsutofuretsudosen Bagun
Fuon Daeene Berufu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Leo Pharma AS
Original Assignee
Leo Pharmaceutical Products Ltd AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharmaceutical Products Ltd AS filed Critical Leo Pharmaceutical Products Ltd AS
Publication of JPS55113790A publication Critical patent/JPS55113790A/ja
Publication of JPS6259709B2 publication Critical patent/JPS6259709B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
JP1719780A 1979-02-13 1980-02-13 Novel penicillanic ester derivative and its manufacture and use Granted JPS55113790A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7905020 1979-02-13

Publications (2)

Publication Number Publication Date
JPS55113790A JPS55113790A (en) 1980-09-02
JPS6259709B2 true JPS6259709B2 (en, 2012) 1987-12-12

Family

ID=10503160

Family Applications (2)

Application Number Title Priority Date Filing Date
JP1719780A Granted JPS55113790A (en) 1979-02-13 1980-02-13 Novel penicillanic ester derivative and its manufacture and use
JP62114399A Granted JPS62281879A (ja) 1979-02-13 1987-05-11 β−ラクタム中間体およびその製法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP62114399A Granted JPS62281879A (ja) 1979-02-13 1987-05-11 β−ラクタム中間体およびその製法

Country Status (4)

Country Link
JP (2) JPS55113790A (en, 2012)
KR (1) KR830001903B1 (en, 2012)
BE (1) BE881675A (en, 2012)
ZA (1) ZA80796B (en, 2012)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4714761A (en) * 1979-03-05 1987-12-22 Pfizer Inc. 6,6-dihalopenicillanic acid 1,1-dioxides and process
US4420426A (en) 1979-03-05 1983-12-13 Pfizer Inc. 6-Alpha-halopenicillanic acid 1,1-dioxides
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4309347A (en) 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide
US4364957A (en) 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them
US4478748A (en) * 1981-02-20 1984-10-23 Pfizer Inc. Bis-esters of alkanediols
IN159362B (en, 2012) * 1981-03-23 1987-05-09 Pfizer
US4381263A (en) 1981-03-23 1983-04-26 Pfizer Inc. Process for the preparation of penicillanic acid esters
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
HU196412B (en) * 1981-03-23 1988-11-28 Pfizer Process for production of penicillin-acid-penicillakiroloximethil-esthers
JPS5857384A (ja) * 1981-09-09 1983-04-05 フアイザ−・インコ−ポレ−テツド 抗菌性のペニシラン酸６′‐（２‐アミノ‐２‐〔４‐アシルオキシフェニル〕アセタミド）ペニシラノイルオキシメチル１，１‐ジオキシド化合物
US4582829A (en) * 1981-09-09 1986-04-15 Pfizer Inc. Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
US4540687A (en) * 1981-09-09 1985-09-10 Pfizer Inc. Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
US4351840A (en) * 1981-09-18 1982-09-28 Pfizer Inc. Antibacterial esters of resorcinol with ampicillin and penicillanic acid 1,1-dioxide derivatives
US4359472A (en) * 1981-12-22 1982-11-16 Pfizer Inc. Bis-hydroxymethyl carbonate bridged antibacterial agents
US4444686A (en) * 1982-01-25 1984-04-24 Pfizer Inc. Crystalline penicillin ester intermediate
US4432987A (en) * 1982-04-23 1984-02-21 Pfizer Inc. Crystalline benzenesulfonate salts of sultamicillin
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
US4835674A (en) * 1986-07-28 1989-05-30 Bull Hn Information Systems Inc. Computer network system for multiple processing elements
KR20020028298A (ko) * 2000-10-09 2002-04-17 황해용 초배지 및 그 제조장치
DE102004021281A1 (de) * 2004-04-29 2005-11-24 Boehringer Ingelheim Vetmedica Gmbh Verwendung von Meloxicam-Formulierungen in der Veterinärmedizin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1578128A (en) * 1976-03-30 1980-11-05 Leo Pharm Prod Ltd Amidinopenicillanoyloxyalkyl amoxycillinates

Also Published As

Publication number Publication date
JPS55113790A (en) 1980-09-02
JPH0470315B2 (en, 2012) 1992-11-10
JPS62281879A (ja) 1987-12-07
BE881675A (fr) 1980-08-12
ZA80796B (en) 1981-02-25
KR830001903B1 (ko) 1983-09-19
KR830001947A (ko) 1983-05-21

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