JP7700399B1 - 単一の軸不斉化合物の選択的製造法 - Google Patents
単一の軸不斉化合物の選択的製造法 Download PDFInfo
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- JP7700399B1 JP7700399B1 JP2025523047A JP2025523047A JP7700399B1 JP 7700399 B1 JP7700399 B1 JP 7700399B1 JP 2025523047 A JP2025523047 A JP 2025523047A JP 2025523047 A JP2025523047 A JP 2025523047A JP 7700399 B1 JP7700399 B1 JP 7700399B1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/JP2023/032816 WO2025052649A1 (ja) | 2023-09-08 | 2023-09-08 | 単一の軸不斉化合物の選択的製造法 |
| JPPCT/JP2023/032816 | 2023-09-08 | ||
| PCT/JP2024/031959 WO2025053242A1 (ja) | 2023-09-08 | 2024-09-06 | 単一の軸不斉化合物の選択的製造法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2025053242A1 JPWO2025053242A1 (https=) | 2025-03-13 |
| JP7700399B1 true JP7700399B1 (ja) | 2025-06-30 |
| JPWO2025053242A5 JPWO2025053242A5 (https=) | 2025-08-13 |
Family
ID=94923286
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025523047A Active JP7700399B1 (ja) | 2023-09-08 | 2024-09-06 | 単一の軸不斉化合物の選択的製造法 |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP7700399B1 (https=) |
| CN (1) | CN121843933A (https=) |
| AU (1) | AU2024337896A1 (https=) |
| CO (1) | CO2026004110A2 (https=) |
| TW (1) | TW202527939A (https=) |
| WO (2) | WO2025052649A1 (https=) |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018143315A1 (ja) * | 2017-02-02 | 2018-08-09 | アステラス製薬株式会社 | キナゾリン化合物 |
| WO2022173032A1 (ja) * | 2021-02-15 | 2022-08-18 | アステラス製薬株式会社 | Ｇ１２ｄ変異ｋｒａｓタンパクの分解を誘導するためのキナゾリン化合物 |
| WO2022173033A1 (ja) * | 2021-02-15 | 2022-08-18 | アステラス製薬株式会社 | ４－アミノキナゾリン化合物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2023231912A1 (en) * | 2022-03-11 | 2024-08-15 | Astellas Pharma Inc. | Heterocyclic compound for inducing degradation of g12d mutant kras protein |
| TW202409002A (zh) * | 2022-07-21 | 2024-03-01 | 日商安斯泰來製藥股份有限公司 | 作用於g12d突變kras蛋白之雜環化合物 |
| CN119630656A (zh) * | 2022-08-05 | 2025-03-14 | 安斯泰来制药株式会社 | 用于诱导突变kras蛋白分解的杂环化合物 |
| WO2024034593A1 (ja) * | 2022-08-09 | 2024-02-15 | アステラス製薬株式会社 | Ｇ１２ｖ変異ｋｒａｓタンパクの分解を誘導するための複素環化合物 |
| TW202412790A (zh) * | 2022-08-09 | 2024-04-01 | 日商安斯泰來製藥股份有限公司 | 用於抑制及/或誘導分解kras蛋白之雜環化合物 |
-
2023
- 2023-09-08 WO PCT/JP2023/032816 patent/WO2025052649A1/ja active Pending
-
2024
- 2024-09-06 TW TW113133938A patent/TW202527939A/zh unknown
- 2024-09-06 WO PCT/JP2024/031959 patent/WO2025053242A1/ja active Pending
- 2024-09-06 AU AU2024337896A patent/AU2024337896A1/en active Pending
- 2024-09-06 CN CN202480055263.4A patent/CN121843933A/zh active Pending
- 2024-09-06 JP JP2025523047A patent/JP7700399B1/ja active Active
-
2026
- 2026-03-30 CO CONC2026/0004110A patent/CO2026004110A2/es unknown
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018143315A1 (ja) * | 2017-02-02 | 2018-08-09 | アステラス製薬株式会社 | キナゾリン化合物 |
| JP6587116B2 (ja) * | 2017-02-02 | 2019-10-09 | アステラス製薬株式会社 | キナゾリン化合物 |
| WO2022173032A1 (ja) * | 2021-02-15 | 2022-08-18 | アステラス製薬株式会社 | Ｇ１２ｄ変異ｋｒａｓタンパクの分解を誘導するためのキナゾリン化合物 |
| WO2022173033A1 (ja) * | 2021-02-15 | 2022-08-18 | アステラス製薬株式会社 | ４－アミノキナゾリン化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2025052649A1 (ja) | 2025-03-13 |
| AU2024337896A1 (en) | 2026-03-19 |
| WO2025053242A1 (ja) | 2025-03-13 |
| TW202527939A (zh) | 2025-07-16 |
| CN121843933A (zh) | 2026-04-10 |
| CO2026004110A2 (es) | 2026-04-16 |
| JPWO2025053242A1 (https=) | 2025-03-13 |
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